{"id":"https://openalex.org/W2081542153","doi":"https://doi.org/10.1016/j.neuroimage.2010.04.098","title":"Synthesis and evaluation of [C-11]LY2795050, an antagonist PET imaging tracer for the kappa opioid receptors","display_name":"Synthesis and evaluation of [C-11]LY2795050, an antagonist PET imaging tracer for the kappa opioid receptors","publication_year":2010,"publication_date":"2010-07-08","ids":{"openalex":"https://openalex.org/W2081542153","doi":"https://doi.org/10.1016/j.neuroimage.2010.04.098","mag":"2081542153"},"language":"en","primary_location":{"id":"doi:10.1016/j.neuroimage.2010.04.098","is_oa":false,"landing_page_url":"https://doi.org/10.1016/j.neuroimage.2010.04.098","pdf_url":null,"source":{"id":"https://openalex.org/S103225281","display_name":"NeuroImage","issn_l":"1053-8119","issn":["1053-8119","1095-9572"],"is_oa":false,"is_in_doaj":true,"is_core":true,"host_organization":"https://openalex.org/P4310320990","host_organization_name":"Elsevier BV","host_organization_lineage":["https://openalex.org/P4310320990"],"host_organization_lineage_names":["Elsevier BV"],"type":"journal"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"NeuroImage","raw_type":"journal-article"},"type":"article","indexed_in":["crossref","doaj"],"open_access":{"is_oa":false,"oa_status":"closed","oa_url":null,"any_repository_has_fulltext":false},"authorships":[{"author_position":"first","author":{"id":"https://openalex.org/A5111525497","display_name":"Ming\u2010Qiang Zheng","orcid":null},"institutions":[{"id":"https://openalex.org/I32971472","display_name":"Yale University","ror":"https://ror.org/03v76x132","country_code":"US","type":"education","lineage":["https://openalex.org/I32971472"]}],"countries":["US"],"is_corresponding":true,"raw_author_name":"Ming-Qiang Zheng","raw_affiliation_strings":["PET Center, Yale University School of Medicine, USA"],"affiliations":[{"raw_affiliation_string":"PET Center, Yale University School of Medicine, USA","institution_ids":["https://openalex.org/I32971472"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5006508700","display_name":"Nabeel Nabulsi","orcid":"https://orcid.org/0000-0001-8129-0051"},"institutions":[{"id":"https://openalex.org/I32971472","display_name":"Yale University","ror":"https://ror.org/03v76x132","country_code":"US","type":"education","lineage":["https://openalex.org/I32971472"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"Nabeel Nabulsi","raw_affiliation_strings":["PET Center, Yale University School of Medicine, USA"],"affiliations":[{"raw_affiliation_string":"PET Center, Yale University School of Medicine, USA","institution_ids":["https://openalex.org/I32971472"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5109929002","display_name":"Giampaolo Tomasi","orcid":null},"institutions":[{"id":"https://openalex.org/I32971472","display_name":"Yale University","ror":"https://ror.org/03v76x132","country_code":"US","type":"education","lineage":["https://openalex.org/I32971472"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"Giampaolo Tomasi","raw_affiliation_strings":["PET Center, Yale University School of Medicine, USA"],"affiliations":[{"raw_affiliation_string":"PET Center, Yale University School of Medicine, USA","institution_ids":["https://openalex.org/I32971472"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5110940748","display_name":"Charles H. Mitch","orcid":null},"institutions":[{"id":"https://openalex.org/I168537998","display_name":"Eli Lilly (United States)","ror":"https://ror.org/01qat3289","country_code":"US","type":"company","lineage":["https://openalex.org/I168537998"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"Charles Mitch","raw_affiliation_strings":["Eli LillyandCo., Indianapolis, IN, USA"],"affiliations":[{"raw_affiliation_string":"Eli LillyandCo., Indianapolis, IN, USA","institution_ids":["https://openalex.org/I168537998"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5110599345","display_name":"Steven J. Quimby","orcid":null},"institutions":[{"id":"https://openalex.org/I168537998","display_name":"Eli Lilly (United States)","ror":"https://ror.org/01qat3289","country_code":"US","type":"company","lineage":["https://openalex.org/I168537998"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"Steven