{"id":"https://openalex.org/W2182393979","doi":null,"title":"INSILICO DOCKING ANALYSIS OF KAEMPHEROL AND LUTEOLIN AGAINST DIABETIC DRUG TARGET PEPCK1","display_name":"INSILICO DOCKING ANALYSIS OF KAEMPHEROL AND LUTEOLIN AGAINST DIABETIC DRUG TARGET PEPCK1","publication_year":2014,"publication_date":"2014-01-01","ids":{"openalex":"https://openalex.org/W2182393979","mag":"2182393979"},"language":"en","primary_location":{"id":"mag:2182393979","doi":null,"is_oa":false,"landing_page_url":"http://www.ijpbs.net/cms/php/upload/3801_pdf.pdf","pdf_url":null,"source":{"id":"https://openalex.org/S2764788474","display_name":"International Journal of Pharma and Bio Sciences","issn_l":"0975-6299","issn":["0975-6299"],"is_oa":false,"is_in_doaj":false,"is_core":false,"listed_in":[],"host_organization":"https://openalex.org/P4322697007","host_organization_name":"Ubitech Solutions","host_organization_lineage":["https://openalex.org/P4322697007"],"host_organization_lineage_names":["Ubitech Solutions"],"type":"journal"},"license":null,"license_id":null,"version":null,"is_accepted":false,"is_published":false,"raw_source_name":"International Journal of Pharma and Bio Sciences","raw_type":null},"volume":null,"type":"article","is_traditional":true,"indexed_in":[],"open_access":{"is_oa":false,"oa_status":"closed","oa_url":null,"any_repository_has_fulltext":false},"authorships":[{"author_position":"first","author":{"id":"https://openalex.org/A5026532960","display_name":"Amalorpavam J and Dr. G. A. I. Ebenezer","orcid":null,"observed_orcids":[]},"institutions":[],"countries":[],"is_corresponding":true,"raw_author_name":"Amalorpavam J and Dr. G. A. I. Ebenezer","raw_affiliation_strings":[],"raw_orcid":null,"affiliations":[]}],"institutions":[],"countries_distinct_count":0,"institutions_distinct_count":0,"corresponding_author_ids":["https://openalex.org/A5026532960"],"corresponding_institution_ids":[],"apc_list":null,"apc_paid":null,"fwci":0.0,"has_fulltext":false,"cited_by_count":0,"citation_normalized_percentile":{"value":0.0,"is_in_top_1_percent":false,"is_in_top_10_percent":false},"cited_by_percentile_year":null,"biblio":{"volume":null,"issue":null,"first_page":null,"last_page":null},"is_retracted":false,"is_paratext":false,"is_xpac":false,"primary_topic":{"id":"https://openalex.org/T10211","display_name":"Computational Drug Discovery Methods","score":0.8804000020027161,"subfield":{"id":"https://openalex.org/subfields/3002","display_name":"Drug Discovery"},"field":{"id":"https://openalex.org/fields/30","display_name":"Pharmacology, Toxicology and Pharmaceutics"},"domain":{"id":"https://openalex.org/domains/1","display_name":"Life Sciences"}},"topics":[{"id":"https://openalex.org/T10211","display_name":"Computational Drug Discovery Methods","score":0.8804000020027161,"subfield":{"id":"https://openalex.org/subfields/3002","display_name":"Drug Discovery"},"field":{"id":"https://openalex.org/fields/30","display_name":"Pharmacology, Toxicology and Pharmaceutics"},"domain":{"id":"https://openalex.org/domains/1","display_name":"Life Sciences"}},{"id":"https://openalex.org/T11140","display_name":"Natural Antidiabetic Agents Studies","score":0.09740000218153,"subfield":{"id":"https://openalex.org/subfields/2712","display_name":"Endocrinology, Diabetes and Metabolism"},"field":{"id":"https://openalex.org/fields/27","display_name":"Medicine"},"domain":{"id":"https://openalex.org/domains/4","display_name":"Health Sciences"}},{"id":"https://openalex.org/T12257","display_name":"Bioactive natural compounds","score":0.003800000064074993,"subfield":{"id":"https://openalex.org/subfields/3002","display_name":"Drug Discovery"},"field":{"id":"https://openalex.org/fields/30","display_name":"Pharmacology, Toxicology and Pharmaceutics"},"domain":{"id":"https://openalex.org/domains/1","display_name":"Life Sciences"}}],"keywords":[{"id":"https://openalex.org/keywords/kaempferol","display_name":"kaempferol","score":0.9940000176429749},{"id":"https://openalex.org/keywords/luteolin","display_name":"luteolin","score":1.0},{"id":"https://openalex.org/keywords/pck1","display_name":"PCK1","score":0.9330000281333923},{"id":"https://openalex.org/keywords/flavonoids","display_name":"flavonoids","score":0.9890000224113464},{"id":"https://openalex.org/keywords/antidiabetic-activity","display_name":"antidiabetic