{"id":"https://openalex.org/W2569801166","doi":"https://doi.org/10.3390/ijms18010116","title":"Hydroxypyridinone Chelators: From Iron Scavenging to Radiopharmaceuticals for PET Imaging with Gallium-68","display_name":"Hydroxypyridinone Chelators: From Iron Scavenging to Radiopharmaceuticals for PET Imaging with Gallium-68","publication_year":2017,"publication_date":"2017-01-08","ids":{"openalex":"https://openalex.org/W2569801166","doi":"https://doi.org/10.3390/ijms18010116","mag":"2569801166","pmid":"https://pubmed.ncbi.nlm.nih.gov/28075350","pmcid":"https://www.ncbi.nlm.nih.gov/pmc/articles/5297750"},"language":"en","primary_location":{"id":"doi:10.3390/ijms18010116","doi":"https://doi.org/10.3390/ijms18010116","is_oa":true,"landing_page_url":"https://doi.org/10.3390/ijms18010116","pdf_url":"https://www.mdpi.com/1422-0067/18/1/116/pdf?version=1484131116","source":{"id":"https://openalex.org/S10623703","display_name":"International Journal of Molecular Sciences","issn_l":"1422-0067","issn":["1422-0067","1661-6596"],"is_oa":true,"is_in_doaj":false,"is_core":true,"listed_in":["anvur-scientific","cwts-core","medline","poland-140","russia-white-list-1","vabb-shw"],"host_organization":"https://openalex.org/P4310310987","host_organization_name":"Multidisciplinary Digital Publishing Institute","host_organization_lineage":["https://openalex.org/P4310310987"],"host_organization_lineage_names":["Multidisciplinary Digital Publishing Institute"],"type":"journal"},"license":"cc-by","license_id":"https://openalex.org/licenses/cc-by","version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"International Journal of Molecular Sciences","raw_type":"journal-article"},"volume":null,"type":"review","indexed_in":["crossref","doaj","pubmed"],"open_access":{"is_oa":true,"oa_status":"gold","oa_url":"https://www.mdpi.com/1422-0067/18/1/116/pdf?version=1484131116","any_repository_has_fulltext":true},"authorships":[{"author_position":"first","author":{"id":"https://openalex.org/A5037176957","display_name":"Ruslan Cusnir","orcid":"https://orcid.org/0000-0001-7231-8278","observed_orcids":["https://orcid.org/0000-0001-7231-8278"]},"institutions":[{"id":"https://openalex.org/I1324925910","display_name":"St Thomas' Hospital","ror":"https://ror.org/054gk2851","country_code":"GB","type":"healthcare","lineage":["https://openalex.org/I1324925910","https://openalex.org/I200166805","https://openalex.org/I4210111135"]},{"id":"https://openalex.org/I183935753","display_name":"King's College London","ror":"https://ror.org/0220mzb33","country_code":"GB","type":"education","lineage":["https://openalex.org/I124357947","https://openalex.org/I183935753"]}],"countries":["GB"],"is_corresponding":false,"raw_author_name":"Ruslan Cusnir","raw_affiliation_strings":["Division of Imaging Sciences and Biomedical Engineering, King\u2019s College London, Fourth Floor Lambeth Wing, St. Thomas\u2019 Hospital, London SE1 7EH, UK"],"raw_orcid":"https://orcid.org/0000-0001-7231-8278","affiliations":[{"raw_affiliation_string":"Division of Imaging Sciences and Biomedical Engineering, King\u2019s College London, Fourth Floor Lambeth Wing, St. Thomas\u2019 Hospital, London SE1 7EH, UK","institution_ids":["https://openalex.org/I1324925910","https://openalex.org/I183935753"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5045714214","display_name":"Cinzia Imberti","orcid":"https://orcid.org/0000-0003-1187-7951","observed_orcids":["https://orcid.org/0000-0003-1187-7951"]},"institutions":[{"id":"https://openalex.org/I1324925910","display_name":"St