{"id":"https://openalex.org/W2171990235","doi":"https://doi.org/10.1002/cmdc.201000191","title":"Synthesis and Evaluation of Bombesin Analogues Conjugated to Two Different Triazolyl\u2010Derived Chelators for 99mTc Labeling","display_name":"Synthesis and Evaluation of Bombesin Analogues Conjugated to Two Different Triazolyl\u2010Derived Chelators for 99mTc Labeling","publication_year":2010,"publication_date":"2010-08-30","ids":{"openalex":"https://openalex.org/W2171990235","doi":"https://doi.org/10.1002/cmdc.201000191","mag":"2171990235","pmid":"https://pubmed.ncbi.nlm.nih.gov/20806312"},"language":"en","primary_location":{"id":"doi:10.1002/cmdc.201000191","doi":"https://doi.org/10.1002/cmdc.201000191","is_oa":false,"landing_page_url":"https://doi.org/10.1002/cmdc.201000191","pdf_url":null,"source":{"id":"https://openalex.org/S136164820","display_name":"ChemMedChem","issn_l":"1860-7179","issn":["1860-7179","1860-7187"],"is_oa":false,"is_in_doaj":false,"is_core":true,"listed_in":["cwts-core","dongbi-c","jufo-1","ki-jl-1","medline","norway-1","poland-100","russia-white-list-2","vabb-shw"],"host_organization":"https://openalex.org/P4310320595","host_organization_name":"Wiley","host_organization_lineage":["https://openalex.org/P4310320595"],"host_organization_lineage_names":["Wiley"],"type":"journal"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"ChemMedChem","raw_type":"journal-article"},"volume":null,"type":"article","is_traditional":true,"indexed_in":["crossref","pubmed"],"open_access":{"is_oa":false,"oa_status":"closed","oa_url":null,"any_repository_has_fulltext":false},"authorships":[{"author_position":"first","author":{"id":"https://openalex.org/A5000510379","display_name":"Luc Brans","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I13469542","display_name":"Vrije Universiteit Brussel","ror":"https://ror.org/006e5kg04","country_code":"BE","type":"education","lineage":["https://openalex.org/I13469542"]}],"countries":["BE"],"is_corresponding":false,"raw_author_name":"Luc Brans","raw_affiliation_strings":["Department of Organic Chemistry, Vrije Universiteit Brussel, 1050 Brussels, Belgium"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Department of Organic Chemistry, Vrije Universiteit Brussel, 1050 Brussels, Belgium","institution_ids":["https://openalex.org/I13469542"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5035100973","display_name":"Elisa Garc\u00eda\u2010Garayoa","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I2802229908","display_name":"Paul Scherrer Institute","ror":"https://ror.org/03eh3y714","country_code":"CH","type":"facility","lineage":["https://openalex.org/I2799323385","https://openalex.org/I2802229908"]}],"countries":["CH"],"is_corresponding":false,"raw_author_name":"Elisa Garc\u00eda\u2010Garayoa","raw_affiliation_strings":["Center for Radiopharmaceutical Science, Paul Scherrer Institute, 5232 Villigen-PSI (Switzerland)"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Center for Radiopharmaceutical Science, Paul Scherrer Institute, 5232 Villigen-PSI (Switzerland)","institution_ids":["https://openalex.org/I2802229908"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5089139708","display_name":"Christian Schweinsberg","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I2802229908","display_name":"Paul Scherrer Institute","ror":"https://ror.org/03eh3y714","country_code":"CH","type":"facility","lineage":["https://openalex.org/I2799323385","https://openalex.org/I2802229908"]}],"countries":["CH"],"is_corresponding":false,"raw_author_name":"Christian Schweinsberg","raw_affiliation_strings":["Center for Radiopharmaceutical Science, Paul Scherrer Institute, 5232 Villigen-PSI (Switzerland)"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Center