activity","score":0.9259999990463257},{"id":"https://openalex.org/keywords/diabetes-mellitus","display_name":"diabetes mellitus","score":0.6359999775886536},{"id":"https://openalex.org/keywords/molecular-docking","display_name":"molecular docking","score":0.7129999995231628},{"id":"https://openalex.org/keywords/phytochemical-screening","display_name":"phytochemical screening","score":0.703000009059906},{"id":"https://openalex.org/keywords/methanol-extract","display_name":"methanol extract","score":0.7860000133514404}],"concepts":[{"id":"https://openalex.org/C195475562","wikidata":"https://www.wikidata.org/wiki/Q1639139","display_name":"Phytochemical","level":2,"score":0.7418064475059509},{"id":"https://openalex.org/C41685203","wikidata":"https://www.wikidata.org/wiki/Q1974042","display_name":"Docking (animal)","level":2,"score":0.7410209774971008},{"id":"https://openalex.org/C2776080593","wikidata":"https://www.wikidata.org/wiki/Q415011","display_name":"Luteolin","level":4,"score":0.6025232672691345},{"id":"https://openalex.org/C2779450374","wikidata":"https://www.wikidata.org/wiki/Q27724763","display_name":"International Journal of Pharma and Bio Sciences","level":2,"score":0.5739363431930542},{"id":"https://openalex.org/C2779134260","wikidata":"https://www.wikidata.org/wiki/Q12136","display_name":"Disease","level":2,"score":0.46264350414276123},{"id":"https://openalex.org/C2780035454","wikidata":"https://www.wikidata.org/wiki/Q8386","display_name":"Drug","level":2,"score":0.45787426829338074},{"id":"https://openalex.org/C556039675","wikidata":"https://www.wikidata.org/wiki/Q771035","display_name":"Traditional medicine","level":1,"score":0.4214743971824646},{"id":"https://openalex.org/C71924100","wikidata":"https://www.wikidata.org/wiki/Q11190","display_name":"Medicine","level":0,"score":0.3706657886505127},{"id":"https://openalex.org/C98274493","wikidata":"https://www.wikidata.org/wiki/Q128406","display_name":"Pharmacology","level":1,"score":0.3602815270423889},{"id":"https://openalex.org/C185592680","wikidata":"https://www.wikidata.org/wiki/Q2329","display_name":"Chemistry","level":0,"score":0.2605566382408142},{"id":"https://openalex.org/C55493867","wikidata":"https://www.wikidata.org/wiki/Q7094","display_name":"Biochemistry","level":1,"score":0.15520811080932617},{"id":"https://openalex.org/C17744445","wikidata":"https://www.wikidata.org/wiki/Q36442","display_name":"Political science","level":0,"score":0.1419701874256134},{"id":"https://openalex.org/C199539241","wikidata":"https://www.wikidata.org/wiki/Q7748","display_name":"Law","level":1,"score":0.10742247104644775},{"id":"https://openalex.org/C42972112","wikidata":"https://www.wikidata.org/wiki/Q170201","display_name":"Veterinary medicine","level":1,"score":0.10528188943862915},{"id":"https://openalex.org/C2779054382","wikidata":"https://www.wikidata.org/wiki/Q72185287","display_name":"Flavonoid","level":3,"score":0.07132148742675781},{"id":"https://openalex.org/C126322002","wikidata":"https://www.wikidata.org/wiki/Q11180","display_name":"Internal medicine","level":1,"score":0.07028853893280029},{"id":"https://openalex.org/C2778004101","wikidata":"https://www.wikidata.org/wiki/Q133948","display_name":"Antioxidant","level":2,"score":0.0}],"mesh":[],"locations_count":1,"locations":[{"id":"mag:2182393979","doi":null,"is_oa":false,"landing_page_url":"http://www.ijpbs.net/cms/php/upload/3801_pdf.pdf","pdf_url":null,"source":{"id":"https://openalex.org/S2764788474","display_name":"International Journal of Pharma and Bio Sciences","issn_l":"0975-6299","issn":["0975-6299"],"is_oa":false,"is_in_doaj":false,"is_core":false,"listed_in":[],"host_organization":"https://openalex.org/P4322697007","host_organization_name":"Ubitech Solutions","host_organization_lineage":["https://openalex.org/P4322697007"],"host_organization_lineage_names":["Ubitech Solutions"],"type":"journal"},"license":null,"license_id":null,"version":null,"is_accepted":false,"is_published":false,"raw_source_name":"International Journal of Pharma and Bio Sciences","raw_type":null}],"best_oa_location":null,"sustainable_development_goals":[{"score":0.8048999905586243,"display_name":"Good health and