{"id":"https://openalex.org/W2803607030","doi":"https://doi.org/10.1016/j.bmc.2018.05.023","title":"Chiral analogues of (+)-cyclazosin as potent \u03b11B-adrenoceptor selective antagonist","display_name":"Chiral analogues of (+)-cyclazosin as potent \u03b11B-adrenoceptor selective antagonist","publication_year":2018,"publication_date":"2018-05-17","ids":{"openalex":"https://openalex.org/W2803607030","doi":"https://doi.org/10.1016/j.bmc.2018.05.023","mag":"2803607030","pmid":"https://pubmed.ncbi.nlm.nih.gov/29784274","pmcid":"https://www.ncbi.nlm.nih.gov/pmc/articles/6008244"},"language":"en","primary_location":{"id":"doi:10.1016/j.bmc.2018.05.023","doi":"https://doi.org/10.1016/j.bmc.2018.05.023","is_oa":true,"landing_page_url":"https://doi.org/10.1016/j.bmc.2018.05.023","pdf_url":null,"source":{"id":"https://openalex.org/S10422866","display_name":"Bioorganic & Medicinal Chemistry","issn_l":"0968-0896","issn":["0968-0896","1464-3391"],"is_oa":false,"is_in_doaj":false,"is_core":true,"listed_in":["anvur-scientific","cwts-core","dongbi-c","doyens","jufo-1","ki-jl-1","medline","norway-1","poland-70","russia-white-list-1","vabb-shw"],"host_organization":"https://openalex.org/P4310320990","host_organization_name":"Elsevier BV","host_organization_lineage":["https://openalex.org/P4310320990"],"host_organization_lineage_names":["Elsevier BV"],"type":"journal"},"license":null,"license_id":null,"version":"acceptedVersion","is_accepted":true,"is_published":false,"raw_source_name":"Bioorganic &amp; Medicinal Chemistry","raw_type":"journal-article"},"volume":null,"type":"article","indexed_in":["crossref","pubmed"],"open_access":{"is_oa":true,"oa_status":"bronze","oa_url":"https://doi.org/10.1016/j.bmc.2018.05.023","any_repository_has_fulltext":true},"authorships":[{"author_position":"first","author":{"id":"https://openalex.org/A5032672040","display_name":"Gianni Sagratini","orcid":"https://orcid.org/0000-0001-6231-8709","observed_orcids":["https://orcid.org/0000-0001-6231-8709"]},"institutions":[{"id":"https://openalex.org/I112859197","display_name":"Universit\u00e0 di Camerino","ror":"https://ror.org/0005w8d69","country_code":"IT","type":"education","lineage":["https://openalex.org/I112859197"]}],"countries":["IT"],"is_corresponding":true,"raw_author_name":"Gianni Sagratini","raw_affiliation_strings":["Scuola in Scienze del Farmaco e dei Prodotti della Salute, Universit\u00e0 di Camerino, Via S. Agostino 1, 62032 Camerino, Italy. Electronic address: gianni.sagratini@unicam.it","Scuola in Scienze del Farmaco e dei Prodotti della Salute, Universit\u00e0 di Camerino, Via S. Agostino 1, 62032 Camerino, Italy"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Scuola in Scienze del Farmaco e dei Prodotti della Salute, Universit\u00e0 di Camerino, Via S. Agostino 1, 62032 Camerino, Italy. Electronic address: gianni.sagratini@unicam.it","institution_ids":["https://openalex.org/I112859197"]},{"raw_affiliation_string":"Scuola in Scienze del Farmaco e dei Prodotti della Salute, Universit\u00e0 di Camerino, Via S. Agostino 1, 62032 Camerino, Italy","institution_ids":["https://openalex.org/I112859197"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5048593211","display_name":"Michela Buccioni","orcid":"https://orcid.org/0000-0002-8383-0813","observed_orcids":["https://orcid.org/0000-0002-8383-0813"]},"institutions":[{"id":"https://openalex.org/I112859197","display_name":"Universit\u00e0 di Camerino","ror":"https://ror.org/0005w8d69","country_code":"IT","type":"education","lineage":["https://openalex.org/I112859197"]}],"countries":["IT"],"is_corresponding":false,"raw_author_name":"Michela Buccioni","raw_affiliation_strings":["Scuola in Scienze del Farmaco e dei Prodotti della Salute, Universit\u00e0 di Camerino, Via S. Agostino 1, 62032 Camerino, Italy"],"raw_orcid":"https://orcid.org/0000-0002-8383-0813","affiliations":[{"raw_affiliation_string":"Scuola in Scienze del Farmaco e dei Prodotti della Salute, Universit\u00e0 di Camerino, Via S. Agostino 1, 62032 Camerino, Italy","institution_ids":["https://openalex.org/I112859197"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5067731409","display_name":"Gabriella