{"id":"https://openalex.org/W2951234780","doi":"https://doi.org/10.1002/chin.199649167","title":"ChemInform Abstract: Nonpeptidal P2 Ligands for HIV Protease Inhibitors: Structure\u2010Based Design, Synthesis, and Biological Evaluation.","display_name":"ChemInform Abstract: Nonpeptidal P2 Ligands for HIV Protease Inhibitors: Structure\u2010Based Design, Synthesis, and Biological Evaluation.","publication_year":1996,"publication_date":"1996-12-03","ids":{"openalex":"https://openalex.org/W2951234780","doi":"https://doi.org/10.1002/chin.199649167","mag":"2951234780"},"language":"en","primary_location":{"id":"doi:10.1002/chin.199649167","doi":"https://doi.org/10.1002/chin.199649167","is_oa":false,"landing_page_url":"https://doi.org/10.1002/chin.199649167","pdf_url":null,"source":{"id":"https://openalex.org/S41354064","display_name":"ChemInform","issn_l":"0009-2975","issn":["0009-2975","0931-7597","1431-5890","1522-2667","2199-2924"],"is_oa":false,"is_in_doaj":false,"is_core":false,"listed_in":[],"host_organization":"https://openalex.org/P4310320595","host_organization_name":"Wiley","host_organization_lineage":["https://openalex.org/P4310320595"],"host_organization_lineage_names":["Wiley"],"type":"journal"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"ChemInform","raw_type":"journal-article"},"volume":null,"type":"article","indexed_in":["crossref"],"open_access":{"is_oa":false,"oa_status":"closed","oa_url":null,"any_repository_has_fulltext":false},"authorships":[{"author_position":"first","author":{"id":"https://openalex.org/A5041773055","display_name":"Arun Kumar Ghosh","orcid":"https://orcid.org/0000-0003-2472-1841","observed_orcids":["https://orcid.org/0000-0003-2472-1841"]},"institutions":[{"id":"https://openalex.org/I39422238","display_name":"University of Illinois Chicago","ror":"https://ror.org/02mpq6x41","country_code":"US","type":"education","lineage":["https://openalex.org/I39422238"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"A. K. GHOSH","raw_affiliation_strings":["Dep. Chem., Univ. Ill., Chicago, IL 60607, USA"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Dep. Chem., Univ. Ill., Chicago, IL 60607, USA","institution_ids":["https://openalex.org/I39422238"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5021745178","display_name":"John Kincaid","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I39422238","display_name":"University of Illinois Chicago","ror":"https://ror.org/02mpq6x41","country_code":"US","type":"education","lineage":["https://openalex.org/I39422238"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"J. F. KINCAID","raw_affiliation_strings":["Dep. Chem., Univ. Ill., Chicago, IL 60607, USA"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Dep. Chem., Univ. Ill., Chicago, IL 60607, USA","institution_ids":["https://openalex.org/I39422238"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5045349762","display_name":"D. Eric Walters","orcid":"https://orcid.org/0000-0002-1513-3522","observed_orcids":["https://orcid.org/0000-0002-1513-3522"]},"institutions":[{"id":"https://openalex.org/I39422238","display_name":"University of Illinois Chicago","ror":"https://ror.org/02mpq6x41","country_code":"US","type":"education","lineage":["https://openalex.org/I39422238"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"D. E. WALTERS","raw_affiliation_strings":["Dep. Chem., Univ. Ill., Chicago, IL 60607, USA"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Dep. Chem., Univ. Ill., Chicago, IL 60607, USA","institution_ids":["https://openalex.org/I39422238"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5075899759","display_name":"Y. CHEN","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I39422238","display_name":"University of Illinois Chicago","ror":"https://ror.org/02mpq6x41","country_code":"US","type":"education","lineage":["https://openalex.org/I39422238"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"Y. CHEN","raw_affiliation_strings":["Dep. Chem., Univ. Ill., Chicago, IL 60607, USA"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Dep. Chem., Univ. Ill., Chicago, IL 60607, USA","institution_ids":["https://openalex.org/I39422238"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5023147552","display_name":"N. C. Chaudhuri","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I39422238","display_name":"University of Illinois Chicago","ror":"https://ror.org/02mpq6x41","country_code":"US","type":"education","lineage":["https://openalex.org/I39422238"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"N. C. CHAUDHURI","raw_affiliation_strings":["Dep. Chem., Univ. Ill., Chicago, IL 60607, USA"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Dep. Chem., Univ. Ill., Chicago, IL 60607, USA","institution_ids":["https://openalex.org/I39422238"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5043405937","display_name":"Wayne J. Thompson","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I39422238","display_name":"University of Illinois