Thomas' Hospital","ror":"https://ror.org/054gk2851","country_code":"GB","type":"healthcare","lineage":["https://openalex.org/I1324925910","https://openalex.org/I200166805","https://openalex.org/I4210111135"]},{"id":"https://openalex.org/I183935753","display_name":"King's College London","ror":"https://ror.org/0220mzb33","country_code":"GB","type":"education","lineage":["https://openalex.org/I124357947","https://openalex.org/I183935753"]}],"countries":["GB"],"is_corresponding":false,"raw_author_name":"Cinzia Imberti","raw_affiliation_strings":["Division of Imaging Sciences and Biomedical Engineering, King\u2019s College London, Fourth Floor Lambeth Wing, St. Thomas\u2019 Hospital, London SE1 7EH, UK"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Division of Imaging Sciences and Biomedical Engineering, King\u2019s College London, Fourth Floor Lambeth Wing, St. Thomas\u2019 Hospital, London SE1 7EH, UK","institution_ids":["https://openalex.org/I1324925910","https://openalex.org/I183935753"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5020843793","display_name":"Robert C. Hider","orcid":"https://orcid.org/0000-0003-1330-5797","observed_orcids":["https://orcid.org/0000-0003-1330-5797"]},"institutions":[{"id":"https://openalex.org/I183935753","display_name":"King's College London","ror":"https://ror.org/0220mzb33","country_code":"GB","type":"education","lineage":["https://openalex.org/I124357947","https://openalex.org/I183935753"]}],"countries":["GB"],"is_corresponding":false,"raw_author_name":"Robert Hider","raw_affiliation_strings":["Institute of Pharmaceutical Science, King\u2019s College London, Franklin-Wilkins Building, 150 Stamford Street, London SE1 9NH, UK"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Institute of Pharmaceutical Science, King\u2019s College London, Franklin-Wilkins Building, 150 Stamford Street, London SE1 9NH, UK","institution_ids":["https://openalex.org/I183935753"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5049873829","display_name":"Philip J. Blower","orcid":"https://orcid.org/0000-0001-6290-1590","observed_orcids":["https://orcid.org/0000-0001-6290-1590"]},"institutions":[{"id":"https://openalex.org/I1324925910","display_name":"St Thomas' Hospital","ror":"https://ror.org/054gk2851","country_code":"GB","type":"healthcare","lineage":["https://openalex.org/I1324925910","https://openalex.org/I200166805","https://openalex.org/I4210111135"]},{"id":"https://openalex.org/I183935753","display_name":"King's College London","ror":"https://ror.org/0220mzb33","country_code":"GB","type":"education","lineage":["https://openalex.org/I124357947","https://openalex.org/I183935753"]}],"countries":["GB"],"is_corresponding":false,"raw_author_name":"Philip Blower","raw_affiliation_strings":["Division of Imaging Sciences and Biomedical Engineering, King\u2019s College London, Fourth Floor Lambeth Wing, St. Thomas\u2019 Hospital, London SE1 7EH, UK"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Division of Imaging Sciences and Biomedical Engineering, King\u2019s College London, Fourth Floor Lambeth Wing, St. Thomas\u2019 Hospital, London SE1 7EH, UK","institution_ids":["https://openalex.org/I1324925910","https://openalex.org/I183935753"]}]},{"author_position":"last","author":{"id":"https://openalex.org/A5023837325","display_name":"Michelle Ma","orcid":"https://orcid.org/0000-0002-3349-7346","observed_orcids":["https://orcid.org/0000-0002-3349-7346"]},"institutions":[{"id":"https://openalex.org/I1324925910","display_name":"St