{"id":"https://openalex.org/W2893045005","doi":"https://doi.org/10.1016/j.poly.2018.09.053","title":"Synthesis, DNA binding, topoisomerase I inhibition and antiproliferation activities of three new binuclear terpyridine platinum(II) complexes","display_name":"Synthesis, DNA binding, topoisomerase I inhibition and antiproliferation activities of three new binuclear terpyridine platinum(II) complexes","publication_year":2018,"publication_date":"2018-09-28","ids":{"openalex":"https://openalex.org/W2893045005","doi":"https://doi.org/10.1016/j.poly.2018.09.053","mag":"2893045005"},"language":"en","primary_location":{"id":"doi:10.1016/j.poly.2018.09.053","doi":"https://doi.org/10.1016/j.poly.2018.09.053","is_oa":false,"landing_page_url":"https://doi.org/10.1016/j.poly.2018.09.053","pdf_url":null,"source":{"id":"https://openalex.org/S171616156","display_name":"Polyhedron","issn_l":"0277-5387","issn":["0277-5387","1873-3719"],"is_oa":false,"is_in_doaj":false,"is_core":true,"listed_in":["anvur-scientific","cwts-core","dongbi-c","jufo-1","norway-1","poland-100","russia-white-list-2"],"host_organization":"https://openalex.org/P4310320990","host_organization_name":"Elsevier BV","host_organization_lineage":["https://openalex.org/P4310320990"],"host_organization_lineage_names":["Elsevier BV"],"type":"journal"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"Polyhedron","raw_type":"journal-article"},"volume":null,"type":"article","is_traditional":true,"indexed_in":["crossref"],"open_access":{"is_oa":false,"oa_status":"closed","oa_url":null,"any_repository_has_fulltext":false},"authorships":[{"author_position":"first","author":{"id":"https://openalex.org/A5114040834","display_name":"Keke Chai","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I41317344","display_name":"Jiangxi Science and Technology Normal University","ror":"https://ror.org/04r1zkp10","country_code":"CN","type":"education","lineage":["https://openalex.org/I41317344"]}],"countries":["CN"],"is_corresponding":false,"raw_author_name":"Keke Chai","raw_affiliation_strings":["Jiangxi Provincial Key Laboratory of Drug Design and Evaluation, School of Pharmacy, Jiangxi Science & Technology Normal University, Nanchang 330013, PR China"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Jiangxi Provincial Key Laboratory of Drug Design and Evaluation, School of Pharmacy, Jiangxi Science & Technology Normal University, Nanchang 330013, PR China","institution_ids":["https://openalex.org/I41317344"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5030478315","display_name":"Yihui Jiang","orcid":"https://orcid.org/0000-0002-6309-2040","observed_orcids":["https://orcid.org/0000-0002-6309-2040"]},"institutions":[{"id":"https://openalex.org/I41317344","display_name":"Jiangxi Science and Technology Normal University","ror":"https://ror.org/04r1zkp10","country_code":"CN","type":"education","lineage":["https://openalex.org/I41317344"]}],"countries":["CN"],"is_corresponding":false,"raw_author_name":"Yihui Jiang","raw_affiliation_strings":["Jiangxi Provincial Key Laboratory of Drug Design and Evaluation, School of Pharmacy, Jiangxi Science & Technology Normal University, Nanchang 330013, PR China"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Jiangxi Provincial Key Laboratory of Drug Design and Evaluation, School of Pharmacy, Jiangxi Science & Technology Normal University, Nanchang 330013, PR China","institution_ids":["https://openalex.org/I41317344"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5044450014","display_name":"Tianzhi Han","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I41317344","display_name":"Jiangxi Science and Technology Normal University","ror":"https://ror.org/04r1zkp10","country_code":"CN","type":"education","lineage":["https://openalex.org/I41317344"]}],"countries":["CN"],"is_corresponding":false,"raw_author_name":"Tianzhi Han","raw_affiliation_strings":["Jiangxi Provincial Key Laboratory of Drug Design and Evaluation, School of Pharmacy, Jiangxi Science & Technology Normal University, Nanchang 330013, PR China"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Jiangxi Provincial Key Laboratory of Drug Design and Evaluation, School of Pharmacy, Jiangxi Science & Technology Normal University, Nanchang 330013, PR