Chicago","ror":"https://ror.org/02mpq6x41","country_code":"US","type":"education","lineage":["https://openalex.org/I39422238"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"W. J. THOMPSON","raw_affiliation_strings":["Dep. Chem., Univ. Ill., Chicago, IL 60607, USA"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Dep. Chem., Univ. Ill., Chicago, IL 60607, USA","institution_ids":["https://openalex.org/I39422238"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5112105938","display_name":"Chris Culberson","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I39422238","display_name":"University of Illinois Chicago","ror":"https://ror.org/02mpq6x41","country_code":"US","type":"education","lineage":["https://openalex.org/I39422238"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"C. CULBERSON","raw_affiliation_strings":["Dep. Chem., Univ. Ill., Chicago, IL 60607, USA"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Dep. Chem., Univ. Ill., Chicago, IL 60607, USA","institution_ids":["https://openalex.org/I39422238"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5011257479","display_name":"P. M. D. Fitzgerald","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I39422238","display_name":"University of Illinois Chicago","ror":"https://ror.org/02mpq6x41","country_code":"US","type":"education","lineage":["https://openalex.org/I39422238"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"P. M. D. FITZGERALD","raw_affiliation_strings":["Dep. Chem., Univ. Ill., Chicago, IL 60607, USA"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Dep. Chem., Univ. Ill., Chicago, IL 60607, USA","institution_ids":["https://openalex.org/I39422238"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5025168375","display_name":"H. Y. LEE","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I39422238","display_name":"University of Illinois Chicago","ror":"https://ror.org/02mpq6x41","country_code":"US","type":"education","lineage":["https://openalex.org/I39422238"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"H. Y. LEE","raw_affiliation_strings":["Dep. Chem., Univ. Ill., Chicago, IL 60607, USA"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Dep. Chem., Univ. Ill., Chicago, IL 60607, USA","institution_ids":["https://openalex.org/I39422238"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5041852182","display_name":"Sean P. McKee","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I39422238","display_name":"University of Illinois Chicago","ror":"https://ror.org/02mpq6x41","country_code":"US","type":"education","lineage":["https://openalex.org/I39422238"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"S. P. MCKEE","raw_affiliation_strings":["Dep. Chem., Univ. Ill., Chicago, IL 60607, USA"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Dep. Chem., Univ. Ill., Chicago, IL 60607, USA","institution_ids":["https://openalex.org/I39422238"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5072861581","display_name":"Peter M. Munson","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I39422238","display_name":"University of Illinois Chicago","ror":"https://ror.org/02mpq6x41","country_code":"US","type":"education","lineage":["https://openalex.org/I39422238"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"P. M. MUNSON","raw_affiliation_strings":["Dep. Chem., Univ. Ill., Chicago, IL 60607, USA"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Dep. Chem., Univ. Ill., Chicago, IL 60607, USA","institution_ids":["https://openalex.org/I39422238"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5114237732","display_name":"Tien T. Duong","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I39422238","display_name":"University of Illinois Chicago","ror":"https://ror.org/02mpq6x41","country_code":"US","type":"education","lineage":["https://openalex.org/I39422238"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"T. T. DUONG","raw_affiliation_strings":["Dep. Chem., Univ. Ill., Chicago, IL 60607, USA"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Dep. Chem., Univ. Ill., Chicago, IL 60607, USA","institution_ids":["https://openalex.org/I39422238"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5035072487","display_name":"Paul L. Darke","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I39422238","display_name":"University of Illinois Chicago","ror":"https://ror.org/02mpq6x41","country_code":"US","type":"education","lineage":["https://openalex.org/I39422238"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"P. L. DARKE","raw_affiliation_strings":["Dep. Chem., Univ. Ill., Chicago, IL 60607, USA"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Dep. Chem., Univ. Ill., Chicago, IL 60607, USA","institution_ids":["https://openalex.org/I39422238"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5084996174","display_name":"Joan A. Zugay","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I39422238","display_name":"University of Illinois