Quimby","raw_affiliation_strings":["Eli LillyandCo., Indianapolis, IN, USA"],"affiliations":[{"raw_affiliation_string":"Eli LillyandCo., Indianapolis, IN, USA","institution_ids":["https://openalex.org/I168537998"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5016886412","display_name":"Vanessa Barth","orcid":null},"institutions":[{"id":"https://openalex.org/I168537998","display_name":"Eli Lilly (United States)","ror":"https://ror.org/01qat3289","country_code":"US","type":"company","lineage":["https://openalex.org/I168537998"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"Vanessa Barth","raw_affiliation_strings":["Eli LillyandCo., Indianapolis, IN, USA"],"affiliations":[{"raw_affiliation_string":"Eli LillyandCo., Indianapolis, IN, USA","institution_ids":["https://openalex.org/I168537998"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5037315198","display_name":"Karen Rash","orcid":null},"institutions":[{"id":"https://openalex.org/I168537998","display_name":"Eli Lilly (United States)","ror":"https://ror.org/01qat3289","country_code":"US","type":"company","lineage":["https://openalex.org/I168537998"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"Karen Rash","raw_affiliation_strings":["Eli LillyandCo., Indianapolis, IN, USA"],"affiliations":[{"raw_affiliation_string":"Eli LillyandCo., Indianapolis, IN, USA","institution_ids":["https://openalex.org/I168537998"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5074131055","display_name":"John J. Masters","orcid":null},"institutions":[{"id":"https://openalex.org/I168537998","display_name":"Eli Lilly (United States)","ror":"https://ror.org/01qat3289","country_code":"US","type":"company","lineage":["https://openalex.org/I168537998"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"John Masters","raw_affiliation_strings":["Eli LillyandCo., Indianapolis, IN, USA"],"affiliations":[{"raw_affiliation_string":"Eli LillyandCo., Indianapolis, IN, USA","institution_ids":["https://openalex.org/I168537998"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5085760951","display_name":"Antonio Navarro","orcid":"https://orcid.org/0000-0002-3623-0946"},"institutions":[{"id":"https://openalex.org/I168537998","display_name":"Eli Lilly (United States)","ror":"https://ror.org/01qat3289","country_code":"US","type":"company","lineage":["https://openalex.org/I168537998"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"Antonio Navarro","raw_affiliation_strings":["Eli LillyandCo., Indianapolis, IN, USA"],"affiliations":[{"raw_affiliation_string":"Eli LillyandCo., Indianapolis, IN, USA","institution_ids":["https://openalex.org/I168537998"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5014477543","display_name":"Eric P. Seest","orcid":null},"institutions":[{"id":"https://openalex.org/I168537998","display_name":"Eli Lilly (United States)","ror":"https://ror.org/01qat3289","country_code":"US","type":"company","lineage":["https://openalex.org/I168537998"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"Eric Seest","raw_affiliation_strings":["Eli LillyandCo., Indianapolis, IN, USA"],"affiliations":[{"raw_affiliation_string":"Eli LillyandCo., Indianapolis, IN, USA","institution_ids":["https://openalex.org/I168537998"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5012357230","display_name":"Richard E. Carson","orcid":"https://orcid.org/0000-0002-9338-7966"},"institutions":[{"id":"https://openalex.org/I32971472","display_name":"Yale University","ror":"https://ror.org/03v76x132","country_code":"US","type":"education","lineage":["https://openalex.org/I32971472"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"Richard E. Carson","raw_affiliation_strings":["PET Center, Yale University School of Medicine, USA"],"affiliations":[{"raw_affiliation_string":"PET Center, Yale University School of Medicine, USA","institution_ids":["https://openalex.org/I32971472"]}]},{"author_position":"last","author":{"id":"https://openalex.org/A5055576170","display_name":"Yiyun Huang","orcid":null},"institutions":[{"id":"https://openalex.org/I32971472","display_name":"Yale