Thomas' Hospital","ror":"https://ror.org/054gk2851","country_code":"GB","type":"healthcare","lineage":["https://openalex.org/I1324925910","https://openalex.org/I200166805","https://openalex.org/I4210111135"]},{"id":"https://openalex.org/I183935753","display_name":"King's College London","ror":"https://ror.org/0220mzb33","country_code":"GB","type":"education","lineage":["https://openalex.org/I124357947","https://openalex.org/I183935753"]}],"countries":["GB"],"is_corresponding":true,"raw_author_name":"Michelle Ma","raw_affiliation_strings":["Division of Imaging Sciences and Biomedical Engineering, King\u2019s College London, Fourth Floor Lambeth Wing, St. Thomas\u2019 Hospital, London SE1 7EH, UK"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Division of Imaging Sciences and Biomedical Engineering, King\u2019s College London, Fourth Floor Lambeth Wing, St. Thomas\u2019 Hospital, London SE1 7EH, UK","institution_ids":["https://openalex.org/I1324925910","https://openalex.org/I183935753"]}]}],"institutions":[],"countries_distinct_count":1,"institutions_distinct_count":2,"corresponding_author_ids":["https://openalex.org/A5023837325"],"corresponding_institution_ids":["https://openalex.org/I1324925910","https://openalex.org/I183935753"],"apc_list":{"value":2900,"currency":"CHF","value_usd":3499},"apc_paid":{"value":2900,"currency":"CHF","value_usd":3499},"fwci":1.4543,"has_fulltext":true,"cited_by_count":67,"citation_normalized_percentile":{"value":0.81272727,"is_in_top_1_percent":false,"is_in_top_10_percent":false},"cited_by_percentile_year":{"min":88,"max":99},"biblio":{"volume":"18","issue":"1","first_page":"116","last_page":"116"},"is_retracted":false,"is_paratext":false,"is_xpac":false,"primary_topic":{"id":"https://openalex.org/T11395","display_name":"Radiopharmaceutical Chemistry and Applications","score":0.9994999766349792,"subfield":{"id":"https://openalex.org/subfields/2741","display_name":"Radiology, Nuclear Medicine and Imaging"},"field":{"id":"https://openalex.org/fields/27","display_name":"Medicine"},"domain":{"id":"https://openalex.org/domains/4","display_name":"Health Sciences"}},"topics":[{"id":"https://openalex.org/T11395","display_name":"Radiopharmaceutical Chemistry and Applications","score":0.9994999766349792,"subfield":{"id":"https://openalex.org/subfields/2741","display_name":"Radiology, Nuclear Medicine and Imaging"},"field":{"id":"https://openalex.org/fields/27","display_name":"Medicine"},"domain":{"id":"https://openalex.org/domains/4","display_name":"Health Sciences"}},{"id":"https://openalex.org/T10522","display_name":"Medical Imaging Techniques and Applications","score":9.999999747378752e-05,"subfield":{"id":"https://openalex.org/subfields/2741","display_name":"Radiology, Nuclear Medicine and Imaging"},"field":{"id":"https://openalex.org/fields/27","display_name":"Medicine"},"domain":{"id":"https://openalex.org/domains/4","display_name":"Health Sciences"}},{"id":"https://openalex.org/T13561","display_name":"Chemical Reactions and Isotopes","score":9.999999747378752e-05,"subfield":{"id":"https://openalex.org/subfields/3003","display_name":"Pharmaceutical Science"},"field":{"id":"https://openalex.org/fields/30","display_name":"Pharmacology, Toxicology and Pharmaceutics"},"domain":{"id":"https://openalex.org/domains/1","display_name":"Life Sciences"}}],"keywords":[{"id":"https://openalex.org/keywords/iron-chelation","display_name":"iron