Chicago","ror":"https://ror.org/02mpq6x41","country_code":"US","type":"education","lineage":["https://openalex.org/I39422238"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"J. A. ZUGAY","raw_affiliation_strings":["Dep. Chem., Univ. Ill., Chicago, IL 60607, USA"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Dep. Chem., Univ. Ill., Chicago, IL 60607, USA","institution_ids":["https://openalex.org/I39422238"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5030101432","display_name":"William A. Schleif","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I39422238","display_name":"University of Illinois Chicago","ror":"https://ror.org/02mpq6x41","country_code":"US","type":"education","lineage":["https://openalex.org/I39422238"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"W. A. SCHLEIF","raw_affiliation_strings":["Dep. Chem., Univ. Ill., Chicago, IL 60607, USA"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Dep. Chem., Univ. Ill., Chicago, IL 60607, USA","institution_ids":["https://openalex.org/I39422238"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5024929715","display_name":"M. G. AXEL","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I39422238","display_name":"University of Illinois Chicago","ror":"https://ror.org/02mpq6x41","country_code":"US","type":"education","lineage":["https://openalex.org/I39422238"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"M. G. AXEL","raw_affiliation_strings":["Dep. Chem., Univ. Ill., Chicago, IL 60607, USA"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Dep. Chem., Univ. Ill., Chicago, IL 60607, USA","institution_ids":["https://openalex.org/I39422238"]}]},{"author_position":"middle","author":{"id":null,"display_name":"J. LIN","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I39422238","display_name":"University of Illinois Chicago","ror":"https://ror.org/02mpq6x41","country_code":"US","type":"education","lineage":["https://openalex.org/I39422238"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"J. LIN","raw_affiliation_strings":["Dep. Chem., Univ. Ill., Chicago, IL 60607, USA"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Dep. Chem., Univ. Ill., Chicago, IL 60607, USA","institution_ids":["https://openalex.org/I39422238"]}]},{"author_position":"last","author":{"id":"https://openalex.org/A5056177752","display_name":"Joel R. Huff","orcid":"https://orcid.org/0009-0002-0695-6540","observed_orcids":["https://orcid.org/0009-0002-0695-6540"]},"institutions":[{"id":"https://openalex.org/I39422238","display_name":"University of Illinois Chicago","ror":"https://ror.org/02mpq6x41","country_code":"US","type":"education","lineage":["https://openalex.org/I39422238"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"J. R. HUFF","raw_affiliation_strings":["Dep. Chem., Univ. Ill., Chicago, IL 60607, USA"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Dep. Chem., Univ. Ill., Chicago, IL 60607, USA","institution_ids":["https://openalex.org/I39422238"]}]}],"institutions":[],"countries_distinct_count":1,"institutions_distinct_count":1,"corresponding_author_ids":[],"corresponding_institution_ids":["https://openalex.org/I39422238"],"apc_list":null,"apc_paid":null,"fwci":0.0,"has_fulltext":false,"cited_by_count":0,"citation_normalized_percentile":{"value":0.41607496,"is_in_top_1_percent":false,"is_in_top_10_percent":false},"cited_by_percentile_year":null,"biblio":{"volume":"27","issue":"49","first_page":null,"last_page":null},"is_retracted":false,"is_paratext":false,"is_xpac":false,"primary_topic":{"id":"https://openalex.org/T10526","display_name":"HIV/AIDS drug development and treatment","score":0.6807000041007996,"subfield":{"id":"https://openalex.org/subfields/2725","display_name":"Infectious Diseases"},"field":{"id":"https://openalex.org/fields/27","display_name":"Medicine"},"domain":{"id":"https://openalex.org/domains/4","display_name":"Health Sciences"}},"topics":[{"id":"https://openalex.org/T10526","display_name":"HIV/AIDS drug development and treatment","score":0.6807000041007996,"subfield":{"id":"https://openalex.org/subfields/2725","display_name":"Infectious Diseases"},"field":{"id":"https://openalex.org/fields/27","display_name":"Medicine"},"domain":{"id":"https://openalex.org/domains/4","display_name":"Health Sciences"}},{"id":"https://openalex.org/T10211","display_name":"Computational Drug Discovery Methods","score":0.17319999635219574,"subfield":{"id":"https://openalex.org/subfields/1703","display_name":"Computational Theory and Mathematics"},"field":{"id":"https://openalex.org/fields/17","display_name":"Computer Science"},"domain":{"id":"https://openalex.org/domains/3","display_name":"Physical Sciences"}},{"id":"https://openalex.org/T10911","display_name":"Chemical Synthesis and Analysis","score":0.023099999874830246,"subfield":{"id":"https://openalex.org/subfields/1312","display_name":"Molecular Biology"},"field":{"id":"https://openalex.org/fields/13","display_name":"Biochemistry, Genetics and Molecular Biology"},"domain":{"id":"https://openalex.org/domains/1","display_name":"Life