{"id":"https://openalex.org/W4361908315","doi":"https://doi.org/10.1158/1078-0432.22449923","title":"Supplementary Methods from Cellular Uptake of Imatinib into Leukemic Cells Is Independent of Human Organic Cation Transporter 1 (OCT1)","display_name":"Supplementary Methods from Cellular Uptake of Imatinib into Leukemic Cells Is Independent of Human Organic Cation Transporter 1 (OCT1)","publication_year":2023,"publication_date":"2023-03-31","ids":{"openalex":"https://openalex.org/W4361908315","doi":"https://doi.org/10.1158/1078-0432.22449923"},"language":"en","primary_location":{"id":"doi:10.1158/1078-0432.22449923","doi":"https://doi.org/10.1158/1078-0432.22449923","is_oa":true,"landing_page_url":"http://dx.doi.org/10.1158/1078-0432.22449923","pdf_url":"https://aacr.figshare.com/articles/journal_contribution/Supplementary_Methods_from_Cellular_Uptake_of_Imatinib_into_Leukemic_Cells_Is_Independent_of_Human_Organic_Cation_Transporter_1_OCT1_/22449923/1/files/39900983.pdf","source":null,"license":"cc-by","license_id":"https://openalex.org/licenses/cc-by","version":"acceptedVersion","is_accepted":true,"is_published":false,"raw_source_name":"American Association for Cancer Research","raw_type":"posted-content"},"volume":null,"type":"supplementary-materials","indexed_in":["crossref"],"open_access":{"is_oa":true,"oa_status":"gold","oa_url":"https://aacr.figshare.com/articles/journal_contribution/Supplementary_Methods_from_Cellular_Uptake_of_Imatinib_into_Leukemic_Cells_Is_Independent_of_Human_Organic_Cation_Transporter_1_OCT1_/22449923/1/files/39900983.pdf","any_repository_has_fulltext":true},"authorships":[{"author_position":"first","author":{"id":"https://openalex.org/A5065181138","display_name":"Anne T. Nies","orcid":"https://orcid.org/0000-0001-6862-0730","observed_orcids":["https://orcid.org/0000-0001-6862-0730"]},"institutions":[],"countries":[],"is_corresponding":false,"raw_author_name":"Anne T. Nies","raw_affiliation_strings":[],"raw_orcid":null,"affiliations":[]},{"author_position":"middle","author":{"id":"https://openalex.org/A5066057635","display_name":"Elke Schaeffeler","orcid":"https://orcid.org/0009-0005-2997-0355","observed_orcids":["https://orcid.org/0009-0005-2997-0355"]},"institutions":[],"countries":[],"is_corresponding":false,"raw_author_name":"Elke Schaeffeler","raw_affiliation_strings":[],"raw_orcid":null,"affiliations":[]},{"author_position":"middle","author":{"id":"https://openalex.org/A5084729483","display_name":"Heiko van der Kuip","orcid":null,"observed_orcids":[]},"institutions":[],"countries":[],"is_corresponding":false,"raw_author_name":"Heiko van der Kuip","raw_affiliation_strings":[],"raw_orcid":null,"affiliations":[]},{"author_position":"middle","author":{"id":"https://openalex.org/A5059195101","display_name":"Ingolf Cascorbi","orcid":"https://orcid.org/0000-0002-2182-9534","observed_orcids":["https://orcid.org/0000-0002-2182-9534"]},"institutions":[],"countries":[],"is_corresponding":false,"raw_author_name":"Ingolf Cascorbi","raw_affiliation_strings":[],"raw_orcid":null,"affiliations":[]},{"author_position":"middle","author":{"id":"https://openalex.org/A5079746940","display_name":"Oliver Bruhn","orcid":null,"observed_orcids":[]},"institutions":[],"countries":[],"is_corresponding":false,"raw_author_name":"Oliver Bruhn","raw_affiliation_strings":[],"raw_orcid":null,"affiliations":[]},{"author_position":"middle","author":{"id":"https://openalex.org/A5061380659","display_name":"Michael