for Radiopharmaceutical Science, Paul Scherrer Institute, 5232 Villigen-PSI (Switzerland)","institution_ids":["https://openalex.org/I2802229908"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5111368110","display_name":"V\u00e9ronique Maes","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I13469542","display_name":"Vrije Universiteit Brussel","ror":"https://ror.org/006e5kg04","country_code":"BE","type":"education","lineage":["https://openalex.org/I13469542"]}],"countries":["BE"],"is_corresponding":false,"raw_author_name":"Veronique Maes","raw_affiliation_strings":["Department of Organic Chemistry, Vrije Universiteit Brussel, 1050 Brussels (Belgium),"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Department of Organic Chemistry, Vrije Universiteit Brussel, 1050 Brussels (Belgium),","institution_ids":["https://openalex.org/I13469542"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5067357097","display_name":"Harriet Struthers","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I35440088","display_name":"ETH Zurich","ror":"https://ror.org/05a28rw58","country_code":"CH","type":"education","lineage":["https://openalex.org/I2799323385","https://openalex.org/I35440088"]}],"countries":["CH"],"is_corresponding":false,"raw_author_name":"Harriet Struthers","raw_affiliation_strings":["Department of Chemistry and Applied Biosciences, ETH Zurich, 8093 Zurich (Switzerland)"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Department of Chemistry and Applied Biosciences, ETH Zurich, 8093 Zurich (Switzerland)","institution_ids":["https://openalex.org/I35440088"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5041743198","display_name":"Roger Schibli","orcid":"https://orcid.org/0000-0002-1537-3833","observed_orcids":["https://orcid.org/0000-0002-1537-3833"]},"institutions":[{"id":"https://openalex.org/I2802229908","display_name":"Paul Scherrer Institute","ror":"https://ror.org/03eh3y714","country_code":"CH","type":"facility","lineage":["https://openalex.org/I2799323385","https://openalex.org/I2802229908"]},{"id":"https://openalex.org/I35440088","display_name":"ETH Zurich","ror":"https://ror.org/05a28rw58","country_code":"CH","type":"education","lineage":["https://openalex.org/I2799323385","https://openalex.org/I35440088"]}],"countries":["CH"],"is_corresponding":false,"raw_author_name":"Roger Schibli","raw_affiliation_strings":["Center for Radiopharmaceutical Science, Paul Scherrer Institute, 5232 Villigen-PSI (Switzerland)","Department of Chemistry and Applied Biosciences, ETH Zurich, 8093 Zurich (Switzerland)"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Center for Radiopharmaceutical Science, Paul Scherrer Institute, 5232 Villigen-PSI (Switzerland)","institution_ids":["https://openalex.org/I2802229908"]},{"raw_affiliation_string":"Department of Chemistry and Applied Biosciences, ETH Zurich, 8093 Zurich (Switzerland)","institution_ids":["https://openalex.org/I35440088"]}]},{"author_position":"last","author":{"id":"https://openalex.org/A5064093167","display_name":"Dirk Tourw\u00e9","orcid":"https://orcid.org/0000-0002-2329-0798","observed_orcids":["https://orcid.org/0000-0002-2329-0798"]},"institutions":[{"id":"https://openalex.org/I13469542","display_name":"Vrije Universiteit Brussel","ror":"https://ror.org/006e5kg04","country_code":"BE","type":"education","lineage":["https://openalex.org/I13469542"]}],"countries":["BE"],"is_corresponding":true,"raw_author_name":"Dirk Tourw\u00e9","raw_affiliation_strings":["Department of Organic Chemistry, Vrije Universiteit Brussel, 1050 Brussels (Belgium),"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Department of Organic Chemistry, Vrije Universiteit Brussel, 1050 Brussels (Belgium),","institution_ids":["https://openalex.org/I13469542"]}]}],"institutions":[],"countries_distinct_count":2,"institutions_distinct_count":3,"corresponding_author_ids":["https://openalex.org/A5064093167"],"corresponding_institution_ids":["https://openalex.org/I13469542"],"apc_list":{"value":4150,"currency":"USD","value_usd":4150},"apc_paid":null,"fwci":1.4989,"has_fulltext":false,"cited_by_count":22,"citation_normalized_percentile":{"value":0.79556437,"is_in_top_1_percent":false,"is_in_top_10_percent":false},"cited_by_percentile_year":{"min":88,"max":97},"biblio":{"volume":"5","issue":"10","first_page":"1717","last_page":"1725"},"is_retracted":false,"is_paratext":false,"is_xpac":false,"primary_topic":{"id":"https://openalex.org/T11395","display_name":"Radiopharmaceutical Chemistry and Applications","score":0.9945999979972839,"subfield":{"id":"https://openalex.org/subfields/2741","display_name":"Radiology, Nuclear Medicine and Imaging"},"field":{"id":"https://openalex.org/fields/27","display_name":"Medicine"},"domain":{"id":"https://openalex.org/domains/4","display_name":"Health Sciences"}},"topics":[{"id":"https://openalex.org/T11395","display_name":"Radiopharmaceutical Chemistry and Applications","score":0.9945999979972839,"subfield":{"id":"https://openalex.org/subfields/2741","display_name":"Radiology, Nuclear Medicine and Imaging"},"field":{"id":"https://openalex.org/fields/27","display_name":"Medicine"},"domain":{"id":"https://openalex.org/domains/4","display_name":"Health Sciences"}},{"id":"https://openalex.org/T10911","display_name":"Chemical Synthesis and Analysis","score":0.0019000000320374966,"subfield":{"id":"https://openalex.org/subfields/1605","display_name":"Organic Chemistry"},"field":{"id":"https://openalex.org/fields/16","display_name":"Chemistry"},"domain":{"id":"https://openalex.org/domains/3","display_name":"Physical Sciences"}},{"id":"https://openalex.org/T10754","display_name":"Neuroendocrine Tumor Research Advances","score":0.001500000013038516,"subfield":{"id":"https://openalex.org/subfields/2730","display_name":"Oncology"},"field":{"id":"https://openalex.org/fields/27","display_name":"Medicine"},"domain":{"id":"https://openalex.org/domains/4","display_name":"Health Sciences"}}],"keywords":[{"id":"https://openalex.org/keywords/bombesin-analogues","display_name":"bombesin analogues","score":0.996999979019165},{"id":"https://openalex.org/keywords/gastrin-releasing-peptide-receptor","display_name":"gastrin-releasing peptide receptor","score":0.9789999723434448},{"id":"https://openalex.org/keywords/99mtc-radiolabeling","display_name":"99mTc radiolabeling","score":0.8740000128746033},{"id":"https://openalex.org/keywords/click-chemistry","display_name":"click chemistry","score":0.675000011920929},{"id":"https://openalex.org/keywords/glycation","display_name":"glycation","score":0.7900000214576721},{"id":"https://openalex.org/keywords/copper-catalyzed-azide-alkyne-cycloaddition","display_name":"copper-catalyzed azide-alkyne cycloaddition","score":0.8960000276565552},{"id":"https://openalex.org/keywords/tissue-distribution","display_name":"tissue distribution","score":0.8090000152587891},{"id":"https://openalex.org/keywords/tumor-to-background-ratio","display_name":"tumor-to-background ratio","score":0.9779999852180481},{"id":"https://openalex.org/keywords/peptide-radiotracers","display_name":"peptide radiotracers","score":0.5640000104904175},{"id":"https://openalex.org/keywords/tumor-imaging","display_name":"tumor imaging","score":0.33500000834465027}],"concepts":[{"id":"https://openalex.org/C112613896","wikidata":"https://www.wikidata.org/wiki/Q898370","display_name":"Conjugated