China","institution_ids":["https://openalex.org/I41317344"]}]},{"author_position":"middle","author":{"id":null,"display_name":"Junlong Niu","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I41317344","display_name":"Jiangxi Science and Technology Normal University","ror":"https://ror.org/04r1zkp10","country_code":"CN","type":"education","lineage":["https://openalex.org/I41317344"]}],"countries":["CN"],"is_corresponding":false,"raw_author_name":"Junlong Niu","raw_affiliation_strings":["Jiangxi Provincial Key Laboratory of Drug Design and Evaluation, School of Pharmacy, Jiangxi Science & Technology Normal University, Nanchang 330013, PR China"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Jiangxi Provincial Key Laboratory of Drug Design and Evaluation, School of Pharmacy, Jiangxi Science & Technology Normal University, Nanchang 330013, PR China","institution_ids":["https://openalex.org/I41317344"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5054373719","display_name":"Liushuang Yao","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I41317344","display_name":"Jiangxi Science and Technology Normal University","ror":"https://ror.org/04r1zkp10","country_code":"CN","type":"education","lineage":["https://openalex.org/I41317344"]}],"countries":["CN"],"is_corresponding":false,"raw_author_name":"Liushuang Yao","raw_affiliation_strings":["Jiangxi Provincial Key Laboratory of Drug Design and Evaluation, School of Pharmacy, Jiangxi Science & Technology Normal University, Nanchang 330013, PR China"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Jiangxi Provincial Key Laboratory of Drug Design and Evaluation, School of Pharmacy, Jiangxi Science & Technology Normal University, Nanchang 330013, PR China","institution_ids":["https://openalex.org/I41317344"]}]},{"author_position":"middle","author":{"id":null,"display_name":"Haiyu Zhang","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I41317344","display_name":"Jiangxi Science and Technology Normal University","ror":"https://ror.org/04r1zkp10","country_code":"CN","type":"education","lineage":["https://openalex.org/I41317344"]}],"countries":["CN"],"is_corresponding":false,"raw_author_name":"Haiyu Zhang","raw_affiliation_strings":["Jiangxi Provincial Key Laboratory of Drug Design and Evaluation, School of Pharmacy, Jiangxi Science & Technology Normal University, Nanchang 330013, PR China"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Jiangxi Provincial Key Laboratory of Drug Design and Evaluation, School of Pharmacy, Jiangxi Science & Technology Normal University, Nanchang 330013, PR China","institution_ids":["https://openalex.org/I41317344"]}]},{"author_position":"middle","author":{"id":null,"display_name":"Min Zeng","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I41317344","display_name":"Jiangxi Science and Technology Normal University","ror":"https://ror.org/04r1zkp10","country_code":"CN","type":"education","lineage":["https://openalex.org/I41317344"]}],"countries":["CN"],"is_corresponding":false,"raw_author_name":"Min Zeng","raw_affiliation_strings":["Jiangxi Provincial Key Laboratory of Drug Design and Evaluation, School of Pharmacy, Jiangxi Science & Technology Normal University, Nanchang 330013, PR China"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Jiangxi Provincial Key Laboratory of Drug Design and Evaluation, School of Pharmacy, Jiangxi Science & Technology Normal University, Nanchang 330013, PR China","institution_ids":["https://openalex.org/I41317344"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5100425623","display_name":"Li Zhang","orcid":"https://orcid.org/0000-0002-6970-4562","observed_orcids":["https://orcid.org/0000-0002-6970-4562","https://orcid.org/0000-0002-4397-1785"]},"institutions":[{"id":"https://openalex.org/I41317344","display_name":"Jiangxi Science and Technology Normal University","ror":"https://ror.org/04r1zkp10","country_code":"CN","type":"education","lineage":["https://openalex.org/I41317344"]}],"countries":["CN"],"is_corresponding":false,"raw_author_name":"Li Zhang","raw_affiliation_strings":["Jiangxi Provincial Key Laboratory of Drug Design and Evaluation, School of Pharmacy, Jiangxi Science & Technology Normal University, Nanchang 330013, PR