{"id":"https://openalex.org/W3006261578","doi":"https://doi.org/10.1007/978-3-030-41032-2_40","title":"Large-Scale Prediction of the ARS Family Inhibitors of the Oncogenic KRASG12C Mutant","display_name":"Large-Scale Prediction of the ARS Family Inhibitors of the Oncogenic KRASG12C Mutant","publication_year":2020,"publication_date":"2020-01-01","ids":{"openalex":"https://openalex.org/W3006261578","doi":"https://doi.org/10.1007/978-3-030-41032-2_40","mag":"3006261578"},"language":"en","primary_location":{"id":"doi:10.1007/978-3-030-41032-2_40","is_oa":false,"landing_page_url":"https://doi.org/10.1007/978-3-030-41032-2_40","pdf_url":null,"source":{"id":"https://openalex.org/S106296714","display_name":"Lecture notes in computer science","issn_l":"0302-9743","issn":["0302-9743","1611-3349"],"is_oa":false,"is_in_doaj":false,"is_core":true,"host_organization":"https://openalex.org/P4310319900","host_organization_name":"Springer Science+Business Media","host_organization_lineage":["https://openalex.org/P4310319900","https://openalex.org/P4310319965"],"host_organization_lineage_names":["Springer Science+Business Media","Springer Nature"],"type":"book series"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"Lecture Notes in Computer Science","raw_type":"book-chapter"},"type":"book-chapter","indexed_in":["crossref"],"open_access":{"is_oa":false,"oa_status":"closed","oa_url":null,"any_repository_has_fulltext":false},"authorships":[{"author_position":"first","author":{"id":"https://openalex.org/A5037138522","display_name":"A. M. Kulakova","orcid":"https://orcid.org/0000-0002-9732-0996"},"institutions":[{"id":"https://openalex.org/I19880235","display_name":"Lomonosov Moscow State University","ror":"https://ror.org/010pmpe69","country_code":"RU","type":"education","lineage":["https://openalex.org/I19880235"]}],"countries":["RU"],"is_corresponding":true,"raw_author_name":"Anna M. Kulakova","raw_affiliation_strings":["Department of Chemistry, Lomonosov Moscow State University, Moscow, 119991, Russia"],"raw_orcid":"https://orcid.org/0000-0002-9732-0996","affiliations":[{"raw_affiliation_string":"Department of Chemistry, Lomonosov Moscow State University, Moscow, 119991, Russia","institution_ids":["https://openalex.org/I19880235"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5053941657","display_name":"\u0410. V. Popinako","orcid":"https://orcid.org/0000-0002-5179-4627"},"institutions":[{"id":"https://openalex.org/I1313323035","display_name":"Russian Academy of Sciences","ror":"https://ror.org/05qrfxd25","country_code":"RU","type":"government","lineage":["https://openalex.org/I1313323035"]},{"id":"https://openalex.org/I4210144344","display_name":"Federal Research Centre \u00abFundamentals of Biotechnology\u00bb of the Russian Academy of Sciences","ror":"https://ror.org/045sc8e83","country_code":"RU","type":"facility","lineage":["https://openalex.org/I1313323035","https://openalex.org/I4210129690","https://openalex.org/I4210144344"]}],"countries":["RU"],"is_corresponding":false,"raw_author_name":"Anna V. Popinako","raw_affiliation_strings":["Bach Institute of Biochemistry, Federeal Research Center \u201cFundamentals of Biotechnology\u201d of the Russian Academy of Sciences, Moscow, 119071, Russia","Bach Institute of Biochemistry, Federeal Research Center \"Fundamentals of Biotechnology\" of the Russian Academy of Sciences, Moscow, 119071, Russia"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Bach Institute of Biochemistry, Federeal Research Center \u201cFundamentals of Biotechnology\u201d of the Russian Academy of Sciences, Moscow, 119071, Russia","institution_ids":["https://openalex.org/I4210144344","https://openalex.org/I1313323035"]},{"raw_affiliation_string":"Bach Institute of Biochemistry, Federeal Research Center \"Fundamentals of Biotechnology\" of the Russian Academy of Sciences, Moscow, 119071, Russia","institution_ids":["https://openalex.org/I4210144344","https://openalex.org/I1313323035"]}]},{"author_position":"last","author":{"id":"https://openalex.org/A5034349557","display_name":"Maria G. Khrenova","orcid":"https://orcid.org/0000-0001-7117-3089"},"institutions":[{"id":"https://openalex.org/I1313323035","display_name":"Russian Academy of Sciences","ror":"https://ror.org/05qrfxd25","country_code":"RU","type":"government","lineage":["https://openalex.org/I1313323035"]},{"id":"https://openalex.org/I19880235","display_name":"Lomonosov Moscow State University","ror":"https://ror.org/010pmpe69","country_code":"RU","type":"education","lineage":["https://openalex.org/I19880235"]},{"id":"https://openalex.org/I4210144344","display_name":"Federal Research Centre \u00abFundamentals of Biotechnology\u00bb of the Russian Academy of