Sciences"}}],"keywords":[{"id":"https://openalex.org/keywords/hiv-protease-inhibitors","display_name":"HIV protease inhibitors","score":0.9760000109672546},{"id":"https://openalex.org/keywords/structure-based-drug-design","display_name":"structure-based drug design","score":0.9269999861717224},{"id":"https://openalex.org/keywords/antiretroviral-drug-synthesis","display_name":"antiretroviral drug synthesis","score":0.640999972820282},{"id":"https://openalex.org/keywords/biological-evaluation","display_name":"biological evaluation","score":0.6290000081062317}],"concepts":[{"id":"https://openalex.org/C185592680","wikidata":"https://www.wikidata.org/wiki/Q2329","display_name":"Chemistry","level":0,"score":0.9465315341949463},{"id":"https://openalex.org/C3013748606","wikidata":"https://www.wikidata.org/wiki/Q15787","display_name":"Human immunodeficiency virus (HIV)","level":2,"score":0.6171778440475464},{"id":"https://openalex.org/C21951064","wikidata":"https://www.wikidata.org/wiki/Q899212","display_name":"Combinatorial chemistry","level":1,"score":0.5572705864906311},{"id":"https://openalex.org/C2776714187","wikidata":"https://www.wikidata.org/wiki/Q212410","display_name":"Protease","level":3,"score":0.5466776490211487},{"id":"https://openalex.org/C2780378061","wikidata":"https://www.wikidata.org/wiki/Q25351891","display_name":"Service (business)","level":2,"score":0.41949793696403503},{"id":"https://openalex.org/C70721500","wikidata":"https://www.wikidata.org/wiki/Q177005","display_name":"Computational biology","level":1,"score":0.37313249707221985},{"id":"https://openalex.org/C71240020","wikidata":"https://www.wikidata.org/wiki/Q186011","display_name":"Stereochemistry","level":1,"score":0.3545830249786377},{"id":"https://openalex.org/C171250308","wikidata":"https://www.wikidata.org/wiki/Q11468","display_name":"Nanotechnology","level":1,"score":0.35435473918914795},{"id":"https://openalex.org/C55493867","wikidata":"https://www.wikidata.org/wiki/Q7094","display_name":"Biochemistry","level":1,"score":0.19377636909484863},{"id":"https://openalex.org/C159047783","wikidata":"https://www.wikidata.org/wiki/Q7215","display_name":"Virology","level":1,"score":0.17457789182662964},{"id":"https://openalex.org/C181199279","wikidata":"https://www.wikidata.org/wiki/Q8047","display_name":"Enzyme","level":2,"score":0.11701041460037231},{"id":"https://openalex.org/C144133560","wikidata":"https://www.wikidata.org/wiki/Q4830453","display_name":"Business","level":0,"score":0.08623501658439636},{"id":"https://openalex.org/C162853370","wikidata":"https://www.wikidata.org/wiki/Q39809","display_name":"Marketing","level":1,"score":0.0},{"id":"https://openalex.org/C86803240","wikidata":"https://www.wikidata.org/wiki/Q420","display_name":"Biology","level":0,"score":0.0},{"id":"https://openalex.org/C192562407","wikidata":"https://www.wikidata.org/wiki/Q228736","display_name":"Materials science","level":0,"score":0.0}],"mesh":[],"locations_count":1,"locations":[{"id":"doi:10.1002/chin.199649167","doi":"https://doi.org/10.1002/chin.199649167","is_oa":false,"landing_page_url":"https://doi.org/10.1002/chin.199649167","pdf_url":null,"source":{"id":"https://openalex.org/S41354064","display_name":"ChemInform","issn_l":"0009-2975","issn":["0009-2975","0931-7597","1431-5890","1522-2667","2199-2924"],"is_oa":false,"is_in_doaj":false,"is_core":false,"listed_in":[],"host_organization":"https://openalex.org/P4310320595","host_organization_name":"Wiley","host_organization_lineage":["https://openalex.org/P4310320595"],"host_organization_lineage_names":["Wiley"],"type":"journal"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"ChemInform","raw_type":"journal-article"}],"best_oa_location":null,"sustainable_development_goals":[],"study_designs":[],"awards":[],"funders":[],"has_content":{"grobid_xml":false,"pdf":false},"content_urls":null,"referenced_works_count":1,"referenced_works":["https://openalex.org/W1986457945"],"related_works":["https://openalex.org/W2951127150","https://openalex.org/W2951553557","https://openalex.org/W2951709228","https://openalex.org/W2950610167","https://openalex.org/W1979716465","https://openalex.org/W2077240119","https://openalex.org/W2949844236","https://openalex.org/W2950408874","https://openalex.org/W2050966037","https://openalex.org/W2953151950"],"abstract_inverted_index":{"Abstract":[0,25],"ChemInform":[1,24],"is":[2,42],"a":[3,11,23,35],"weekly":[4],"Abstracting":[5],"Service,":[6],"delivering":[7],"concise":[8],"information":[9],"at":[10],"glance":[12],"that":[13],"was":[14,30],"extracted":[15],"from":[16],"about":[17],"100":[18],"leading":[19],"journals.":[20],"To":[21],"access":[22],"of":[26],"an":[27],"article":[28,41],"which":[29],"published":[31],"elsewhere,":[32],"please":[33],"select":[34],"\u201cFull":[36],"Text\u201d":[37],"option.":[38,47],"The":[39],"original":[40],"trackable":[43],"via":[44],"the":[45],"\u201cReferences\u201d":[46]},"counts_by_year":[],"updated_date":"2026-10-14T16:39:01.820549","created_date":"2019-06-27T00:00:00"}