Kneba","orcid":null,"observed_orcids":[]},"institutions":[],"countries":[],"is_corresponding":false,"raw_author_name":"Michael Kneba","raw_affiliation_strings":[],"raw_orcid":null,"affiliations":[]},{"author_position":"middle","author":{"id":"https://openalex.org/A5114444398","display_name":"Christiane Pott","orcid":"https://orcid.org/0009-0005-9260-8340","observed_orcids":["https://orcid.org/0009-0005-9260-8340"]},"institutions":[],"countries":[],"is_corresponding":false,"raw_author_name":"Christiane Pott","raw_affiliation_strings":[],"raw_orcid":null,"affiliations":[]},{"author_position":"middle","author":{"id":"https://openalex.org/A5040542934","display_name":"Ute Hofmann","orcid":"https://orcid.org/0000-0003-0823-9027","observed_orcids":["https://orcid.org/0000-0003-0823-9027"]},"institutions":[],"countries":[],"is_corresponding":false,"raw_author_name":"Ute Hofmann","raw_affiliation_strings":[],"raw_orcid":null,"affiliations":[]},{"author_position":"middle","author":{"id":"https://openalex.org/A5035561994","display_name":"Christopher Volk","orcid":"https://orcid.org/0000-0002-4029-4504","observed_orcids":["https://orcid.org/0000-0002-4029-4504"]},"institutions":[],"countries":[],"is_corresponding":false,"raw_author_name":"Christopher Volk","raw_affiliation_strings":[],"raw_orcid":null,"affiliations":[]},{"author_position":"middle","author":{"id":"https://openalex.org/A5077955893","display_name":"Shuiying Hu","orcid":"https://orcid.org/0000-0002-9806-7734","observed_orcids":["https://orcid.org/0000-0002-9806-7734"]},"institutions":[],"countries":[],"is_corresponding":false,"raw_author_name":"Shuiying Hu","raw_affiliation_strings":[],"raw_orcid":null,"affiliations":[]},{"author_position":"middle","author":{"id":"https://openalex.org/A5077260725","display_name":"Sharyn D. Baker","orcid":"https://orcid.org/0000-0003-3062-3252","observed_orcids":["https://orcid.org/0000-0003-3062-3252"]},"institutions":[],"countries":[],"is_corresponding":false,"raw_author_name":"Sharyn D. Baker","raw_affiliation_strings":[],"raw_orcid":null,"affiliations":[]},{"author_position":"middle","author":{"id":"https://openalex.org/A5065279964","display_name":"Alex Sparreboom","orcid":"https://orcid.org/0000-0003-2660-6644","observed_orcids":["https://orcid.org/0000-0003-2660-6644"]},"institutions":[],"countries":[],"is_corresponding":false,"raw_author_name":"Alex Sparreboom","raw_affiliation_strings":[],"raw_orcid":null,"affiliations":[]},{"author_position":"middle","author":{"id":"https://openalex.org/A5103257809","display_name":"Peter Ruth","orcid":"https://orcid.org/0000-0002-1092-857X","observed_orcids":["https://orcid.org/0000-0002-1092-857X"]},"institutions":[],"countries":[],"is_corresponding":false,"raw_author_name":"Peter Ruth","raw_affiliation_strings":[],"raw_orcid":null,"affiliations":[]},{"author_position":"middle","author":{"id":"https://openalex.org/A5064438527","display_name":"Hermann Koepsell","orcid":"https://orcid.org/0000-0001-5118-7088","observed_orcids":["https://orcid.org/0000-0001-5118-7088"]},"institutions":[],"countries":[],"is_corresponding":false,"raw_author_name":"Hermann Koepsell","raw_affiliation_strings":[],"raw_orcid":null,"affiliations":[]},{"author_position":"last","author":{"id":"https://openalex.org/A5057183308","display_name":"Matthias Georg