University","ror":"https://ror.org/03v76x132","country_code":"US","type":"education","lineage":["https://openalex.org/I32971472"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"Yiyun Huang","raw_affiliation_strings":["PET Center, Yale University School of Medicine, USA"],"affiliations":[{"raw_affiliation_string":"PET Center, Yale University School of Medicine, USA","institution_ids":["https://openalex.org/I32971472"]}]}],"institutions":[],"countries_distinct_count":1,"institutions_distinct_count":12,"corresponding_author_ids":["https://openalex.org/A5111525497"],"corresponding_institution_ids":["https://openalex.org/I32971472"],"apc_list":{"value":3450,"currency":"USD","value_usd":3450},"apc_paid":null,"fwci":0.2422,"has_fulltext":false,"cited_by_count":1,"citation_normalized_percentile":{"value":0.63515441,"is_in_top_1_percent":false,"is_in_top_10_percent":false},"cited_by_percentile_year":null,"biblio":{"volume":"52","issue":null,"first_page":"S120","last_page":"S120"},"is_retracted":false,"is_paratext":false,"is_xpac":false,"primary_topic":{"id":"https://openalex.org/T11395","display_name":"Radiopharmaceutical Chemistry and Applications","score":0.9868999719619751,"subfield":{"id":"https://openalex.org/subfields/2741","display_name":"Radiology, Nuclear Medicine and Imaging"},"field":{"id":"https://openalex.org/fields/27","display_name":"Medicine"},"domain":{"id":"https://openalex.org/domains/4","display_name":"Health Sciences"}},"topics":[{"id":"https://openalex.org/T11395","display_name":"Radiopharmaceutical Chemistry and Applications","score":0.9868999719619751,"subfield":{"id":"https://openalex.org/subfields/2741","display_name":"Radiology, Nuclear Medicine and Imaging"},"field":{"id":"https://openalex.org/fields/27","display_name":"Medicine"},"domain":{"id":"https://openalex.org/domains/4","display_name":"Health Sciences"}},{"id":"https://openalex.org/T10522","display_name":"Medical Imaging Techniques and Applications","score":0.980400025844574,"subfield":{"id":"https://openalex.org/subfields/2741","display_name":"Radiology, Nuclear Medicine and Imaging"},"field":{"id":"https://openalex.org/fields/27","display_name":"Medicine"},"domain":{"id":"https://openalex.org/domains/4","display_name":"Health Sciences"}},{"id":"https://openalex.org/T11752","display_name":"Cancer Treatment and Pharmacology","score":0.9577000141143799,"subfield":{"id":"https://openalex.org/subfields/2730","display_name":"Oncology"},"field":{"id":"https://openalex.org/fields/27","display_name":"Medicine"},"domain":{"id":"https://openalex.org/domains/4","display_name":"Health Sciences"}}],"keywords":[{"id":"https://openalex.org/keywords/\u03ba-opioid-receptor","display_name":"\u03ba-opioid receptor","score":0.735725998878479},{"id":"https://openalex.org/keywords/kappa","display_name":"Kappa","score":0.7082279324531555},{"id":"https://openalex.org/keywords/opioid","display_name":"Opioid","score":0.5449683666229248},{"id":"https://openalex.org/keywords/antagonist","display_name":"Antagonist","score":0.5193208456039429},{"id":"https://openalex.org/keywords/tracer","display_name":"TRACER","score":0.47139909863471985},{"id":"https://openalex.org/keywords/pet-imaging","display_name":"Pet imaging","score":0.45944488048553467},{"id":"https://openalex.org/keywords/chemistry","display_name":"Chemistry","score":0.3803367614746094},{"id":"https://openalex.org/keywords/pharmacology","display_name":"Pharmacology","score":0.3714636564254761},{"id":"https://openalex.org/keywords/nuclear-medicine","display_name":"Nuclear medicine","score":0.3540774881839752},{"id":"https://openalex.org/keywords/receptor","display_name":"Receptor","score":0.3499756455421448},{"id":"https://openalex.org/keywords/medicine","display_name":"Medicine","score":0.3204374313354492},{"id":"https://openalex.org/keywords/positron-emission-tomography","display_name":"Positron emission tomography","score":0.269208699464798},{"id":"https://openalex.org/keywords/internal-medicine","display_name":"Internal medicine","score":0.2607918977737427},{"id":"https://openalex.org/keywords/physics","display_name":"Physics","score":0.18434211611747742},{"id":"https://openalex.org/keywords/mathematics","display_name":"Mathematics","score":0.1743365228176117},{"id":"https://openalex.org/keywords/nuclear-physics","display_name":"Nuclear