Marucci","orcid":"https://orcid.org/0000-0002-9856-9873","observed_orcids":["https://orcid.org/0000-0002-9856-9873"]},"institutions":[{"id":"https://openalex.org/I112859197","display_name":"Universit\u00e0 di Camerino","ror":"https://ror.org/0005w8d69","country_code":"IT","type":"education","lineage":["https://openalex.org/I112859197"]}],"countries":["IT"],"is_corresponding":false,"raw_author_name":"Gabriella Marucci","raw_affiliation_strings":["Scuola in Scienze del Farmaco e dei Prodotti della Salute, Universit\u00e0 di Camerino, Via S. Agostino 1, 62032 Camerino, Italy"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Scuola in Scienze del Farmaco e dei Prodotti della Salute, Universit\u00e0 di Camerino, Via S. Agostino 1, 62032 Camerino, Italy","institution_ids":["https://openalex.org/I112859197"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5054132162","display_name":"Elena Poggesi","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I4210134517","display_name":"Recordati (Italy)","ror":"https://ror.org/03ekprg18","country_code":"IT","type":"company","lineage":["https://openalex.org/I4210134517"]}],"countries":["IT"],"is_corresponding":false,"raw_author_name":"Elena Poggesi","raw_affiliation_strings":["Drug Discovery Division, Recordati SpA, Via Civitali 1, 20148 Milano, Italy"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Drug Discovery Division, Recordati SpA, Via Civitali 1, 20148 Milano, Italy","institution_ids":["https://openalex.org/I4210134517"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5052592114","display_name":"Matthew Skorski","orcid":"https://orcid.org/0000-0003-1114-2509","observed_orcids":["https://orcid.org/0000-0003-1114-2509"]},"institutions":[{"id":"https://openalex.org/I181401687","display_name":"American University","ror":"https://ror.org/052w4zt36","country_code":"US","type":"education","lineage":["https://openalex.org/I181401687"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"Matthew Skorski","raw_affiliation_strings":["Department of Chemistry, American University, Washington, DC 20016, USA"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Department of Chemistry, American University, Washington, DC 20016, USA","institution_ids":["https://openalex.org/I181401687"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5021219075","display_name":"Stefano Costanzi","orcid":"https://orcid.org/0000-0003-3183-7332","observed_orcids":["https://orcid.org/0000-0003-3183-7332"]},"institutions":[{"id":"https://openalex.org/I181401687","display_name":"American University","ror":"https://ror.org/052w4zt36","country_code":"US","type":"education","lineage":["https://openalex.org/I181401687"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"Stefano Costanzi","raw_affiliation_strings":["Department of Chemistry, American University, Washington, DC 20016, USA; Center for Behavioral Neuroscience, American University, Washington, DC 20016, USA","Center for Behavioral Neuroscience, American University, Washington, DC 20016, USA","Department of Chemistry, American University, Washington, DC 20016, USA"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Department of Chemistry, American University, Washington, DC 20016, USA; Center for Behavioral Neuroscience, American University, Washington, DC 20016, USA","institution_ids":["https://openalex.org/I181401687"]},{"raw_affiliation_string":"Center for Behavioral Neuroscience, American University, Washington, DC 20016, USA","institution_ids":["https://openalex.org/I181401687"]},{"raw_affiliation_string":"Department of Chemistry, American University, Washington, DC 20016, USA","institution_ids":["https://openalex.org/I181401687"]}]},{"author_position":"last","author":{"id":"https://openalex.org/A5069538779","display_name":"Dario Giardin\u00e0","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I112859197","display_name":"Universit\u00e0 di Camerino","ror":"https://ror.org/0005w8d69","country_code":"IT","type":"education","lineage":["https://openalex.org/I112859197"]}],"countries":["IT"],"is_corresponding":false,"raw_author_name":"Dario