well-being","id":"https://metadata.un.org/sdg/3"}],"study_designs":[],"awards":[],"funders":[],"has_content":{"grobid_xml":false,"pdf":false},"content_urls":null,"referenced_works_count":44,"referenced_works":["https://openalex.org/W206274772","https://openalex.org/W1523821527","https://openalex.org/W1582510238","https://openalex.org/W1964750028","https://openalex.org/W1964911695","https://openalex.org/W1964958542","https://openalex.org/W1965260442","https://openalex.org/W1968697272","https://openalex.org/W1981071038","https://openalex.org/W1982315657","https://openalex.org/W1983304433","https://openalex.org/W1985570405","https://openalex.org/W1985588649","https://openalex.org/W1986240377","https://openalex.org/W2001003469","https://openalex.org/W2018214249","https://openalex.org/W2021791229","https://openalex.org/W2024105693","https://openalex.org/W2038053883","https://openalex.org/W2043919345","https://openalex.org/W2050159278","https://openalex.org/W2050456292","https://openalex.org/W2053987900","https://openalex.org/W2056620406","https://openalex.org/W2064318120","https://openalex.org/W2069506489","https://openalex.org/W2073598814","https://openalex.org/W2074854450","https://openalex.org/W2097744068","https://openalex.org/W2099434989","https://openalex.org/W2100349340","https://openalex.org/W2114025369","https://openalex.org/W2114779636","https://openalex.org/W2120487488","https://openalex.org/W2124241917","https://openalex.org/W2135732933","https://openalex.org/W2147818946","https://openalex.org/W2158534713","https://openalex.org/W2161849974","https://openalex.org/W2163187611","https://openalex.org/W2233170308","https://openalex.org/W2330273698","https://openalex.org/W2411681898","https://openalex.org/W4211208250"],"related_works":["https://openalex.org/W7211943941","https://openalex.org/W4323786619","https://openalex.org/W4379196647","https://openalex.org/W6941604522","https://openalex.org/W4390515799","https://openalex.org/W2187001552","https://openalex.org/W7218810819","https://openalex.org/W7196951154","https://openalex.org/W4386751751","https://openalex.org/W4404966408"],"abstract_inverted_index":{"The":[0,96,136,169],"fast":[1],"and":[2,40,93,152,182],"electronic":[3],"gadgetic,":[4],"lifestyle":[5],"have":[6,75],"led":[7],"mankind":[8],"to":[9,14,37,54,57,83,91,102,176],"a":[10],"complicated":[11],"mesh":[12],"leading":[13],"many":[15,47,51],"diseases":[16,104],"that":[17,32,87],"passively":[18],"spreads":[19],"into":[20],"the":[21,58,69,81,106,117,121,128,140,144,160,165,172],"population":[22],"producing":[23],"an":[24],"unhealthy":[25],"society.":[26],"Diabetes":[27],"is":[28,33,125,175],"one":[29],"such":[30],"disease":[31,92],"gaining":[34],"ground":[35],"due":[36],"eating":[38],"habits":[39],"sedentary":[41],"lifesyte.":[42],"Even":[43],"though":[44],"there":[45],"are":[46,88],"pharmaceutical":[48],"products":[49],"available":[50],"patients":[52],"prefer":[53],"revert":[55],"back":[56],"slow":[59],"healthy":[60],"approach":[61],"integrated":[62],"with":[63],"natural":[64],"therapeutics.":[65],"In":[66,112],"recent":[67],"years,":[68],"demands":[70],"on":[71],"drug":[72],"discovery":[73],"process":[74],"increased":[76],"dramatically,":[77],"partly":[78],"because":[79],"of":[80,98,116,139,143,171,180],"necessity":[82],"recognize":[84],"novel":[85],"target":[86,166],"both":[89],"pertinent":[90],"chemically":[94],"tractable.":[95],"emergence":[97],"bioinformatics":[99],"gives":[100],"room":[101],"investigate":[103],"at":[105],"molecular":[107],"level":[108],"using":[109],"computational":[110],"techniques.":[111],"this":[113],"study,":[114],"some":[115],"flavonoids":[118,156],"present":[119,173],"in":[120,127],"tamarind":[122,145],"seed":[123,146],"coat":[124,147],"used":[126],"insilico":[129,161],"docking":[130,162],"analysis":[131,163],"against":[132,164,184],"phosphoenolpyruvate":[133],"carboxykinase":[134],"(PEPCK1).":[135],"phytochemical":[137],"investigation":[138],"methanolic":[141],"extract":[142],"was":[148],"positive":[149],"for":[150,159],"Kaempherol":[151],"luteolin.":[153],"These":[154],"two":[155],"were":[157],"selected":[158],"protein":[167],"PEPCK1.":[168,185],"aim":[170],"study":[174],"describe":[177],"antidiabetic":[178],"role":[179],"kaempherol":[181],"lately":[183]},"counts_by_year":[],"updated_date":"2026-11-04T10:54:05.112534","created_date":"2016-06-24T00:00:00"}
