{"id":"https://openalex.org/W2950425558","doi":"https://doi.org/10.3987/com-04-10071","title":"Facile Methods for Preparation of Thiazolopyridine and Tetrahydro-thiazolopyridine Derivatives","display_name":"Facile Methods for Preparation of Thiazolopyridine and Tetrahydro-thiazolopyridine Derivatives","publication_year":2004,"publication_date":"2004-01-01","ids":{"openalex":"https://openalex.org/W2950425558","doi":"https://doi.org/10.3987/com-04-10071","mag":"2950425558"},"language":"en","primary_location":{"id":"doi:10.3987/com-04-10071","doi":"https://doi.org/10.3987/com-04-10071","is_oa":false,"landing_page_url":"https://doi.org/10.3987/com-04-10071","pdf_url":null,"source":{"id":"https://openalex.org/S27298842","display_name":"Heterocycles","issn_l":"0385-5414","issn":["0385-5414","1881-0942"],"is_oa":false,"is_in_doaj":false,"is_core":true,"listed_in":["cwts-core","jufo-1","norway-1","poland-40","russia-white-list-4"],"host_organization":"https://openalex.org/P4310320990","host_organization_name":"Elsevier BV","host_organization_lineage":["https://openalex.org/P4310320990"],"host_organization_lineage_names":["Elsevier BV"],"type":"journal"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"HETEROCYCLES","raw_type":"journal-article"},"volume":null,"type":"article","is_traditional":true,"indexed_in":["crossref"],"open_access":{"is_oa":false,"oa_status":"closed","oa_url":null,"any_repository_has_fulltext":false},"authorships":[{"author_position":"first","author":{"id":"https://openalex.org/A5043627463","display_name":"Noriyasu Haginoya","orcid":null,"observed_orcids":[]},"institutions":[],"countries":[],"is_corresponding":true,"raw_author_name":"Noriyasu Haginoya","raw_affiliation_strings":["Medicinal Chemistry Reseach Laboratoty, Daiichi Pharmaceutical Co., Ltd, 1-16-13, Kita-Kasai, Edogawa-ku, Tokyo 134-8630, Japan;"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Medicinal Chemistry Reseach Laboratoty, Daiichi Pharmaceutical Co., Ltd, 1-16-13, Kita-Kasai, Edogawa-ku, Tokyo 134-8630, Japan;","institution_ids":[]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5017854667","display_name":"Satoshi Komoriya","orcid":"https://orcid.org/0000-0003-3809-6290","observed_orcids":["https://orcid.org/0000-0003-3809-6290"]},"institutions":[],"countries":[],"is_corresponding":false,"raw_author_name":"Satoshi Komoriya","raw_affiliation_strings":["Medicinal Chemistry Reseach Laboratoty, Daiichi Pharmaceutical Co., Ltd, 1-16-13, Kita-Kasai, Edogawa-ku, Tokyo 134-8630, Japan;"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Medicinal Chemistry Reseach Laboratoty, Daiichi Pharmaceutical Co., Ltd, 1-16-13, Kita-Kasai, Edogawa-ku, Tokyo 134-8630, Japan;","institution_ids":[]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5110641697","display_name":"Ken Osanai","orcid":null,"observed_orcids":[]},"institutions":[],"countries":[],"is_corresponding":false,"raw_author_name":"Ken Osanai","raw_affiliation_strings":["Medicinal Chemistry Reseach Laboratoty, Daiichi Pharmaceutical Co., Ltd, 1-16-13, Kita-Kasai, Edogawa-ku, Tokyo 134-8630, Japan;"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Medicinal Chemistry Reseach Laboratoty, Daiichi Pharmaceutical Co., Ltd, 1-16-13, Kita-Kasai, Edogawa-ku, Tokyo 134-8630, Japan;","institution_ids":[]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5113580718","display_name":"Toshiharu Yoshino","orcid":null,"observed_orcids":[]},"institutions":[],"countries":[],"is_corresponding":false,"raw_author_name":"Toshiharu