Giardin\u00e0","raw_affiliation_strings":["Scuola in Scienze del Farmaco e dei Prodotti della Salute, Universit\u00e0 di Camerino, Via S. Agostino 1, 62032 Camerino, Italy"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Scuola in Scienze del Farmaco e dei Prodotti della Salute, Universit\u00e0 di Camerino, Via S. Agostino 1, 62032 Camerino, Italy","institution_ids":["https://openalex.org/I112859197"]}]}],"institutions":[],"countries_distinct_count":2,"institutions_distinct_count":3,"corresponding_author_ids":["https://openalex.org/A5032672040"],"corresponding_institution_ids":["https://openalex.org/I112859197"],"apc_list":{"value":3960,"currency":"USD","value_usd":3960},"apc_paid":null,"fwci":0.2666,"has_fulltext":false,"cited_by_count":5,"citation_normalized_percentile":{"value":0.50063179,"is_in_top_1_percent":false,"is_in_top_10_percent":false},"cited_by_percentile_year":{"min":88,"max":96},"biblio":{"volume":"26","issue":"12","first_page":"3502","last_page":"3513"},"is_retracted":false,"is_paratext":false,"is_xpac":false,"primary_topic":{"id":"https://openalex.org/T11178","display_name":"Receptor Mechanisms and Signaling","score":0.9740999937057495,"subfield":{"id":"https://openalex.org/subfields/1312","display_name":"Molecular Biology"},"field":{"id":"https://openalex.org/fields/13","display_name":"Biochemistry, Genetics and Molecular Biology"},"domain":{"id":"https://openalex.org/domains/1","display_name":"Life Sciences"}},"topics":[{"id":"https://openalex.org/T11178","display_name":"Receptor Mechanisms and Signaling","score":0.9740999937057495,"subfield":{"id":"https://openalex.org/subfields/1312","display_name":"Molecular Biology"},"field":{"id":"https://openalex.org/fields/13","display_name":"Biochemistry, Genetics and Molecular Biology"},"domain":{"id":"https://openalex.org/domains/1","display_name":"Life Sciences"}},{"id":"https://openalex.org/T13160","display_name":"Synthesis and Biological Evaluation","score":0.008999999612569809,"subfield":{"id":"https://openalex.org/subfields/1605","display_name":"Organic Chemistry"},"field":{"id":"https://openalex.org/fields/16","display_name":"Chemistry"},"domain":{"id":"https://openalex.org/domains/3","display_name":"Physical Sciences"}},{"id":"https://openalex.org/T10274","display_name":"Synthesis and biological activity","score":0.004600000102072954,"subfield":{"id":"https://openalex.org/subfields/1605","display_name":"Organic Chemistry"},"field":{"id":"https://openalex.org/fields/16","display_name":"Chemistry"},"domain":{"id":"https://openalex.org/domains/3","display_name":"Physical Sciences"}}],"keywords":[{"id":"https://openalex.org/keywords/alpha1b-adrenoceptor","display_name":"alpha1B-adrenoceptor","score":0.8460000157356262},{"id":"https://openalex.org/keywords/adrenergic-antagonists","display_name":"adrenergic antagonists","score":0.6650000214576721},{"id":"https://openalex.org/keywords/stereochemistry","display_name":"stereochemistry","score":0.5289999842643738},{"id":"https://openalex.org/keywords/receptor-selectivity","display_name":"receptor selectivity","score":0.7009999752044678},{"id":"https://openalex.org/keywords/molecular-modeling","display_name":"molecular modeling","score":0.6600000262260437}],"concepts":[{"id":"https://openalex.org/C185592680","wikidata":"https://www.wikidata.org/wiki/Q2329","display_name":"Chemistry","level":0,"score":0.9294419288635254},{"id":"https://openalex.org/C118792377","wikidata":"https://www.wikidata.org/wiki/Q108584245","display_name":"Selectivity","level":3,"score":0.8809635639190674},{"id":"https://openalex.org/C2776568683","wikidata":"https://www.wikidata.org/wiki/Q23005640","display_name":"Moiety","level":2,"score":0.7377170920372009},{"id":"https://openalex.org/C71240020","wikidata":"https://www.wikidata.org/wiki/Q186011","display_name":"Stereochemistry","level":1,"score":0.7374101281166077},{"id":"https://openalex.org/C486523","wikidata":"https://www.wikidata.org/wiki/Q494483","display_name":"Enantiomer","level":2,"score":0.7188725471496582},{"id":"https://openalex.org/C131779359","wikidata":"https://www.wikidata.org/wiki/Q471875","display_name":"Amine