{"id":"https://openalex.org/W2133875871","doi":"https://doi.org/10.1109/cec.2012.6256578","title":"Differential evolution-binary particle swarm optimization algorithm for the analysis of aryl &amp;#x03B2;-diketo acids for HIV-1 integrase inhibition","display_name":"Differential evolution-binary particle swarm optimization algorithm for the analysis of aryl &amp;#x03B2;-diketo acids for HIV-1 integrase inhibition","publication_year":2012,"publication_date":"2012-06-01","ids":{"openalex":"https://openalex.org/W2133875871","doi":"https://doi.org/10.1109/cec.2012.6256578","mag":"2133875871"},"language":"en","primary_location":{"id":"doi:10.1109/cec.2012.6256578","is_oa":false,"landing_page_url":"https://doi.org/10.1109/cec.2012.6256578","pdf_url":null,"source":null,"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"2012 IEEE Congress on Evolutionary Computation","raw_type":"proceedings-article"},"type":"article","indexed_in":["crossref"],"open_access":{"is_oa":true,"oa_status":"green","oa_url":"https://zenodo.org/record/1266185","any_repository_has_fulltext":true},"authorships":[{"author_position":"first","author":{"id":"https://openalex.org/A5060263926","display_name":"Gene M. Ko","orcid":"https://orcid.org/0000-0003-1672-9202"},"institutions":[{"id":"https://openalex.org/I26538001","display_name":"San Diego State University","ror":"https://ror.org/0264fdx42","country_code":"US","type":"education","lineage":["https://openalex.org/I26538001"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"Gene M. Ko","raw_affiliation_strings":["Computational Science Research Center, San Diego State University, San Diego, CA, USA","Computational Science Research Center, San Diego State University, CA 92182-1245, USA"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Computational Science Research Center, San Diego State University, San Diego, CA, USA","institution_ids":["https://openalex.org/I26538001"]},{"raw_affiliation_string":"Computational Science Research Center, San Diego State University, CA 92182-1245, USA","institution_ids":["https://openalex.org/I26538001"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5101892558","display_name":"A. Srinivas Reddy","orcid":"https://orcid.org/0000-0003-4212-1460"},"institutions":[{"id":"https://openalex.org/I4210133661","display_name":"La Jolla Bioengineering Institute","ror":"https://ror.org/03sgbh608","country_code":"US","type":"nonprofit","lineage":["https://openalex.org/I4210133661"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"A. Srinivas Reddy","raw_affiliation_strings":["La Jolla Bioengineering Institute, San Diego, CA, USA","La Jolla Bioengineering Institute, San Diego, CA, 92121, USA"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"La Jolla Bioengineering Institute, San Diego, CA, USA","institution_ids":["https://openalex.org/I4210133661"]},{"raw_affiliation_string":"La Jolla Bioengineering Institute, San Diego, CA, 92121, USA","institution_ids":["https://openalex.org/I4210133661"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5110248651","display_name":"Sunil Kumar","orcid":null},"institutions":[{"id":"https://openalex.org/I26538001","display_name":"San Diego State University","ror":"https://ror.org/0264fdx42","country_code":"US","type":"education","lineage":["https://openalex.org/I26538001"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"Sunil Kumar","raw_affiliation_strings":["Department of Electrical and Computer Engineering, San Diego State University, San Diego, CA, USA","Department of Electrical and Computer Engineering, San Diego State University, CA 92182-1309, USA"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Department of Electrical and Computer Engineering, San Diego State University, San Diego, CA, USA","institution_ids":["https://openalex.org/I26538001"]},{"raw_affiliation_string":"Department of Electrical and Computer Engineering, San Diego State University, CA 92182-1309, USA","institution_ids":["https://openalex.org/I26538001"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5022652844","display_name":"Rajni Garg","orcid":"https://orcid.org/0000-0002-9629-8141"},"institutions":[{"id":"https://openalex.org/I26538001","display_name":"San Diego State University","ror":"https://ror.org/0264fdx42","country_code":"US","type":"education","lineage":["https://openalex.org/I26538001"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"Rajni Garg","raw_affiliation_strings":["Computational Science Research Center, San Diego State University, San