chelation","score":0.7549999952316284},{"id":"https://openalex.org/keywords/deferoxamine","display_name":"deferoxamine","score":0.734000027179718},{"id":"https://openalex.org/keywords/iron-overload","display_name":"iron overload","score":0.828000009059906},{"id":"https://openalex.org/keywords/gallium-68","display_name":"gallium-68","score":0.9179999828338623},{"id":"https://openalex.org/keywords/radiopharmaceuticals","display_name":"radiopharmaceuticals","score":0.7940000295639038},{"id":"https://openalex.org/keywords/positron-emission-tomography","display_name":"positron emission tomography","score":0.7990000247955322},{"id":"https://openalex.org/keywords/radiosynthesis","display_name":"radiotracer synthesis","score":0.8820000290870667},{"id":"https://openalex.org/keywords/renal-excretion","display_name":"renal excretion","score":0.718999981880188},{"id":"https://openalex.org/keywords/bifunctional-chelators","display_name":"bifunctional chelators","score":0.9150000214576721}],"concepts":[{"id":"https://openalex.org/C550372918","wikidata":"https://www.wikidata.org/wiki/Q861","display_name":"Gallium","level":2,"score":0.6408959627151489},{"id":"https://openalex.org/C2777807096","wikidata":"https://www.wikidata.org/wiki/Q1285257","display_name":"Scavenging","level":3,"score":0.6337057948112488},{"id":"https://openalex.org/C185592680","wikidata":"https://www.wikidata.org/wiki/Q2329","display_name":"Chemistry","level":0,"score":0.5904496908187866},{"id":"https://openalex.org/C207001950","wikidata":"https://www.wikidata.org/wiki/Q141124","display_name":"In vivo","level":2,"score":0.5507305264472961},{"id":"https://openalex.org/C197404232","wikidata":"https://www.wikidata.org/wiki/Q319827","display_name":"Chelation","level":2,"score":0.4144715666770935},{"id":"https://openalex.org/C177322064","wikidata":"https://www.wikidata.org/wiki/Q750955","display_name":"Radiochemistry","level":1,"score":0.3551770746707916},{"id":"https://openalex.org/C55493867","wikidata":"https://www.wikidata.org/wiki/Q7094","display_name":"Biochemistry","level":1,"score":0.2870215177536011},{"id":"https://openalex.org/C179104552","wikidata":"https://www.wikidata.org/wiki/Q11165","display_name":"Inorganic chemistry","level":1,"score":0.23504650592803955},{"id":"https://openalex.org/C178790620","wikidata":"https://www.wikidata.org/wiki/Q11351","display_name":"Organic chemistry","level":1,"score":0.1944175660610199},{"id":"https://openalex.org/C86803240","wikidata":"https://www.wikidata.org/wiki/Q420","display_name":"Biology","level":0,"score":0.12691879272460938},{"id":"https://openalex.org/C2778004101","wikidata":"https://www.wikidata.org/wiki/Q133948","display_name":"Antioxidant","level":2,"score":0.10988166928291321},{"id":"https://openalex.org/C150903083","wikidata":"https://www.wikidata.org/wiki/Q7108","display_name":"Biotechnology","level":1,"score":0.056070804595947266}],"mesh":[{"descriptor_ui":"D000818","descriptor_name":"Animals","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D002614","descriptor_name":"Chelating Agents","qualifier_ui":"Q000494","qualifier_name":"pharmacology","is_major_topic":true},{"descriptor_ui":"D005710","descriptor_name":"Gallium