gas treating","level":2,"score":0.5645052790641785},{"id":"https://openalex.org/C2776885963","wikidata":"https://www.wikidata.org/wiki/Q245204","display_name":"Antagonist","level":3,"score":0.5001881122589111},{"id":"https://openalex.org/C178910836","wikidata":"https://www.wikidata.org/wiki/Q2196961","display_name":"Molecular model","level":2,"score":0.4594572186470032},{"id":"https://openalex.org/C193042331","wikidata":"https://www.wikidata.org/wiki/Q1772003","display_name":"Structure\u2013activity relationship","level":3,"score":0.45628225803375244},{"id":"https://openalex.org/C3018358672","wikidata":"https://www.wikidata.org/wiki/Q167198","display_name":"Tertiary amine","level":2,"score":0.4291543662548065},{"id":"https://openalex.org/C170493617","wikidata":"https://www.wikidata.org/wiki/Q208467","display_name":"Receptor","level":2,"score":0.22734349966049194},{"id":"https://openalex.org/C202751555","wikidata":"https://www.wikidata.org/wiki/Q221681","display_name":"In vitro","level":2,"score":0.17237353324890137},{"id":"https://openalex.org/C55493867","wikidata":"https://www.wikidata.org/wiki/Q7094","display_name":"Biochemistry","level":1,"score":0.12328314781188965},{"id":"https://openalex.org/C178790620","wikidata":"https://www.wikidata.org/wiki/Q11351","display_name":"Organic chemistry","level":1,"score":0.07488152384757996},{"id":"https://openalex.org/C161790260","wikidata":"https://www.wikidata.org/wiki/Q82264","display_name":"Catalysis","level":2,"score":0.0}],"mesh":[{"descriptor_ui":"D000818","descriptor_name":"Animals","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D001011","descriptor_name":"Aorta","qualifier_ui":"Q000378","qualifier_name":"metabolism","is_major_topic":false},{"descriptor_ui":"D001665","descriptor_name":"Binding Sites","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D007700","descriptor_name":"Kinetics","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D008297","descriptor_name":"Male","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D011799","descriptor_name":"Quinazolines","qualifier_ui":"Q000138","qualifier_name":"chemical synthesis","is_major_topic":false},{"descriptor_ui":"D011799","descriptor_name":"Quinazolines","qualifier_ui":"Q000378","qualifier_name":"metabolism","is_major_topic":false},{"descriptor_ui":"D011799","descriptor_name":"Quinazolines","qualifier_ui":"Q000737","qualifier_name":"chemistry","is_major_topic":true},{"descriptor_ui":"D011810","descriptor_name":"Quinoxalines","qualifier_ui":"Q000138","qualifier_name":"chemical synthesis","is_major_topic":false},{"descriptor_ui":"D011810","descriptor_name":"Quinoxalines","qualifier_ui":"Q000378","qualifier_name":"metabolism","is_major_topic":false},{"descriptor_ui":"D011810","descriptor_name":"Quinoxalines","qualifier_ui":"Q000737","qualifier_name":"chemistry","is_major_topic":true},{"descriptor_ui":"D013154","descriptor_name":"Spleen","qualifier_ui":"Q000378","qualifier_name":"metabolism","is_major_topic":false},{"descriptor_ui":"D013237","descriptor_name":"Stereoisomerism","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D017208","descriptor_name":"Rats, Wistar","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D017434","descriptor_name":"Protein Structure, Tertiary","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D018340","descriptor_name":"Receptors, Adrenergic, alpha-1","qualifier_ui":"Q000378","qualifier_name":"metabolism","is_major_topic":true},{"descriptor_ui":"D018340","descriptor_name":"Receptors, Adrenergic, alpha-1","qualifier_ui":"Q000737","qualifier_name":"chemistry","is_major_topic":false},{"descriptor_ui":"D051381","descriptor_name":"Rats","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D056004","descriptor_name":"Molecular Dynamics Simulation","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D058668","descriptor_name":"Adrenergic alpha-1 Receptor Antagonists","qualifier_ui":"Q000138","qualifier_name":"chemical synthesis","is_major_topic":false},{"descriptor_ui":"D058668","descriptor_name":"Adrenergic alpha-1 Receptor