Schwab","orcid":"https://orcid.org/0000-0002-9984-075X","observed_orcids":["https://orcid.org/0000-0002-9984-075X","https://orcid.org/0000-0001-6999-1795"]},"institutions":[],"countries":[],"is_corresponding":false,"raw_author_name":"Matthias Schwab","raw_affiliation_strings":[],"raw_orcid":null,"affiliations":[]}],"institutions":[],"countries_distinct_count":0,"institutions_distinct_count":0,"corresponding_author_ids":[],"corresponding_institution_ids":[],"apc_list":null,"apc_paid":null,"fwci":null,"has_fulltext":true,"cited_by_count":0,"citation_normalized_percentile":null,"cited_by_percentile_year":null,"biblio":{"volume":null,"issue":null,"first_page":null,"last_page":null},"is_retracted":false,"is_paratext":false,"is_xpac":false,"primary_topic":{"id":"https://openalex.org/T10570","display_name":"Drug Transport and Resistance Mechanisms","score":0.9994999766349792,"subfield":{"id":"https://openalex.org/subfields/2730","display_name":"Oncology"},"field":{"id":"https://openalex.org/fields/27","display_name":"Medicine"},"domain":{"id":"https://openalex.org/domains/4","display_name":"Health Sciences"}},"topics":[{"id":"https://openalex.org/T10570","display_name":"Drug Transport and Resistance Mechanisms","score":0.9994999766349792,"subfield":{"id":"https://openalex.org/subfields/2730","display_name":"Oncology"},"field":{"id":"https://openalex.org/fields/27","display_name":"Medicine"},"domain":{"id":"https://openalex.org/domains/4","display_name":"Health Sciences"}},{"id":"https://openalex.org/T10375","display_name":"Pharmacogenetics and Drug Metabolism","score":9.999999747378752e-05,"subfield":{"id":"https://openalex.org/subfields/3004","display_name":"Pharmacology"},"field":{"id":"https://openalex.org/fields/30","display_name":"Pharmacology, Toxicology and Pharmaceutics"},"domain":{"id":"https://openalex.org/domains/1","display_name":"Life Sciences"}},{"id":"https://openalex.org/T11215","display_name":"Chronic Myeloid Leukemia Treatments","score":9.999999747378752e-05,"subfield":{"id":"https://openalex.org/subfields/2720","display_name":"Hematology"},"field":{"id":"https://openalex.org/fields/27","display_name":"Medicine"},"domain":{"id":"https://openalex.org/domains/4","display_name":"Health Sciences"}}],"keywords":[{"id":"https://openalex.org/keywords/imatinib","display_name":"imatinib","score":0.9929999709129333},{"id":"https://openalex.org/keywords/cellular-uptake","display_name":"cellular uptake","score":0.9200000166893005},{"id":"https://openalex.org/keywords/leukemia-cells","display_name":"leukemia cells","score":0.7379999756813049},{"id":"https://openalex.org/keywords/oct1","display_name":"OCT1","score":0.9649999737739563},{"id":"https://openalex.org/keywords/drug-transport","display_name":"drug transport","score":0.6019999980926514},{"id":"https://openalex.org/keywords/shrna-knockdown","display_name":"shRNA knockdown","score":0.7960000038146973},{"id":"https://openalex.org/keywords/leukemia","display_name":"leukemia","score":0.35499998927116394}],"concepts":[{"id":"https://openalex.org/C189613389","wikidata":"https://www.wikidata.org/wiki/Q70479817","display_name":"Organic cation transport proteins","level":4,"score":0.7883962392807007},{"id":"https://openalex.org/C553184892","wikidata":"https://www.wikidata.org/wiki/Q1141429","display_name":"Flow