Radioisotopes","qualifier_ui":"Q000737","qualifier_name":"chemistry","is_major_topic":true},{"descriptor_ui":"D006801","descriptor_name":"Humans","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D007501","descriptor_name":"Iron","qualifier_ui":"Q000378","qualifier_name":"metabolism","is_major_topic":true},{"descriptor_ui":"D011728","descriptor_name":"Pyridones","qualifier_ui":"Q000494","qualifier_name":"pharmacology","is_major_topic":true},{"descriptor_ui":"D011728","descriptor_name":"Pyridones","qualifier_ui":"Q000737","qualifier_name":"chemistry","is_major_topic":false},{"descriptor_ui":"D019275","descriptor_name":"Radiopharmaceuticals","qualifier_ui":"Q000494","qualifier_name":"pharmacology","is_major_topic":true},{"descriptor_ui":"D049268","descriptor_name":"Positron-Emission Tomography","qualifier_ui":null,"qualifier_name":null,"is_major_topic":true}],"locations_count":5,"locations":[{"id":"doi:10.3390/ijms18010116","doi":"https://doi.org/10.3390/ijms18010116","is_oa":true,"landing_page_url":"https://doi.org/10.3390/ijms18010116","pdf_url":"https://www.mdpi.com/1422-0067/18/1/116/pdf?version=1484131116","source":{"id":"https://openalex.org/S10623703","display_name":"International Journal of Molecular Sciences","issn_l":"1422-0067","issn":["1422-0067","1661-6596"],"is_oa":true,"is_in_doaj":false,"is_core":true,"listed_in":["anvur-scientific","cwts-core","medline","poland-140","russia-white-list-1","vabb-shw"],"host_organization":"https://openalex.org/P4310310987","host_organization_name":"Multidisciplinary Digital Publishing Institute","host_organization_lineage":["https://openalex.org/P4310310987"],"host_organization_lineage_names":["Multidisciplinary Digital Publishing Institute"],"type":"journal"},"license":"cc-by","license_id":"https://openalex.org/licenses/cc-by","version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"International Journal of Molecular Sciences","raw_type":"journal-article"},{"id":"pmh:oai:pubmedcentral.nih.gov:5297750","doi":null,"is_oa":true,"landing_page_url":"https://www.ncbi.nlm.nih.gov/pmc/articles/5297750","pdf_url":null,"source":{"id":"https://openalex.org/S2764455111","display_name":"PubMed Central","issn_l":null,"issn":null,"is_oa":true,"is_in_doaj":false,"is_core":false,"listed_in":[],"host_organization":"https://openalex.org/I1299303238","host_organization_name":"National Institutes of Health","host_organization_lineage":["https://openalex.org/I1299303238"],"host_organization_lineage_names":[],"type":"repository"},"license":"cc-by","license_id":"https://openalex.org/licenses/cc-by","version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"Int J Mol Sci","raw_type":"Text"},{"id":"pmid:28075350","doi":null,"is_oa":false,"landing_page_url":"https://pubmed.ncbi.nlm.nih.gov/28075350","pdf_url":null,"source":{"id":"https://openalex.org/S4306525036","display_name":"PubMed","issn_l":null,"issn":null,"is_oa":false,"is_in_doaj":false,"is_core":false,"listed_in":[],"host_organization":"https://openalex.org/I1299303238","host_organization_name":"National Institutes of Health","host_organization_lineage":["https://openalex.org/I1299303238"],"host_organization_lineage_names":[],"type":"repository"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"International journal of molecular sciences","raw_type":"Journal Article"},{"id":"pmh:oai:kclpure.kcl.ac.uk:openaire/6324e9e5-69bf-4f6b-9d89-7796bd38d4e0","doi":null,"is_oa":true,"landing_page_url":"https://kclpure.kcl.ac.uk/portal/files/63174527/ijms_18_00116_v3_1_.pdf","pdf_url":"https://kclpure.kcl.ac.uk/ws/files/63174527/ijms_18_00116_v3_1_.pdf","source":{"id":"https://openalex.org/S4306400216","display_name":"Research Portal (King's College London)","issn_l":null,"issn":null,"is_oa":false,"is_in_doaj":false,"is_core":false,"listed_in":[],"host_organization":"https://openalex.org/I183935753","host_organization_name":"King's College