China"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Jiangxi Provincial Key Laboratory of Drug Design and Evaluation, School of Pharmacy, Jiangxi Science & Technology Normal University, Nanchang 330013, PR China","institution_ids":["https://openalex.org/I41317344"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5032132780","display_name":"Xuemin Duan","orcid":"https://orcid.org/0000-0001-9636-1297","observed_orcids":["https://orcid.org/0000-0001-9636-1297"]},"institutions":[{"id":"https://openalex.org/I41317344","display_name":"Jiangxi Science and Technology Normal University","ror":"https://ror.org/04r1zkp10","country_code":"CN","type":"education","lineage":["https://openalex.org/I41317344"]}],"countries":["CN"],"is_corresponding":true,"raw_author_name":"Xuemin Duan","raw_affiliation_strings":["Jiangxi Provincial Key Laboratory of Drug Design and Evaluation, School of Pharmacy, Jiangxi Science & Technology Normal University, Nanchang 330013, PR China"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Jiangxi Provincial Key Laboratory of Drug Design and Evaluation, School of Pharmacy, Jiangxi Science & Technology Normal University, Nanchang 330013, PR China","institution_ids":["https://openalex.org/I41317344"]}]},{"author_position":"last","author":{"id":"https://openalex.org/A5100379896","display_name":"Jintao Wang","orcid":"https://orcid.org/0000-0003-4489-5531","observed_orcids":["https://orcid.org/0000-0003-4489-5531"]},"institutions":[{"id":"https://openalex.org/I41317344","display_name":"Jiangxi Science and Technology Normal University","ror":"https://ror.org/04r1zkp10","country_code":"CN","type":"education","lineage":["https://openalex.org/I41317344"]}],"countries":["CN"],"is_corresponding":true,"raw_author_name":"Jintao Wang","raw_affiliation_strings":["Jiangxi Provincial Key Laboratory of Drug Design and Evaluation, School of Pharmacy, Jiangxi Science & Technology Normal University, Nanchang 330013, PR China"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Jiangxi Provincial Key Laboratory of Drug Design and Evaluation, School of Pharmacy, Jiangxi Science & Technology Normal University, Nanchang 330013, PR China","institution_ids":["https://openalex.org/I41317344"]}]}],"institutions":[],"countries_distinct_count":1,"institutions_distinct_count":1,"corresponding_author_ids":["https://openalex.org/A5032132780","https://openalex.org/A5100379896"],"corresponding_institution_ids":["https://openalex.org/I41317344"],"apc_list":{"value":3740,"currency":"USD","value_usd":3740},"apc_paid":null,"fwci":0.8346,"has_fulltext":false,"cited_by_count":16,"citation_normalized_percentile":{"value":0.74194872,"is_in_top_1_percent":false,"is_in_top_10_percent":false},"cited_by_percentile_year":{"min":88,"max":96},"biblio":{"volume":"157","issue":null,"first_page":"124","last_page":"130"},"is_retracted":false,"is_paratext":false,"is_xpac":false,"primary_topic":{"id":"https://openalex.org/T10163","display_name":"Metal complexes synthesis and properties","score":0.9994999766349792,"subfield":{"id":"https://openalex.org/subfields/2730","display_name":"Oncology"},"field":{"id":"https://openalex.org/fields/27","display_name":"Medicine"},"domain":{"id":"https://openalex.org/domains/4","display_name":"Health Sciences"}},"topics":[{"id":"https://openalex.org/T10163","display_name":"Metal complexes synthesis and properties","score":0.9994999766349792,"subfield":{"id":"https://openalex.org/subfields/2730","display_name":"Oncology"},"field":{"id":"https://openalex.org/fields/27","display_name":"Medicine"},"domain":{"id":"https://openalex.org/domains/4","display_name":"Health Sciences"}},{"id":"https://openalex.org/T11845","display_name":"Cancer therapeutics and mechanisms","score":0.0003000000142492354,"subfield":{"id":"https://openalex.org/subfields/1312","display_name":"Molecular Biology"},"field":{"id":"https://openalex.org/fields/13","display_name":"Biochemistry, Genetics and Molecular Biology"},"domain":{"id":"https://openalex.org/domains/1","display_name":"Life Sciences"}},{"id":"https://openalex.org/T13105","display_name":"Synthesis and pharmacology of benzodiazepine derivatives","score":0.0,"subfield":{"id":"https://openalex.org/subfields/1605","display_name":"Organic