Diego, CA, USA","Computational Science Research Center, San Diego State University, CA 92182-1245, USA"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Computational Science Research Center, San Diego State University, San Diego, CA, USA","institution_ids":["https://openalex.org/I26538001"]},{"raw_affiliation_string":"Computational Science Research Center, San Diego State University, CA 92182-1245, USA","institution_ids":["https://openalex.org/I26538001"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5112488675","display_name":"Barbara Bailey","orcid":null},"institutions":[{"id":"https://openalex.org/I26538001","display_name":"San Diego State University","ror":"https://ror.org/0264fdx42","country_code":"US","type":"education","lineage":["https://openalex.org/I26538001"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"Barbara A. Bailey","raw_affiliation_strings":["Department of Mathematics and Statistics, San Diego State University, San Diego, CA, USA","Department of Mathematics and Statistics, San Diego State University, CA 92182-7720, USA"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Department of Mathematics and Statistics, San Diego State University, San Diego, CA, USA","institution_ids":["https://openalex.org/I26538001"]},{"raw_affiliation_string":"Department of Mathematics and Statistics, San Diego State University, CA 92182-7720, USA","institution_ids":["https://openalex.org/I26538001"]}]},{"author_position":"last","author":{"id":"https://openalex.org/A5111510365","display_name":"Ahmad Hadaegh","orcid":null},"institutions":[{"id":"https://openalex.org/I226560621","display_name":"California State University, San Marcos","ror":"https://ror.org/01j8e0j24","country_code":"US","type":"education","lineage":["https://openalex.org/I226560621"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"Ahmad R. Hadaegh","raw_affiliation_strings":["Department of Computer Science and Information Systems, California State University San Marcos, San Marcos, CA, USA","Dept. of Computer Science and Information Systems, California State University San Marcos, 92096-0001, USA"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Department of Computer Science and Information Systems, California State University San Marcos, San Marcos, CA, USA","institution_ids":["https://openalex.org/I226560621"]},{"raw_affiliation_string":"Dept. of Computer Science and Information Systems, California State University San Marcos, 92096-0001, USA","institution_ids":["https://openalex.org/I226560621"]}]}],"institutions":[],"countries_distinct_count":1,"institutions_distinct_count":3,"corresponding_author_ids":[],"corresponding_institution_ids":[],"apc_list":null,"apc_paid":null,"fwci":0.6265,"has_fulltext":false,"cited_by_count":9,"citation_normalized_percentile":{"value":0.68207929,"is_in_top_1_percent":false,"is_in_top_10_percent":false},"cited_by_percentile_year":{"min":89,"max":98},"biblio":{"volume":null,"issue":null,"first_page":null,"last_page":null},"is_retracted":false,"is_paratext":false,"is_xpac":false,"primary_topic":{"id":"https://openalex.org/T10835","display_name":"Carbohydrate Chemistry and Synthesis","score":0.9939000010490417,"subfield":{"id":"https://openalex.org/subfields/1605","display_name":"Organic Chemistry"},"field":{"id":"https://openalex.org/fields/16","display_name":"Chemistry"},"domain":{"id":"https://openalex.org/domains/3","display_name":"Physical Sciences"}},"topics":[{"id":"https://openalex.org/T10835","display_name":"Carbohydrate Chemistry and Synthesis","score":0.9939000010490417,"subfield":{"id":"https://openalex.org/subfields/1605","display_name":"Organic Chemistry"},"field":{"id":"https://openalex.org/fields/16","display_name":"Chemistry"},"domain":{"id":"https://openalex.org/domains/3","display_name":"Physical Sciences"}},{"id":"https://openalex.org/T10526","display_name":"HIV/AIDS drug development and treatment","score":0.9919000267982483,"subfield":{"id":"https://openalex.org/subfields/2725","display_name":"Infectious Diseases"},"field":{"id":"https://openalex.org/fields/27","display_name":"Medicine"},"domain":{"id":"https://openalex.org/domains/4","display_name":"Health Sciences"}},{"id":"https://openalex.org/T10908","display_name":"Analytical Chemistry and Chromatography","score":0.9850000143051147,"subfield":{"id":"https://openalex.org/subfields/1607","display_name":"Spectroscopy"},"field":{"id":"https://openalex.org/fields/16","display_name":"Chemistry"},"domain":{"id":"https://openalex.org/domains/3","display_name":"Physical