London","host_organization_lineage":["https://openalex.org/I183935753"],"host_organization_lineage_names":[],"type":"repository"},"license":"cc-by","license_id":"https://openalex.org/licenses/cc-by","version":"submittedVersion","is_accepted":false,"is_published":false,"raw_source_name":"Cusnir, R, Imberti, C, Hider, R C, Blower, P J & Ma, M T 2017, 'Hydroxypyridinone Chelators: From Iron Scavenging to Radiopharmaceuticals for PET Imaging with Gallium-68', International Journal of Molecular Sciences, vol. 18, no. 1, 116. https://doi.org/10.3390/ijms18010116","raw_type":"info:eu-repo/semantics/article"},{"id":"pmh:oai:doaj.org/article:b100490767f74989876b6c8a9dab46d7","doi":null,"is_oa":true,"landing_page_url":"https://doaj.org/article/b100490767f74989876b6c8a9dab46d7","pdf_url":null,"source":{"id":"https://openalex.org/S4306401280","display_name":"DOAJ (DOAJ: Directory of Open Access Journals)","issn_l":null,"issn":null,"is_oa":false,"is_in_doaj":false,"is_core":false,"listed_in":[],"host_organization":null,"host_organization_name":null,"host_organization_lineage":[],"host_organization_lineage_names":[],"type":"repository"},"license":"cc-by-sa","license_id":"https://openalex.org/licenses/cc-by-sa","version":"submittedVersion","is_accepted":false,"is_published":false,"raw_source_name":"International Journal of Molecular Sciences, Vol 18, Iss 1, p 116 (2017)","raw_type":"article"}],"best_oa_location":{"id":"doi:10.3390/ijms18010116","doi":"https://doi.org/10.3390/ijms18010116","is_oa":true,"landing_page_url":"https://doi.org/10.3390/ijms18010116","pdf_url":"https://www.mdpi.com/1422-0067/18/1/116/pdf?version=1484131116","source":{"id":"https://openalex.org/S10623703","display_name":"International Journal of Molecular Sciences","issn_l":"1422-0067","issn":["1422-0067","1661-6596"],"is_oa":true,"is_in_doaj":false,"is_core":true,"listed_in":["anvur-scientific","cwts-core","medline","poland-140","russia-white-list-1","vabb-shw"],"host_organization":"https://openalex.org/P4310310987","host_organization_name":"Multidisciplinary Digital Publishing Institute","host_organization_lineage":["https://openalex.org/P4310310987"],"host_organization_lineage_names":["Multidisciplinary Digital Publishing Institute"],"type":"journal"},"license":"cc-by","license_id":"https://openalex.org/licenses/cc-by","version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"International Journal of Molecular Sciences","raw_type":"journal-article"},"sustainable_development_goals":[{"display_name":"Good health and well-being","score":0.5683000087738037,"id":"https://metadata.un.org/sdg/3"}],"study_designs":[],"awards":[{"id":"https://openalex.org/G1565451380","display_name":"Development and preclinical testing of a bifunctional chelator for 89Zr binding and a novel 89Zr radiotracer for ImmunoPET imaging of PD-1 checkpoint expression","funder_award_id":"168441","funder_id":"https://openalex.org/F4320320924","funder_display_name":"Schweizerischer Nationalfonds zur F\u00f6rderung der Wissenschaftlichen Forschung"},{"id":"https://openalex.org/G1721109152","display_name":null,"funder_award_id":"WT088641","funder_id":"https://openalex.org/F4320311904","funder_display_name":"Wellcome Trust"},{"id":"https://openalex.org/G2073892509","display_name":null,"funder_award_id":"WT 088641/Z/09/Z","funder_id":"https://openalex.org/F4320334627","funder_display_name":"Engineering and Physical Sciences Research Council"},{"id":"https://openalex.org/G3337424878","display_name":null,"funder_award_id":"WT088641 \u2044Z \u2044 09 \u2044 Z","funder_id":"https://openalex.org/F4320311904","funder_display_name":"Wellcome Trust"},{"id":"https://openalex.org/G5161675118","display_name":null,"funder_award_id":"16463","funder_id":"https://openalex.org/F4320319985","funder_display_name":"Cancer Research UK"},{"id":"https://openalex.org/G8526282538","display_name":null,"funder_award_id":"P2LAP3","funder_id":"https://openalex.org/F4320320924","funder_display_name":"Schweizerischer Nationalfonds zur F\u00f6rderung der Wissenschaftlichen Forschung"}],"funders":[{"id":"https://openalex.org/F4320306076","display_name":"National Science Foundation","ror":"https://ror.org/021nxhr62"},{"id":"https://openalex.org/F4320311904","display_name":"Wellcome Trust","ror":"https://ror.org/029chgv08"},{"id":"https://openalex.org/F4320315071","display_name":"NIHR Biomedical Research Centre, Royal Marsden NHS Foundation Trust/Institute of Cancer Research","ror":"https://ror.org/0187kwz08"},{"id":"https://openalex.org/F4320319985","display_name":"Cancer Research UK","ror":"https://ror.org/054225q67"},{"id":"https://openalex.org/F4320319990","display_name":"National Institute for Health and Care Research","ror":"https://ror.org/0187kwz08"},{"id":"https://openalex.org/F4320320285","display_name":"King's College London","ror":"https://ror.org/0220mzb33"},{"id":"https://openalex.org/F4320320286","display_name":"University College London","ror":"https://ror.org/02jx3x895"},{"id":"https://openalex.org/F4320320924","display_name":"Schweizerischer Nationalfonds zur F\u00f6rderung der Wissenschaftlichen Forschung","ror":"https://ror.org/00yjd3n13"},{"id":"https://openalex.org/F4320334626","display_name":"Medical Research Council","ror":"https://ror.org/03x94j517"},{"id":"https://openalex.org/F4320334627","display_name":"Engineering and Physical Sciences Research Council","ror":"https://ror.org/0439y7842"}],"has_content":{"grobid_xml":true,"pdf":true},"content_urls":{"pdf":"https://content.openalex.org/works/W2569801166.pdf","grobid_xml":"https://content.openalex.org/works/W2569801166.grobid-xml"},"referenced_works_count":70,"referenced_works":["https://openalex.org/W1423295325","https://openalex.org/W1520088546","https://openalex.org/W1565486843","https://openalex.org/W1862590115","https://openalex.org/W1920139082","https://openalex.org/W1966335626","https://openalex.org/W1971403832","https://openalex.org/W1973773380","https://openalex.org/W1974592901","https://openalex.org/W1974603642","https://openalex.org/W1974868569","https://openalex.org/W1976103847","https://openalex.org/W1979986689","https://openalex.org/W1984552257","https://openalex.org/W1988872182","https://openalex.org/W1990645562","https://openalex.org/W2004283265","https://openalex.org/W2006250045","https://openalex.org/W2008386216","https://openalex.org/W2012655209","https://openalex.org/W2013363580","https://openalex.org/W2018768546","https://openalex.org/W2019760194","https://openalex.org/W2020296930","https://openalex.org/W2020893960","https://openalex.org/W2021147596","https://openalex.org/W2022194542","https://openalex.org/W2023098302","https://openalex.org/W2023833723","https://openalex.org/W2028066320","https://openalex.org/W2031572086","https://openalex.org/W2033066083","https://openalex.org/W2034260204","https://openalex.org/W2036519391","https://openalex.org/W2046429311","https://openalex.org/W2046771337","https://openalex.org/W2049294159","https://openalex.org/W2054308752","https://openalex.org/W2056537429","https://openalex.org/W2056570094","https://