Chemistry"},"field":{"id":"https://openalex.org/fields/16","display_name":"Chemistry"},"domain":{"id":"https://openalex.org/domains/3","display_name":"Physical Sciences"}}],"keywords":[{"id":"https://openalex.org/keywords/binuclear-platinum-ii-complexes","display_name":"binuclear platinum(II) complexes","score":0.9860000014305115},{"id":"https://openalex.org/keywords/terpyridyl-ligands","display_name":"terpyridine ligands","score":0.9760000109672546},{"id":"https://openalex.org/keywords/dna-binding","display_name":"DNA binding","score":0.8759999871253967},{"id":"https://openalex.org/keywords/topoisomerase-i-inhibition","display_name":"topoisomerase I inhibition","score":0.9990000128746033},{"id":"https://openalex.org/keywords/antiproliferative-activity","display_name":"antiproliferative activity","score":0.9810000061988831},{"id":"https://openalex.org/keywords/pi-pi-stacking","display_name":"\u03c0-\u03c0 stacking","score":0.734000027179718},{"id":"https://openalex.org/keywords/ethidium-bromide-displacement","display_name":"ethidium bromide displacement","score":0.8560000061988831},{"id":"https://openalex.org/keywords/cytotoxicity","display_name":"cytotoxicity","score":0.7710000276565552},{"id":"https://openalex.org/keywords/platinum-based-anticancer-drugs","display_name":"platinum anticancer drugs","score":0.6129999756813049}],"concepts":[{"id":"https://openalex.org/C185592680","wikidata":"https://www.wikidata.org/wiki/Q2329","display_name":"Chemistry","level":0,"score":0.9341527819633484},{"id":"https://openalex.org/C2776907736","wikidata":"https://www.wikidata.org/wiki/Q408634","display_name":"Ethidium bromide","level":3,"score":0.7726874351501465},{"id":"https://openalex.org/C147897179","wikidata":"https://www.wikidata.org/wiki/Q407828","display_name":"Topoisomerase","level":3,"score":0.6725993156433105},{"id":"https://openalex.org/C2778271344","wikidata":"https://www.wikidata.org/wiki/Q903395","display_name":"Agarose gel electrophoresis","level":3,"score":0.6350146532058716},{"id":"https://openalex.org/C552990157","wikidata":"https://www.wikidata.org/wiki/Q7430","display_name":"DNA","level":2,"score":0.6322599649429321},{"id":"https://openalex.org/C2781350956","wikidata":"https://www.wikidata.org/wiki/Q408228","display_name":"Terpyridine","level":3,"score":0.6010972261428833},{"id":"https://openalex.org/C71240020","wikidata":"https://www.wikidata.org/wiki/Q186011","display_name":"Stereochemistry","level":1,"score":0.5262643098831177},{"id":"https://openalex.org/C137824038","wikidata":"https://www.wikidata.org/wiki/Q175562","display_name":"Intercalation (chemistry)","level":2,"score":0.472102552652359},{"id":"https://openalex.org/C8010536","wikidata":"https://www.wikidata.org/wiki/Q160398","display_name":"Crystallography","level":1,"score":0.4652135670185089},{"id":"https://openalex.org/C32786932","wikidata":"https://www.wikidata.org/wiki/Q4914013","display_name":"Binding constant","level":3,"score":0.4509822130203247},{"id":"https://openalex.org/C116084860","wikidata":"https://www.wikidata.org/wiki/Q48255","display_name":"Gel electrophoresis","level":2,"score":0.42488405108451843},{"id":"https://openalex.org/C107824862","wikidata":"https://www.wikidata.org/wiki/Q616005","display_name":"Binding site","level":2,"score":0.29414451122283936},{"id":"https://openalex.org/C544153396","wikidata":"https://www.wikidata.org/wiki/Q11426","display_name":"Metal","level":2,"score":0.20389986038208008},{"id":"https://openalex.org/C55493867","wikidata":"https://www.wikidata.org/wiki/Q7094","display_name":"Biochemistry","level":1,"score":0.11942499876022339},{"id":"https://openalex.org/C179104552","wikidata":"https://www.wikidata.org/wiki/Q11165","display_name":"Inorganic chemistry","level":1,"score":0.0886603593826294},{"id":"https://openalex.org/C178790620","wikidata":"https://www.wikidata.org/wiki/Q11351","display_name":"Organic chemistry","level":1,"score":0.0}],"mesh":[],"locations_count":1,"locations":[{"id":"doi:10.1016/j.poly.2018.09.053","doi":"https://doi.org/10.1016/j.poly.2018.09.053","is_oa":false,"landing_page_url":"https://doi.org/10.1016/j.poly.2018.09.053","pdf_url":null,"source":{"id":"https://openalex.org/S171616156","display_name":"Polyhedron","issn_l":"0277-5387","issn":["0277-5387","1873-3719"],"is_oa":false,"is_in_doaj":false,"is_core":true,"listed_in":["anvur-scientific","cwts-core","dongbi-c","jufo-1","norway-1","poland-100","russia-white-list-2"],"host_organization":"https://openalex.org/P4310320990","host_organization_name":"Elsevier