Sciences"}}],"keywords":[{"id":"https://openalex.org/keywords/quantitative-structure\u2013activity-relationship","display_name":"Quantitative structure\u2013activity relationship","score":0.693587064743042},{"id":"https://openalex.org/keywords/particle-swarm-optimization","display_name":"Particle swarm optimization","score":0.6195425391197205},{"id":"https://openalex.org/keywords/integrase","display_name":"Integrase","score":0.5744726061820984},{"id":"https://openalex.org/keywords/binary-number","display_name":"Binary number","score":0.5338023900985718},{"id":"https://openalex.org/keywords/algorithm","display_name":"Algorithm","score":0.5160967707633972},{"id":"https://openalex.org/keywords/computer-science","display_name":"Computer science","score":0.4028935432434082},{"id":"https://openalex.org/keywords/mathematics","display_name":"Mathematics","score":0.34454917907714844},{"id":"https://openalex.org/keywords/biological-system","display_name":"Biological system","score":0.328914999961853},{"id":"https://openalex.org/keywords/human-immunodeficiency-virus","display_name":"Human immunodeficiency virus (HIV)","score":0.24598848819732666},{"id":"https://openalex.org/keywords/biology","display_name":"Biology","score":0.1507091522216797},{"id":"https://openalex.org/keywords/machine-learning","display_name":"Machine learning","score":0.12786227464675903}],"concepts":[{"id":"https://openalex.org/C164126121","wikidata":"https://www.wikidata.org/wiki/Q766383","display_name":"Quantitative structure\u2013activity relationship","level":2,"score":0.693587064743042},{"id":"https://openalex.org/C85617194","wikidata":"https://www.wikidata.org/wiki/Q2072794","display_name":"Particle swarm optimization","level":2,"score":0.6195425391197205},{"id":"https://openalex.org/C14430832","wikidata":"https://www.wikidata.org/wiki/Q412550","display_name":"Integrase","level":3,"score":0.5744726061820984},{"id":"https://openalex.org/C48372109","wikidata":"https://www.wikidata.org/wiki/Q3913","display_name":"Binary number","level":2,"score":0.5338023900985718},{"id":"https://openalex.org/C11413529","wikidata":"https://www.wikidata.org/wiki/Q8366","display_name":"Algorithm","level":1,"score":0.5160967707633972},{"id":"https://openalex.org/C41008148","wikidata":"https://www.wikidata.org/wiki/Q21198","display_name":"Computer science","level":0,"score":0.4028935432434082},{"id":"https://openalex.org/C33923547","wikidata":"https://www.wikidata.org/wiki/Q395","display_name":"Mathematics","level":0,"score":0.34454917907714844},{"id":"https://openalex.org/C186060115","wikidata":"https://www.wikidata.org/wiki/Q30336093","display_name":"Biological system","level":1,"score":0.328914999961853},{"id":"https://openalex.org/C3013748606","wikidata":"https://www.wikidata.org/wiki/Q15787","display_name":"Human immunodeficiency virus (HIV)","level":2,"score":0.24598848819732666},{"id":"https://openalex.org/C86803240","wikidata":"https://www.wikidata.org/wiki/Q420","display_name":"Biology","level":0,"score":0.1507091522216797},{"id":"https://openalex.org/C119857082","wikidata":"https://www.wikidata.org/wiki/Q2539","display_name":"Machine learning","level":1,"score":0.12786227464675903},{"id":"https://openalex.org/C203014093","wikidata":"https://www.wikidata.org/wiki/Q101929","display_name":"Immunology","level":1,"score":0.0},{"id":"https://openalex.org/C94375191","wikidata":"https://www.wikidata.org/wiki/Q11205","display_name":"Arithmetic","level":1,"score":0.0}],"mesh":[],"locations_count":2,"locations":[{"id":"doi:10.1109/cec.2012.6256578","is_oa":false,"landing_page_url":"https://doi.org/10.1109/cec.2012.6256578","pdf_url":null,"source":null,"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"2012 IEEE Congress on Evolutionary Computation","raw_type":"proceedings-article"},{"id":"pmh:oai:zenodo.org:1266185","is_oa":true,"landing_page_url":"https://zenodo.org/record/1266185","pdf_url":null,"source":{"id":"https://openalex.org/S4306400562","display_name":"Zenodo (CERN European Organization for Nuclear Research)","issn_l":null,"issn":null,"is_oa":true,"is_in_doaj":false,"is_core":false,"host_organization":"https://openalex.org/I67311998","host_organization_name":"European Organization for Nuclear