Yoshino","raw_affiliation_strings":["Medicinal Chemistry Reseach Laboratoty, Daiichi Pharmaceutical Co., Ltd, 1-16-13, Kita-Kasai, Edogawa-ku, Tokyo 134-8630, Japan;"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Medicinal Chemistry Reseach Laboratoty, Daiichi Pharmaceutical Co., Ltd, 1-16-13, Kita-Kasai, Edogawa-ku, Tokyo 134-8630, Japan;","institution_ids":[]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5108571100","display_name":"Tsutomu Nagata","orcid":null,"observed_orcids":[]},"institutions":[],"countries":[],"is_corresponding":false,"raw_author_name":"Tsutomu Nagata","raw_affiliation_strings":["Medicinal Chemistry Reseach Laboratoty, Daiichi Pharmaceutical Co., Ltd, 1-16-13, Kita-Kasai, Edogawa-ku, Tokyo 134-8630, Japan;"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Medicinal Chemistry Reseach Laboratoty, Daiichi Pharmaceutical Co., Ltd, 1-16-13, Kita-Kasai, Edogawa-ku, Tokyo 134-8630, Japan;","institution_ids":[]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5065836713","display_name":"Masatoshi Nagamochi","orcid":null,"observed_orcids":[]},"institutions":[],"countries":[],"is_corresponding":false,"raw_author_name":"Masatoshi Nagamochi","raw_affiliation_strings":["Medicinal Chemistry Reseach Laboratoty, Daiichi Pharmaceutical Co., Ltd, 1-16-13, Kita-Kasai, Edogawa-ku, Tokyo 134-8630, Japan;"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Medicinal Chemistry Reseach Laboratoty, Daiichi Pharmaceutical Co., Ltd, 1-16-13, Kita-Kasai, Edogawa-ku, Tokyo 134-8630, Japan;","institution_ids":[]}]},{"author_position":"middle","author":{"id":null,"display_name":"Ryo Muto","orcid":null,"observed_orcids":[]},"institutions":[],"countries":[],"is_corresponding":false,"raw_author_name":"Ryo Muto","raw_affiliation_strings":["Medicinal Chemistry Reseach Laboratoty, Daiichi Pharmaceutical Co., Ltd, 1-16-13, Kita-Kasai, Edogawa-ku, Tokyo 134-8630, Japan;"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Medicinal Chemistry Reseach Laboratoty, Daiichi Pharmaceutical Co., Ltd, 1-16-13, Kita-Kasai, Edogawa-ku, Tokyo 134-8630, Japan;","institution_ids":[]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5032849902","display_name":"Mitsuhiro Yamaguchi","orcid":"https://orcid.org/0009-0009-7360-8408","observed_orcids":["https://orcid.org/0009-0009-7360-8408"]},"institutions":[],"countries":[],"is_corresponding":false,"raw_author_name":"Mitsuhiro Yamaguchi","raw_affiliation_strings":["Medicinal Chemistry Reseach Laboratoty, Daiichi Pharmaceutical Co., Ltd, 1-16-13, Kita-Kasai, Edogawa-ku, Tokyo 134-8630, Japan;"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Medicinal Chemistry Reseach Laboratoty, Daiichi Pharmaceutical Co., Ltd, 1-16-13, Kita-Kasai, Edogawa-ku, Tokyo 134-8630, Japan;","institution_ids":[]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5020913363","display_name":"Takayasu Nagahara","orcid":null,"observed_orcids":[]},"institutions":[],"countries":[],"is_corresponding":false,"raw_author_name":"Takayasu Nagahara","raw_affiliation_strings":["Medicinal Chemistry Reseach Laboratoty, Daiichi Pharmaceutical Co., Ltd, 1-16-13, Kita-Kasai, Edogawa-ku, Tokyo 134-8630, Japan;"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Medicinal Chemistry Reseach Laboratoty, Daiichi Pharmaceutical Co., Ltd, 1-16-13, Kita-Kasai, Edogawa-ku, Tokyo 