Sciences","ror":"https://ror.org/045sc8e83","country_code":"RU","type":"facility","lineage":["https://openalex.org/I1313323035","https://openalex.org/I4210129690","https://openalex.org/I4210144344"]}],"countries":["RU"],"is_corresponding":false,"raw_author_name":"Maria G. Khrenova","raw_affiliation_strings":["Bach Institute of Biochemistry, Federeal Research Center \u201cFundamentals of Biotechnology\u201d of the Russian Academy of Sciences, Moscow, 119071, Russia","Department of Chemistry, Lomonosov Moscow State University, Moscow, 119991, Russia","Bach Institute of Biochemistry, Federeal Research Center \"Fundamentals of Biotechnology\" of the Russian Academy of Sciences, Moscow, 119071, Russia"],"raw_orcid":"https://orcid.org/0000-0001-7117-3089","affiliations":[{"raw_affiliation_string":"Bach Institute of Biochemistry, Federeal Research Center \u201cFundamentals of Biotechnology\u201d of the Russian Academy of Sciences, Moscow, 119071, Russia","institution_ids":["https://openalex.org/I4210144344","https://openalex.org/I1313323035"]},{"raw_affiliation_string":"Department of Chemistry, Lomonosov Moscow State University, Moscow, 119991, Russia","institution_ids":["https://openalex.org/I19880235"]},{"raw_affiliation_string":"Bach Institute of Biochemistry, Federeal Research Center \"Fundamentals of Biotechnology\" of the Russian Academy of Sciences, Moscow, 119071, Russia","institution_ids":["https://openalex.org/I4210144344","https://openalex.org/I1313323035"]}]}],"institutions":[],"countries_distinct_count":1,"institutions_distinct_count":3,"corresponding_author_ids":["https://openalex.org/A5037138522"],"corresponding_institution_ids":["https://openalex.org/I19880235"],"apc_list":{"value":5000,"currency":"EUR","value_usd":5392},"apc_paid":null,"fwci":0.0,"has_fulltext":false,"cited_by_count":0,"citation_normalized_percentile":{"value":0.03161714,"is_in_top_1_percent":false,"is_in_top_10_percent":false},"cited_by_percentile_year":null,"biblio":{"volume":null,"issue":null,"first_page":"348","last_page":"355"},"is_retracted":false,"is_paratext":false,"is_xpac":false,"primary_topic":{"id":"https://openalex.org/T10169","display_name":"Protein Kinase Regulation and GTPase Signaling","score":0.9994999766349792,"subfield":{"id":"https://openalex.org/subfields/1312","display_name":"Molecular Biology"},"field":{"id":"https://openalex.org/fields/13","display_name":"Biochemistry, Genetics and Molecular Biology"},"domain":{"id":"https://openalex.org/domains/1","display_name":"Life Sciences"}},"topics":[{"id":"https://openalex.org/T10169","display_name":"Protein Kinase Regulation and GTPase Signaling","score":0.9994999766349792,"subfield":{"id":"https://openalex.org/subfields/1312","display_name":"Molecular Biology"},"field":{"id":"https://openalex.org/fields/13","display_name":"Biochemistry, Genetics and Molecular Biology"},"domain":{"id":"https://openalex.org/domains/1","display_name":"Life Sciences"}},{"id":"https://openalex.org/T11162","display_name":"Enzyme Structure and Function","score":0.9983000159263611,"subfield":{"id":"https://openalex.org/subfields/2505","display_name":"Materials Chemistry"},"field":{"id":"https://openalex.org/fields/25","display_name":"Materials Science"},"domain":{"id":"https://openalex.org/domains/3","display_name":"Physical Sciences"}},{"id":"https://openalex.org/T12827","display_name":"Biochemical and Molecular Research","score":0.9937999844551086,"subfield":{"id":"https://openalex.org/subfields/1312","display_name":"Molecular Biology"},"field":{"id":"https://openalex.org/fields/13","display_name":"Biochemistry, Genetics and Molecular Biology"},"domain":{"id":"https://openalex.org/domains/1","display_name":"Life Sciences"}}],"keywords":[{"id":"https://openalex.org/keywords/kras","display_name":"KRAS","score":0.8498842120170593},{"id":"https://openalex.org/keywords/dissociation-constant","display_name":"Dissociation constant","score":0.5483366847038269},{"id":"https://openalex.org/keywords/point-mutation","display_name":"Point mutation","score":0.5290687680244446},{"id":"https://openalex.org/keywords/mutant","display_name":"Mutant","score":0.49619728326797485},{"id":"https://openalex.org/keywords/gtp","display_name":"GTP'","score":0.48104050755500793},{"id":"https://openalex.org/keywords/cancer-research","display_name":"Cancer research","score":0.4229428768157959},{"id":"https://openalex.org/keywords/computer-science","display_name":"Computer science","score":0.4074982702732086},{"id":"https://openalex.org/keywords/mutation","display_name":"Mutation","score":0.356650173664093},{"id":"https://openalex.org/keywords/chemistry","display_name":"Chemistry","score":0.35525548458099365},{"id":"https://openalex.org/keywords/computational-biology","display_name":"Computational