Antagonists","qualifier_ui":"Q000378","qualifier_name":"metabolism","is_major_topic":false},{"descriptor_ui":"D058668","descriptor_name":"Adrenergic alpha-1 Receptor Antagonists","qualifier_ui":"Q000737","qualifier_name":"chemistry","is_major_topic":true}],"locations_count":5,"locations":[{"id":"doi:10.1016/j.bmc.2018.05.023","doi":"https://doi.org/10.1016/j.bmc.2018.05.023","is_oa":true,"landing_page_url":"https://doi.org/10.1016/j.bmc.2018.05.023","pdf_url":null,"source":{"id":"https://openalex.org/S10422866","display_name":"Bioorganic & Medicinal Chemistry","issn_l":"0968-0896","issn":["0968-0896","1464-3391"],"is_oa":false,"is_in_doaj":false,"is_core":true,"listed_in":["anvur-scientific","cwts-core","dongbi-c","doyens","jufo-1","ki-jl-1","medline","norway-1","poland-70","russia-white-list-1","vabb-shw"],"host_organization":"https://openalex.org/P4310320990","host_organization_name":"Elsevier BV","host_organization_lineage":["https://openalex.org/P4310320990"],"host_organization_lineage_names":["Elsevier BV"],"type":"journal"},"license":null,"license_id":null,"version":"acceptedVersion","is_accepted":true,"is_published":false,"raw_source_name":"Bioorganic &amp; Medicinal Chemistry","raw_type":"journal-article"},{"id":"pmid:29784274","doi":null,"is_oa":false,"landing_page_url":"https://pubmed.ncbi.nlm.nih.gov/29784274","pdf_url":null,"source":{"id":"https://openalex.org/S4306525036","display_name":"PubMed","issn_l":null,"issn":null,"is_oa":false,"is_in_doaj":false,"is_core":false,"listed_in":[],"host_organization":"https://openalex.org/I1299303238","host_organization_name":"National Institutes of Health","host_organization_lineage":["https://openalex.org/I1299303238"],"host_organization_lineage_names":[],"type":"repository"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"Bioorganic & medicinal chemistry","raw_type":"Journal Article"},{"id":"pmh:oai:europepmc.org:5600028","doi":null,"is_oa":true,"landing_page_url":"https://www.ncbi.nlm.nih.gov/pmc/articles/6008244","pdf_url":null,"source":{"id":"https://openalex.org/S4306400806","display_name":"Europe PMC (PubMed Central)","issn_l":null,"issn":null,"is_oa":false,"is_in_doaj":false,"is_core":false,"listed_in":[],"host_organization":"https://openalex.org/I1303153112","host_organization_name":"European Bioinformatics Institute","host_organization_lineage":["https://openalex.org/I1303153112"],"host_organization_lineage_names":[],"type":"repository"},"license":null,"license_id":null,"version":"acceptedVersion","is_accepted":true,"is_published":false,"raw_source_name":null,"raw_type":"Text"},{"id":"pmh:oai:pubmedcentral.nih.gov:6008244","doi":null,"is_oa":true,"landing_page_url":"https://www.ncbi.nlm.nih.gov/pmc/articles/6008244","pdf_url":null,"source":{"id":"https://openalex.org/S2764455111","display_name":"PubMed Central","issn_l":null,"issn":null,"is_oa":true,"is_in_doaj":false,"is_core":false,"listed_in":[],"host_organization":"https://openalex.org/I1299303238","host_organization_name":"National Institutes of Health","host_organization_lineage":["https://openalex.org/I1299303238"],"host_organization_lineage_names":[],"type":"repository"},"license":null,"license_id":null,"version":"acceptedVersion","is_accepted":true,"is_published":false,"raw_source_name":"Bioorg Med Chem","raw_type":"Text"},{"id":"pmh:oai:pubblicazioni.unicam.it:11581/427365","doi":null,"is_oa":false,"landing_page_url":"http://hdl.handle.net/11581/427365","pdf_url":null,"source":{"id":"https://openalex.org/S4306400819","display_name":"Unicam Scientific Publications (University of Camerino)","issn_l":null,"issn":null,"is_oa":false,"is_in_doaj":false,"is_core":false,"listed_in":[],"host_organization":"https://openalex.org/I112859197","host_organization_name":"Universit\u00e0 di Camerino","host_organization_lineage":["https://openalex.org/I112859197"],"host_organization_lineage_names":[],"type":"repository"},"license":null,"license_id":null,"version":"submittedVersion","is_accepted":false,"is_published":false,"raw_source_name":null,"raw_type":"info:eu-repo/semantics/article"}],"best_oa_location":{"id":"doi:10.1016/j.bmc.2018.05.023","doi":"https://doi.org/10.1016/j.bmc.2018.05.023","is_oa":true,"landing_page_url":"https://doi.org/10.1016/j.bmc.2018.05.023","pdf_url":null,"source":{"id":"https://openalex.org/S10422866","display_name":"Bioorganic & Medicinal Chemistry","issn_l":"0968-0896","issn":["0968-0896","1464-3391"],"is_oa":false,"is_in_doaj":false,"is_core":true,"listed_in":["anvur-scientific","cwts-core","dongbi-c","doyens","jufo-1","ki-jl-1","medline","norway-1","poland-70","russia-white-list-1","vabb-shw"],"host_organization":"https://openalex.org/P4310320990","host_organization_name":"Elsevier BV","host_organization_lineage":["https://openalex.org/P4310320990"],"host_organization_lineage_names":["Elsevier BV"],"type":"journal"},"license":null,"license_id":null,"version":"acceptedVersion","is_accepted":true,"is_published":false,"raw_source_name":"Bioorganic &amp; Medicinal Chemistry","raw_type":"journal-article"},"sustainable_development_goals":[],"study_designs":[],"awards":[{"id":"https://openalex.org/G4608142559","display_name":"MRI:  Acquisition of HPC at AU (Expanding Capabilities for Research and Research Training at American University through Shared High-Performance Computing)","funder_award_id":"1039497","funder_id":"https://openalex.org/F4320306076","funder_display_name":"National Science Foundation"},{"id":"https://openalex.org/G6824874546","display_name":"Enabling the application of Virtual Screening to GPCR Homology Models","funder_award_id":"R15GM119084","funder_id":"https://openalex.org/F4320337354","funder_display_name":"National Institute of General Medical Sciences"}],"funders":[{"id":"https://openalex.org/F4320306076","display_name":"National Science Foundation","ror":"https://ror.org/021nxhr62"},{"id":"https://openalex.org/F4320326607","display_name":"Universit\u00e0 degli Studi di Camerino","ror":"https://ror.org/0005w8d69"},{"id":"https://openalex.org/F4320337354","display_name":"National Institute of General Medical Sciences","ror":"https://ror.org/04q48ey07"}],"has_content":{"grobid_xml":false,"pdf":false},"content_urls":null,"referenced_works_count":39,"referenced_works":["https://openalex.org/W44420309","https://openalex.org/W148895274","https://openalex.org/W1581652555","https://openalex.org/W1936333617","https://openalex.org/W1970723337","https://openalex.org/W1973171224","https://openalex.org/W1979254549","https://openalex.org/W1981135552","https://openalex.org/W1990724722","https://openalex.org/W1991689277","https://openalex.org/W2005738368","https://openalex.org/W2010115581","https://openalex.org/W2010740081","https://openalex.org/W2015642465","https://openalex.org/W2027423337","https://openalex.org/W2029439915","https://openalex.org/W2031168104","https://openalex.org/W2035436935","https://openalex.org/W2047007104","https://openalex.org/W2048158428","https://openalex.org/W2049564609","https://openalex.org/W2053551029","https://openalex.org/W2057971042","https://openalex.org/W2063494908","https://openalex.org/W2071502429","https://openalex.org/W2074631079","https://openalex.org/W2079788836","https://openalex.org/W2082201094","https://openalex.org/W2090406558","https://openalex.org/W2104961861","https://openalex.org/W2124394725","https://openalex.org/W2131313775","https://openalex.org/W2163312887","https://openalex.org/W2174198570","https://openalex.org/W2178366283","https://openalex.org/W2223822401","https://openalex.org/W2258115004","https://openalex.org/W2529629629","https://openalex.org/W2617061729"],"related_works":["https://openalex.org/W1981135552","https://openalex.org/W2174198570","https://openalex.org/W7033841024","https://openalex.org/W6999504293","https://openalex.org/W2049564609","https://openalex.org/W2047007104","https://openalex.org/W2029439915","https://openalex.org/W2061423032","https://openalex.org/W1984149204","https://openalex.org/W1480646162"],"abstract_inverted_index":null,"counts_by_year":[{"year":2024,"cited_by_count":1},{"year":2023,"cited_by_count":1},{"year":2020,"cited_by_count":1},{"year":2019,"cited_by_count":2}],"updated_date":"2026-10-31T12:09:11.096373","created_date":"2018-06-01T00:00:00"}