Research","host_organization_lineage":["https://openalex.org/I67311998"],"host_organization_lineage_names":[],"type":"repository"},"license":"public-domain","license_id":"https://openalex.org/licenses/public-domain","version":"submittedVersion","is_accepted":false,"is_published":false,"raw_source_name":"","raw_type":"info:eu-repo/semantics/conferencePaper"}],"best_oa_location":{"id":"pmh:oai:zenodo.org:1266185","is_oa":true,"landing_page_url":"https://zenodo.org/record/1266185","pdf_url":null,"source":{"id":"https://openalex.org/S4306400562","display_name":"Zenodo (CERN European Organization for Nuclear Research)","issn_l":null,"issn":null,"is_oa":true,"is_in_doaj":false,"is_core":false,"host_organization":"https://openalex.org/I67311998","host_organization_name":"European Organization for Nuclear Research","host_organization_lineage":["https://openalex.org/I67311998"],"host_organization_lineage_names":[],"type":"repository"},"license":"public-domain","license_id":"https://openalex.org/licenses/public-domain","version":"submittedVersion","is_accepted":false,"is_published":false,"raw_source_name":"","raw_type":"info:eu-repo/semantics/conferencePaper"},"sustainable_development_goals":[{"score":0.7799999713897705,"display_name":"Good health and well-being","id":"https://metadata.un.org/sdg/3"}],"awards":[],"funders":[],"has_content":{"grobid_xml":false,"pdf":false},"content_urls":null,"referenced_works_count":35,"referenced_works":["https://openalex.org/W127941512","https://openalex.org/W1483051834","https://openalex.org/W1496518737","https://openalex.org/W1595159159","https://openalex.org/W1991057723","https://openalex.org/W2000808481","https://openalex.org/W2004200900","https://openalex.org/W2004389946","https://openalex.org/W2009194688","https://openalex.org/W2017422910","https://openalex.org/W2025344323","https://openalex.org/W2031318909","https://openalex.org/W2037452557","https://openalex.org/W2039715647","https://openalex.org/W2042174016","https://openalex.org/W2047563128","https://openalex.org/W2049824131","https://openalex.org/W2055855178","https://openalex.org/W2056799414","https://openalex.org/W2068095506","https://openalex.org/W2074681440","https://openalex.org/W2079198822","https://openalex.org/W2088424609","https://openalex.org/W2099846405","https://openalex.org/W2124457330","https://openalex.org/W2140534639","https://openalex.org/W2147571602","https://openalex.org/W2152195021","https://openalex.org/W2161316542","https://openalex.org/W2163646378","https://openalex.org/W2236499470","https://openalex.org/W2950636979","https://openalex.org/W2999197824","https://openalex.org/W6629803284","https://openalex.org/W6674895100"],"related_works":["https://openalex.org/W2382340815","https://openalex.org/W1972650408","https://openalex.org/W2551736466","https://openalex.org/W2057222603","https://openalex.org/W2375449733","https://openalex.org/W1997566113","https://openalex.org/W3189652131","https://openalex.org/W60134212","https://openalex.org/W2908740012","https://openalex.org/W2253664354"],"abstract_inverted_index":{"A":[0],"hybrid":[1],"differential":[2],"evolution-binary":[3],"particle":[4,34],"swarm":[5,35],"optimization":[6],"(DE-BPSO)":[7],"algorithm":[8,15,81],"is":[9,26],"proposed":[10],"as":[11],"a":[12,38],"feature":[13],"selection":[14],"in":[16,124],"the":[17,30,33,46,50,75,92,100,108,117,121,126,133],"development":[18],"of":[19,32,40,49,94,102,110,116,129,135],"quantitative":[20],"structure-activity":[21],"relationship":[22],"(QSAR)":[23],"models.":[24],"DE":[25],"used":[27,43,63,84],"to":[28,44,64,73,85],"evolve":[29],"velocities":[31],"from":[36],"which":[37,53],"series":[39],"rules":[41],"are":[42,61],"determine":[45],"discrete":[47],"values":[48],"position":[51],"vectors":[52],"form":[54],"chemical":[55],"descriptor":[56,59],"subsets.":[57],"These":[58],"subsets":[60],"then":[62,83],"develop":[65,86],"models":[66,90],"for":[67,91,99,132],"QSAR":[68],"analysis.":[69],"DE-BPSO":[70,80],"was":[71,82],"found":[72],"outperform":[74],"standalone":[76],"BPSO":[77],"algorithm.":[78],"The":[79],"multiple":[87],"linear":[88],"regression":[89],"analysis":[93],"aryl":[95],"\u03b2-diketo":[96],"acid":[97],"compounds":[98,131],"inhibition":[101,134],"HIV-1":[103,136],"integrase.":[104,137],"This":[105],"model":[106],"highlights":[107],"significance":[109],"hydrophobicity":[111],"and":[112],"partial":[113],"positive":[114],"charges":[115],"hydrogen":[118],"atoms":[119],"on":[120],"molecular":[122],"surface":[123],"influencing":[125],"biological":[127],"activities":[128],"these":[130]},"counts_by_year":[{"year":2022,"cited_by_count":1},{"year":2021,"cited_by_count":3},{"year":2017,"cited_by_count":1},{"year":2015,"cited_by_count":4}],"updated_date":"2026-07-02T09:51:11.867554","created_date":"2016-06-24T00:00:00"}