BV","host_organization_lineage":["https://openalex.org/P4310320990"],"host_organization_lineage_names":["Elsevier BV"],"type":"journal"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"Polyhedron","raw_type":"journal-article"}],"best_oa_location":null,"sustainable_development_goals":[],"study_designs":[],"awards":[{"id":"https://openalex.org/G6216533392","display_name":null,"funder_award_id":"20171103057","funder_id":"https://openalex.org/F4320328114","funder_display_name":"Jiangxi Science and Technology Normal University"},{"id":"https://openalex.org/G6805409452","display_name":null,"funder_award_id":"21401105","funder_id":"https://openalex.org/F4320321001","funder_display_name":"National Natural Science Foundation of China"},{"id":"https://openalex.org/G7513271662","display_name":null,"funder_award_id":"GJJ170695","funder_id":"https://openalex.org/F4320325626","funder_display_name":"Education Department of Jiangxi Province"},{"id":"https://openalex.org/G8501469122","display_name":null,"funder_award_id":"20181BAB213001","funder_id":"https://openalex.org/F4320322665","funder_display_name":"Natural Science Foundation of Jiangxi Province"},{"id":"https://openalex.org/G958686652","display_name":null,"funder_award_id":"3000990404","funder_id":"https://openalex.org/F4320328114","funder_display_name":"Jiangxi Science and Technology Normal University"}],"funders":[{"id":"https://openalex.org/F4320321001","display_name":"National Natural Science Foundation of China","ror":"https://ror.org/01h0zpd94"},{"id":"https://openalex.org/F4320322665","display_name":"Natural Science Foundation of Jiangxi Province","ror":null},{"id":"https://openalex.org/F4320325626","display_name":"Education Department of Jiangxi Province","ror":"https://ror.org/04d8xwh61"},{"id":"https://openalex.org/F4320328114","display_name":"Jiangxi Science and Technology Normal University","ror":"https://ror.org/04r1zkp10"}],"has_content":{"pdf":false,"grobid_xml":false},"content_urls":null,"referenced_works_count":36,"referenced_works":["https://openalex.org/W1590106897","https://openalex.org/W1969360633","https://openalex.org/W1984345087","https://openalex.org/W1984790214","https://openalex.org/W1993837819","https://openalex.org/W1995837528","https://openalex.org/W2007036666","https://openalex.org/W2012108057","https://openalex.org/W2013542366","https://openalex.org/W2035130691","https://openalex.org/W2038822441","https://openalex.org/W2043465974","https://openalex.org/W2048008698","https://openalex.org/W2055575798","https://openalex.org/W2063196204","https://openalex.org/W2064367068","https://openalex.org/W2065630179","https://openalex.org/W2067878166","https://openalex.org/W2077183901","https://openalex.org/W2089731664","https://openalex.org/W2090537798","https://openalex.org/W2092522778","https://openalex.org/W2093500137","https://openalex.org/W2126695283","https://openalex.org/W2167229423","https://openalex.org/W2169171285","https://openalex.org/W2198448841","https://openalex.org/W2216339699","https://openalex.org/W2270272511","https://openalex.org/W2287841932","https://openalex.org/W2340670430","https://openalex.org/W2419256959","https://openalex.org/W2512718425","https://openalex.org/W2549858084","https://openalex.org/W2588137061","https://openalex.org/W3137139169"],"related_works":["https://openalex.org/W2905555534","https://openalex.org/W2810731610","https://openalex.org/W2151196136","https://openalex.org/W2186804847","https://openalex.org/W2035495580","https://openalex.org/W2895928456","https://openalex.org/W2562308922","https://openalex.org/W2095282865","https://openalex.org/W2172400360","https://openalex.org/W1968735393"],"abstract_inverted_index":null,"counts_by_year":[{"year":2026,"cited_by_count":1},{"year":2024,"cited_by_count":2},{"year":2023,"cited_by_count":2},{"year":2022,"cited_by_count":3},{"year":2021,"cited_by_count":2},{"year":2020,"cited_by_count":3},{"year":2019,"cited_by_count":2},{"year":2018,"cited_by_count":1}],"updated_date":"2026-11-04T10:54:05.112534","created_date":"2018-10-05T00:00:00"}