cytometry","level":2,"score":0.6781063079833984},{"id":"https://openalex.org/C2777583451","wikidata":"https://www.wikidata.org/wiki/Q177094","display_name":"Imatinib","level":3,"score":0.640935480594635},{"id":"https://openalex.org/C173396325","wikidata":"https://www.wikidata.org/wiki/Q1501275","display_name":"Gene knockdown","level":3,"score":0.6298989057540894},{"id":"https://openalex.org/C190232843","wikidata":"https://www.wikidata.org/wiki/Q1950808","display_name":"Small hairpin RNA","level":4,"score":0.6188125610351562},{"id":"https://openalex.org/C185592680","wikidata":"https://www.wikidata.org/wiki/Q2329","display_name":"Chemistry","level":0,"score":0.5481642484664917},{"id":"https://openalex.org/C149011108","wikidata":"https://www.wikidata.org/wiki/Q652985","display_name":"Transporter","level":3,"score":0.5069546699523926},{"id":"https://openalex.org/C95444343","wikidata":"https://www.wikidata.org/wiki/Q7141","display_name":"Cell biology","level":1,"score":0.4839184880256653},{"id":"https://openalex.org/C2779178360","wikidata":"https://www.wikidata.org/wiki/Q902045","display_name":"Confocal microscopy","level":2,"score":0.45960238575935364},{"id":"https://openalex.org/C81885089","wikidata":"https://www.wikidata.org/wiki/Q189082","display_name":"Cell culture","level":2,"score":0.45052558183670044},{"id":"https://openalex.org/C3019892230","wikidata":"https://www.wikidata.org/wiki/Q177094","display_name":"Imatinib mesylate","level":4,"score":0.44939571619033813},{"id":"https://openalex.org/C502942594","wikidata":"https://www.wikidata.org/wiki/Q3421914","display_name":"Cancer research","level":1,"score":0.4408688545227051},{"id":"https://openalex.org/C153911025","wikidata":"https://www.wikidata.org/wiki/Q7202","display_name":"Molecular biology","level":1,"score":0.39517271518707275},{"id":"https://openalex.org/C86803240","wikidata":"https://www.wikidata.org/wiki/Q420","display_name":"Biology","level":0,"score":0.27038896083831787},{"id":"https://openalex.org/C55493867","wikidata":"https://www.wikidata.org/wiki/Q7094","display_name":"Biochemistry","level":1,"score":0.20191076397895813},{"id":"https://openalex.org/C104317684","wikidata":"https://www.wikidata.org/wiki/Q7187","display_name":"Gene","level":2,"score":0.09313973784446716},{"id":"https://openalex.org/C54355233","wikidata":"https://www.wikidata.org/wiki/Q7162","display_name":"Genetics","level":1,"score":0.06514498591423035},{"id":"https://openalex.org/C2778729363","wikidata":"https://www.wikidata.org/wiki/Q11688946","display_name":"Myeloid leukemia","level":2,"score":0.0}],"mesh":[],"locations_count":3,"locations":[{"id":"doi:10.1158/1078-0432.22449923","doi":"https://doi.org/10.1158/1078-0432.22449923","is_oa":true,"landing_page_url":"http://dx.doi.org/10.1158/1078-0432.22449923","pdf_url":"https://aacr.figshare.com/articles/journal_contribution/Supplementary_Methods_from_Cellular_Uptake_of_Imatinib_into_Leukemic_Cells_Is_Independent_of_Human_Organic_Cation_Transporter_1_OCT1_/22449923/1/files/39900983.pdf","source":null,"license":"cc-by","license_id":"https://openalex.org/licenses/cc-by","version":"acceptedVersion","is_accepted":true,"is_published":false,"raw_source_name":"American Association for Cancer Research","raw_type":"posted-content"},{"id":"doi:10.1158/1078-0432.22449923.v1","doi":"https://doi.org/10.1158/1078-0432.22449923.v1","is_oa":true,"landing_page_url":"https://doi.org/10.1158/1078-0432.22449923.v1","pdf_url":null,"source":null,"license":"cc-by","license_id":"https://openalex.org/licenses/cc-by","version":"acceptedVersion","is_accepted":true,"is_published":false,"raw_source_name":"American