openalex.org/W2057426811","https://openalex.org/W2059715782","https://openalex.org/W2061352340","https://openalex.org/W2068566410","https://openalex.org/W2074712830","https://openalex.org/W2078920454","https://openalex.org/W2080006760","https://openalex.org/W2083125064","https://openalex.org/W2092446767","https://openalex.org/W2095260497","https://openalex.org/W2102971043","https://openalex.org/W2104324067","https://openalex.org/W2107301029","https://openalex.org/W2149259388","https://openalex.org/W2151127435","https://openalex.org/W2157187629","https://openalex.org/W2163393284","https://openalex.org/W2167590372","https://openalex.org/W2172796913","https://openalex.org/W2192838961","https://openalex.org/W2209913242","https://openalex.org/W2261107289","https://openalex.org/W2263922604","https://openalex.org/W2290990628","https://openalex.org/W2406418570","https://openalex.org/W2418918484","https://openalex.org/W2501073592","https://openalex.org/W2516044053","https://openalex.org/W2536268804","https://openalex.org/W6675465224"],"related_works":["https://openalex.org/W2023098302","https://openalex.org/W2922285995","https://openalex.org/W3148582570","https://openalex.org/W2263922604","https://openalex.org/W2062987476","https://openalex.org/W2916904628","https://openalex.org/W1974868569","https://openalex.org/W4390102572","https://openalex.org/W2100762530","https://openalex.org/W7046933865"],"abstract_inverted_index":{"Derivatives":[0],"of":[1,22,90,98],"3,4-hydroxypyridinones":[2],"have":[3,46],"been":[4],"extensively":[5],"studied":[6],"for":[7,19,41,51,57,67],"in":[8,70,108],"vivo":[9],"Fe3+":[10,31],"sequestration.":[11],"Deferiprone,":[12],"a":[13,115],"1,2-dimethyl-3,4-hydroxypyridinone,":[14],"is":[15,64],"now":[16],"routinely":[17],"used":[18,66],"clinical":[20],"treatment":[21],"iron":[23,35],"overload":[24],"disease.":[25],"Hexadentate":[26],"tris(3,4-hydroxypyridinone)":[27],"ligands":[28],"(THP)":[29],"complex":[30,80],"at":[32,82,105],"very":[33],"low":[34],"concentrations,":[36],"and":[37,78,87,110],"their":[38,49],"high":[39,119],"affinities":[40],"oxophilic":[42],"trivalent":[43],"metal":[44],"ions":[45],"led":[47],"to":[48,95],"development":[50],"new":[52],"applications":[53],"as":[54],"bifunctional":[55],"chelators":[56],"the":[58],"positron":[59,71],"emitting":[60],"radiometal,":[61],"68Ga3+,":[62],"which":[63],"clinically":[65],"molecular":[68],"imaging":[69],"emission":[72],"tomography":[73],"(PET).":[74],"THP-peptide":[75],"bioconjugates":[76],"rapidly":[77],"quantitatively":[79],"68Ga3+":[81],"ambient":[83],"temperature,":[84],"neutral":[85],"pH":[86],"micromolar":[88],"concentrations":[89],"ligand,":[91],"making":[92],"them":[93],"amenable":[94],"kit-based":[96],"radiosynthesis":[97],"68Ga":[99],"PET":[100,121],"radiopharmaceuticals.":[101],"68Ga-labelled":[102],"THP-peptides":[103],"accumulate":[104],"target":[106],"tissue":[107],"vivo,":[109],"are":[111],"excreted":[112],"largely":[113],"via":[114],"renal":[116],"pathway,":[117],"providing":[118],"quality":[120],"images.":[122]},"counts_by_year":[{"year":2026,"cited_by_count":4},{"year":2025,"cited_by_count":6},{"year":2024,"cited_by_count":8},{"year":2023,"cited_by_count":1},{"year":2022,"cited_by_count":6},{"year":2021,"cited_by_count":6},{"year":2020,"cited_by_count":9},{"year":2019,"cited_by_count":12},{"year":2018,"cited_by_count":6},{"year":2017,"cited_by_count":8},{"year":2015,"cited_by_count":1}],"updated_date":"2026-11-04T10:54:05.112534","created_date":"2017-01-13T00:00:00"}