134-8630, Japan;","institution_ids":[]}]},{"author_position":"last","author":{"id":"https://openalex.org/A5113478814","display_name":"Hideyuki Kanno","orcid":null,"observed_orcids":[]},"institutions":[],"countries":[],"is_corresponding":false,"raw_author_name":"Hideyuki Kanno","raw_affiliation_strings":["Medicinal Chemistry Reseach Laboratoty, Daiichi Pharmaceutical Co., Ltd, 1-16-13, Kita-Kasai, Edogawa-ku, Tokyo 134-8630, Japan;"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Medicinal Chemistry Reseach Laboratoty, Daiichi Pharmaceutical Co., Ltd, 1-16-13, Kita-Kasai, Edogawa-ku, Tokyo 134-8630, Japan;","institution_ids":[]}]}],"institutions":[],"countries_distinct_count":0,"institutions_distinct_count":0,"corresponding_author_ids":["https://openalex.org/A5043627463"],"corresponding_institution_ids":[],"apc_list":null,"apc_paid":null,"fwci":1.4173,"has_fulltext":false,"cited_by_count":22,"citation_normalized_percentile":{"value":0.78893785,"is_in_top_1_percent":false,"is_in_top_10_percent":false},"cited_by_percentile_year":{"min":88,"max":95},"biblio":{"volume":"63","issue":"7","first_page":"1555","last_page":"1555"},"is_retracted":false,"is_paratext":false,"is_xpac":false,"primary_topic":{"id":"https://openalex.org/T13208","display_name":"Synthesis of heterocyclic compounds","score":0.9345999956130981,"subfield":{"id":"https://openalex.org/subfields/1605","display_name":"Organic Chemistry"},"field":{"id":"https://openalex.org/fields/16","display_name":"Chemistry"},"domain":{"id":"https://openalex.org/domains/3","display_name":"Physical Sciences"}},"topics":[{"id":"https://openalex.org/T13208","display_name":"Synthesis of heterocyclic compounds","score":0.9345999956130981,"subfield":{"id":"https://openalex.org/subfields/1605","display_name":"Organic Chemistry"},"field":{"id":"https://openalex.org/fields/16","display_name":"Chemistry"},"domain":{"id":"https://openalex.org/domains/3","display_name":"Physical Sciences"}},{"id":"https://openalex.org/T10274","display_name":"Heterocyclic Compound Synthesis and Bioactivity","score":0.0142000000923872,"subfield":{"id":"https://openalex.org/subfields/1605","display_name":"Organic Chemistry"},"field":{"id":"https://openalex.org/fields/16","display_name":"Chemistry"},"domain":{"id":"https://openalex.org/domains/3","display_name":"Physical Sciences"}},{"id":"https://openalex.org/T13304","display_name":"Synthesis and Reactivity of Sulfur-Containing Compounds","score":0.013899999670684338,"subfield":{"id":"https://openalex.org/subfields/1605","display_name":"Organic Chemistry"},"field":{"id":"https://openalex.org/fields/16","display_name":"Chemistry"},"domain":{"id":"https://openalex.org/domains/3","display_name":"Physical Sciences"}}],"keywords":[{"id":"https://openalex.org/keywords/lithium-salts","display_name":"lithium salts","score":0.8980000019073486},{"id":"https://openalex.org/keywords/heterocycle-synthesis","display_name":"heterocyclic synthesis","score":0.75},{"id":"https://openalex.org/keywords/large-scale-synthesis","display_name":"large-scale synthesis","score":0.7760000228881836}],"concepts":[{"id":"https://openalex.org/C185592680","wikidata":"https://www.wikidata.org/wiki/Q2329","display_name":"Chemistry","level":0,"score":0.9477380514144897},{"id":"https://openalex.org/C2779485729","wikidata":"https://www.wikidata.org/wiki/Q210385","display_name":"Pyridine","level":2,"score":0.8629241585731506},{"id":"https://openalex.org/C2778541603","wikidata":"https://www.wikidata.org/wiki/Q152763","display_name":"Lithium (medication)","level":2,"score":0.7225713729858398},{"id":"https://openalex.org/C2779074116","wikidata":"https://www.wikidata.org/wiki/Q134856","display_name":"Carboxylic acid","level":2,"score":0.7095282673835754},{"id":"https://openalex.org/C178790620","wikidata":"https://www.wikidata.org/wiki/Q11351","display_name":"Organic chemistry","level":1,"score":0.5014462471008301},{"id":"https://openalex.org/C21951064","wikidata":"https://www.wikidata.org/wiki/Q899212","display_name":"Combinatorial chemistry","level":1,"score":0.47413966059684753},{"id":"https://openalex.org/C71924100","wikidata":"https://www.wikidata.org/wiki/Q11190","display_name":"Medicine","level":0,"score":0.0},{"id":"https://openalex.org/C134018914","wikidata":"https://www.wikidata.org/wiki/Q162606","display_name":"Endocrinology","level":1,"score":0.0}],"mesh":[],"locations_count":1,"locations":[{"id":"doi:10.3987/com-04-10071","doi":"https://doi.org/10.3987/com-04-10071","is_oa":false,"landing_page_url":"https://doi.org/10.3987/com-04-10071","pdf_url":null,"source":{"id":"https://openalex.org/S27298842","display_name":"Heterocycles","issn_l":"0385-5414","issn":["0385-5414","1881-0942"],"is_oa":false,"is_in_doaj":false,"is_core":true,"listed_in":["cwts-core","jufo-1","norway-1","poland-40","russia-white-list-4"],"host_organization":"https://openalex.org/P4310320990","host_organization_name":"Elsevier BV","host_organization_lineage":["https://openalex.org/P4310320990"],"host_organization_lineage_names":["Elsevier BV"],"type":"journal"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"HETEROCYCLES","raw_type":"journal-article"}],"best_oa_location":null,"sustainable_development_goals":[],"study_designs":[],"awards":[],"funders":[],"has_content":{"pdf":false,"grobid_xml":false},"content_urls":null,"referenced_works_count":9,"referenced_works":["https://openalex.org/W1999725694","https://openalex.org/W2004828627","https://openalex.org/W2031069166","https://openalex.org/W2045540776","https://openalex.org/W2047134066","https://openalex.org/W2085501212","https://openalex.org/W2420229086","https://openalex.org/W2421942984","https://openalex.org/W2951390748"],"related_works":["https://openalex.org/W2438497114","https://openalex.org/W2313112919","https://openalex.org/W2072224151","https://openalex.org/W2016934988","https://openalex.org/W2953352701","https://openalex.org/W2114471487","https://openalex.org/W2038522548","https://openalex.org/W1982402328","https://openalex.org/W2000431775","https://openalex.org/W7042467442"],"abstract_inverted_index":{"The":[0],"improved":[1,19],"routes":[2],"to":[3],"prepare":[4],"tetrahydrothiazolo[5,4-c]pyridine-2-carboxylic":[5,35],"acid":[6,36],"lithium":[7],"salts":[8],"(2":[9],"and":[10,24,49],"3)":[11],"were":[12],"developed.Route":[13],"A":[14],"is":[15,27],"consisted":[16],"of":[17,21,34],"the":[18],"preparation":[20],"thiazolopyridine":[22,48],"intermediates,":[23],"Route":[25],"B":[26],"applicable":[28],"for":[29,46],"a":[30],"large":[31],"scale":[32],"synthesis":[33],"derivatives.The":[37],"methods":[38],"we":[39],"developed":[40],"may":[41],"serve":[42],"as":[43],"facile":[44],"means":[45],"preparing":[47],"tetrahydrothiazolopyridine":[50],"derivatives.":[51]},"counts_by_year":[{"year":2026,"cited_by_count":1},{"year":2017,"cited_by_count":1},{"year":2016,"cited_by_count":1},{"year":2014,"cited_by_count":1}],"updated_date":"2026-11-05T12:25:35.769452","created_date":"2019-06-27T00:00:00"}