biology","score":0.34541356563568115},{"id":"https://openalex.org/keywords/biology","display_name":"Biology","score":0.29960188269615173},{"id":"https://openalex.org/keywords/enzyme","display_name":"Enzyme","score":0.2276061475276947},{"id":"https://openalex.org/keywords/biochemistry","display_name":"Biochemistry","score":0.17616471648216248},{"id":"https://openalex.org/keywords/receptor","display_name":"Receptor","score":0.14083632826805115},{"id":"https://openalex.org/keywords/gene","display_name":"Gene","score":0.09439045190811157}],"concepts":[{"id":"https://openalex.org/C2781187634","wikidata":"https://www.wikidata.org/wiki/Q20969980","display_name":"KRAS","level":4,"score":0.8498842120170593},{"id":"https://openalex.org/C74998103","wikidata":"https://www.wikidata.org/wiki/Q898254","display_name":"Dissociation constant","level":3,"score":0.5483366847038269},{"id":"https://openalex.org/C176944494","wikidata":"https://www.wikidata.org/wiki/Q1415380","display_name":"Point mutation","level":4,"score":0.5290687680244446},{"id":"https://openalex.org/C143065580","wikidata":"https://www.wikidata.org/wiki/Q3285695","display_name":"Mutant","level":3,"score":0.49619728326797485},{"id":"https://openalex.org/C118716","wikidata":"https://www.wikidata.org/wiki/Q5514725","display_name":"GTP'","level":3,"score":0.48104050755500793},{"id":"https://openalex.org/C502942594","wikidata":"https://www.wikidata.org/wiki/Q3421914","display_name":"Cancer research","level":1,"score":0.4229428768157959},{"id":"https://openalex.org/C41008148","wikidata":"https://www.wikidata.org/wiki/Q21198","display_name":"Computer science","level":0,"score":0.4074982702732086},{"id":"https://openalex.org/C501734568","wikidata":"https://www.wikidata.org/wiki/Q42918","display_name":"Mutation","level":3,"score":0.356650173664093},{"id":"https://openalex.org/C185592680","wikidata":"https://www.wikidata.org/wiki/Q2329","display_name":"Chemistry","level":0,"score":0.35525548458099365},{"id":"https://openalex.org/C70721500","wikidata":"https://www.wikidata.org/wiki/Q177005","display_name":"Computational biology","level":1,"score":0.34541356563568115},{"id":"https://openalex.org/C86803240","wikidata":"https://www.wikidata.org/wiki/Q420","display_name":"Biology","level":0,"score":0.29960188269615173},{"id":"https://openalex.org/C181199279","wikidata":"https://www.wikidata.org/wiki/Q8047","display_name":"Enzyme","level":2,"score":0.2276061475276947},{"id":"https://openalex.org/C55493867","wikidata":"https://www.wikidata.org/wiki/Q7094","display_name":"Biochemistry","level":1,"score":0.17616471648216248},{"id":"https://openalex.org/C170493617","wikidata":"https://www.wikidata.org/wiki/Q208467","display_name":"Receptor","level":2,"score":0.14083632826805115},{"id":"https://openalex.org/C104317684","wikidata":"https://www.wikidata.org/wiki/Q7187","display_name":"Gene","level":2,"score":0.09439045190811157}],"mesh":[],"locations_count":1,"locations":[{"id":"doi:10.1007/978-3-030-41032-2_40","is_oa":false,"landing_page_url":"https://doi.org/10.1007/978-3-030-41032-2_40","pdf_url":null,"source":{"id":"https://openalex.org/S106296714","display_name":"Lecture notes in computer science","issn_l":"0302-9743","issn":["0302-9743","1611-3349"],"is_oa":false,"is_in_doaj":false,"is_core":true,"host_organization":"https://openalex.org/P4310319900","host_organization_name":"Springer Science+Business Media","host_organization_lineage":["https://openalex.org/P4310319900","https://openalex.org/P4310319965"],"host_organization_lineage_names":["Springer Science+Business Media","Springer Nature"],"type":"book series"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"Lecture Notes in Computer Science","raw_type":"book-chapter"}],"best_oa_location":null,"sustainable_development_goals":[],"awards":[],"funders":[],"has_content":{"pdf":false,"grobid_xml":false},"content_urls":null,"referenced_works_count":11,"referenced_works":["https://openalex.org/W1833275968","https://openalex.org/W1977598234","https://openalex.org/W2004774286","https://openalex.org/W2018299967","https://openalex.org/W2067711179","https://openalex.org/W2081990599","https://openalex.org/W2105668062","https://openalex.org/W2128339707","https://openalex.org/W2233032895","https://openalex.org/W2300615341","https://openalex.org/W2612770567"],"related_works":["https://openalex.org/W3030972949","https://openalex.org/W2027505083","https://openalex.org/W2550943714","https://openalex.org/W3212350425","https://openalex.org/W2388007221","https://openalex.org/W2511508046","https://openalex.org/W2363458739","https://openalex.org/W2028961943","https://openalex.org/W2375287167","https://openalex.org/W1994083192"],"abstract_inverted_index":null,"counts_by_year":[],"updated_date":"2025-11-06T03:46:38.306776","created_date":"2025-10-10T00:00:00"}