physics","score":0.07102757692337036}],"concepts":[{"id":"https://openalex.org/C184389661","wikidata":"https://www.wikidata.org/wiki/Q14897645","display_name":"\u03ba-opioid receptor","level":4,"score":0.735725998878479},{"id":"https://openalex.org/C2778724333","wikidata":"https://www.wikidata.org/wiki/Q14401","display_name":"Kappa","level":2,"score":0.7082279324531555},{"id":"https://openalex.org/C2781063702","wikidata":"https://www.wikidata.org/wiki/Q427523","display_name":"Opioid","level":3,"score":0.5449683666229248},{"id":"https://openalex.org/C2776885963","wikidata":"https://www.wikidata.org/wiki/Q245204","display_name":"Antagonist","level":3,"score":0.5193208456039429},{"id":"https://openalex.org/C2778863792","wikidata":"https://www.wikidata.org/wiki/Q16909918","display_name":"TRACER","level":2,"score":0.47139909863471985},{"id":"https://openalex.org/C3017724952","wikidata":"https://www.wikidata.org/wiki/Q208376","display_name":"Pet imaging","level":3,"score":0.45944488048553467},{"id":"https://openalex.org/C185592680","wikidata":"https://www.wikidata.org/wiki/Q2329","display_name":"Chemistry","level":0,"score":0.3803367614746094},{"id":"https://openalex.org/C98274493","wikidata":"https://www.wikidata.org/wiki/Q128406","display_name":"Pharmacology","level":1,"score":0.3714636564254761},{"id":"https://openalex.org/C2989005","wikidata":"https://www.wikidata.org/wiki/Q214963","display_name":"Nuclear medicine","level":1,"score":0.3540774881839752},{"id":"https://openalex.org/C170493617","wikidata":"https://www.wikidata.org/wiki/Q208467","display_name":"Receptor","level":2,"score":0.3499756455421448},{"id":"https://openalex.org/C71924100","wikidata":"https://www.wikidata.org/wiki/Q11190","display_name":"Medicine","level":0,"score":0.3204374313354492},{"id":"https://openalex.org/C2775842073","wikidata":"https://www.wikidata.org/wiki/Q208376","display_name":"Positron emission tomography","level":2,"score":0.269208699464798},{"id":"https://openalex.org/C126322002","wikidata":"https://www.wikidata.org/wiki/Q11180","display_name":"Internal medicine","level":1,"score":0.2607918977737427},{"id":"https://openalex.org/C121332964","wikidata":"https://www.wikidata.org/wiki/Q413","display_name":"Physics","level":0,"score":0.18434211611747742},{"id":"https://openalex.org/C33923547","wikidata":"https://www.wikidata.org/wiki/Q395","display_name":"Mathematics","level":0,"score":0.1743365228176117},{"id":"https://openalex.org/C185544564","wikidata":"https://www.wikidata.org/wiki/Q81197","display_name":"Nuclear physics","level":1,"score":0.07102757692337036},{"id":"https://openalex.org/C2524010","wikidata":"https://www.wikidata.org/wiki/Q8087","display_name":"Geometry","level":1,"score":0.0}],"mesh":[],"locations_count":1,"locations":[{"id":"doi:10.1016/j.neuroimage.2010.04.098","is_oa":false,"landing_page_url":"https://doi.org/10.1016/j.neuroimage.2010.04.098","pdf_url":null,"source":{"id":"https://openalex.org/S103225281","display_name":"NeuroImage","issn_l":"1053-8119","issn":["1053-8119","1095-9572"],"is_oa":false,"is_in_doaj":true,"is_core":true,"host_organization":"https://openalex.org/P4310320990","host_organization_name":"Elsevier BV","host_organization_lineage":["https://openalex.org/P4310320990"],"host_organization_lineage_names":["Elsevier BV"],"type":"journal"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"NeuroImage","raw_type":"journal-article"}],"best_oa_location":null,"sustainable_development_goals":[],"awards":[],"funders":[],"has_content":{"grobid_xml":false,"pdf":false},"content_urls":null,"referenced_works_count":0,"referenced_works":[],"related_works":["https://openalex.org/W2271903968","https://openalex.org/W51698146","https://openalex.org/W2981845044","https://openalex.org/W1972127446","https://openalex.org/W2017232769","https://openalex.org/W1997771816","https://openalex.org/W2014127416","https://openalex.org/W2078627033","https://openalex.org/W3121095357","https://openalex.org/W4247267163"],"abstract_inverted_index":null,"counts_by_year":[],"updated_date":"2025-11-06T03:46:38.306776","created_date":"2025-10-10T00:00:00"}