Association for Cancer Research","raw_type":"posted-content"},{"id":"pmh:oai:figshare.com:article/22449923","doi":null,"is_oa":true,"landing_page_url":"https://figshare.com/articles/journal_contribution/Supplementary_Methods_from_Cellular_Uptake_of_Imatinib_into_Leukemic_Cells_Is_Independent_of_Human_Organic_Cation_Transporter_1_OCT1_/22449923","pdf_url":null,"source":{"id":"https://openalex.org/S4377196282","display_name":"Figshare","issn_l":null,"issn":null,"is_oa":false,"is_in_doaj":false,"is_core":false,"listed_in":[],"host_organization":"https://openalex.org/I4210132348","host_organization_name":"Figshare (United Kingdom)","host_organization_lineage":["https://openalex.org/I4210132348"],"host_organization_lineage_names":[],"type":"repository"},"license":"cc-by","license_id":"https://openalex.org/licenses/cc-by","version":"submittedVersion","is_accepted":false,"is_published":false,"raw_source_name":"","raw_type":"Text"}],"best_oa_location":{"id":"doi:10.1158/1078-0432.22449923","doi":"https://doi.org/10.1158/1078-0432.22449923","is_oa":true,"landing_page_url":"http://dx.doi.org/10.1158/1078-0432.22449923","pdf_url":"https://aacr.figshare.com/articles/journal_contribution/Supplementary_Methods_from_Cellular_Uptake_of_Imatinib_into_Leukemic_Cells_Is_Independent_of_Human_Organic_Cation_Transporter_1_OCT1_/22449923/1/files/39900983.pdf","source":null,"license":"cc-by","license_id":"https://openalex.org/licenses/cc-by","version":"acceptedVersion","is_accepted":true,"is_published":false,"raw_source_name":"American Association for Cancer Research","raw_type":"posted-content"},"sustainable_development_goals":[{"id":"https://metadata.un.org/sdg/3","score":0.8199999928474426,"display_name":"Good health and well-being"}],"study_designs":[],"awards":[],"funders":[],"has_content":{"pdf":true,"grobid_xml":true},"content_urls":{"pdf":"https://content.openalex.org/works/W4361908315.pdf","grobid_xml":"https://content.openalex.org/works/W4361908315.grobid-xml"},"referenced_works_count":6,"referenced_works":["https://openalex.org/W1966271190","https://openalex.org/W2030242630","https://openalex.org/W2097072837","https://openalex.org/W2143409207","https://openalex.org/W2235836043","https://openalex.org/W2337788645"],"related_works":["https://openalex.org/W4361950954","https://openalex.org/W2008702214","https://openalex.org/W2068959104","https://openalex.org/W2155229204","https://openalex.org/W2953576043","https://openalex.org/W2092475279","https://openalex.org/W2956127634","https://openalex.org/W1840691103","https://openalex.org/W2093197708","https://openalex.org/W3016785925"],"abstract_inverted_index":{"PDF":[0],"file":[1],"65K,":[2],"Supplementary":[3],"methods":[4],"including":[5],"chemicals,":[6],"generation":[7],"of":[8,25],"a":[9],"cell":[10,21],"line":[11],"expressing":[12],"OCT1":[13],"variant":[14],"p.V408,":[15],"transport":[16],"studies":[17],"using":[18],"oocytes":[19],"and":[20,29,35],"lines,":[22],"LC-MS-MS":[23],"analysis":[24],"imatinib,":[26],"RNA":[27],"isolation":[28],"quantification,":[30],"shRNA":[31],"knockdown,":[32],"flow":[33],"cytometry":[34],"confocal":[36],"laser":[37],"scanning":[38],"microscopy":[39]},"counts_by_year":[],"updated_date":"2026-11-05T12:25:35.769452","created_date":"2023-04-05T00:00:00"}