system","level":3,"score":0.7348236441612244},{"id":"https://openalex.org/C2778448772","wikidata":"https://www.wikidata.org/wiki/Q349427","display_name":"Bombesin","level":4,"score":0.6557953357696533},{"id":"https://openalex.org/C185592680","wikidata":"https://www.wikidata.org/wiki/Q2329","display_name":"Chemistry","level":0,"score":0.6489913463592529},{"id":"https://openalex.org/C21951064","wikidata":"https://www.wikidata.org/wiki/Q899212","display_name":"Combinatorial chemistry","level":1,"score":0.4500274956226349},{"id":"https://openalex.org/C197404232","wikidata":"https://www.wikidata.org/wiki/Q319827","display_name":"Chelation","level":2,"score":0.44519880414009094},{"id":"https://openalex.org/C71240020","wikidata":"https://www.wikidata.org/wiki/Q186011","display_name":"Stereochemistry","level":1,"score":0.3996889889240265},{"id":"https://openalex.org/C177322064","wikidata":"https://www.wikidata.org/wiki/Q750955","display_name":"Radiochemistry","level":1,"score":0.3937881588935852},{"id":"https://openalex.org/C55493867","wikidata":"https://www.wikidata.org/wiki/Q7094","display_name":"Biochemistry","level":1,"score":0.22509941458702087},{"id":"https://openalex.org/C178790620","wikidata":"https://www.wikidata.org/wiki/Q11351","display_name":"Organic chemistry","level":1,"score":0.16148492693901062},{"id":"https://openalex.org/C170493617","wikidata":"https://www.wikidata.org/wiki/Q208467","display_name":"Receptor","level":2,"score":0.12133759260177612},{"id":"https://openalex.org/C521977710","wikidata":"https://www.wikidata.org/wiki/Q81163","display_name":"Polymer","level":2,"score":0.0},{"id":"https://openalex.org/C118303440","wikidata":"https://www.wikidata.org/wiki/Q419968","display_name":"Neuropeptide","level":3,"score":0.0}],"mesh":[{"descriptor_ui":"D000818","descriptor_name":"Animals","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D001839","descriptor_name":"Bombesin","qualifier_ui":"Q000031","qualifier_name":"analogs & derivatives","is_major_topic":true},{"descriptor_ui":"D001839","descriptor_name":"Bombesin","qualifier_ui":"Q000138","qualifier_name":"chemical synthesis","is_major_topic":false},{"descriptor_ui":"D001839","descriptor_name":"Bombesin","qualifier_ui":"Q000493","qualifier_name":"pharmacokinetics","is_major_topic":false},{"descriptor_ui":"D002384","descriptor_name":"Catalysis","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D002614","descriptor_name":"Chelating Agents","qualifier_ui":"Q000138","qualifier_name":"chemical synthesis","is_major_topic":false},{"descriptor_ui":"D002614","descriptor_name":"Chelating Agents","qualifier_ui":"Q000493","qualifier_name":"pharmacokinetics","is_major_topic":false},{"descriptor_ui":"D002614","descriptor_name":"Chelating Agents","qualifier_ui":"Q000737","qualifier_name":"chemistry","is_major_topic":true},{"descriptor_ui":"D003300","descriptor_name":"Copper","qualifier_ui":"Q000737","qualifier_name":"chemistry","is_major_topic":false},{"descriptor_ui":"D006801","descriptor_name":"Humans","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D007553","descriptor_name":"Isotope Labeling","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D008819","descriptor_name":"Mice, Nude","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D013667","descriptor_name":"Technetium","qualifier_ui":"Q000737","qualifier_name":"chemistry","is_major_topic":false},{"descriptor_ui":"D014230","descriptor_name":"Triazoles","qualifier_ui":"Q000737","qualifier_name":"chemistry","is_major_topic":true},{"descriptor_ui":"D015899","descriptor_name":"Tomography, Emission-Computed, Single-Photon","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D018004","descriptor_name":"Receptors, Bombesin","qualifier_ui":"Q000037","qualifier_name":"antagonists & inhibitors","is_major_topic":false},{"descriptor_ui":"D018004","descriptor_name":"Receptors, Bombesin","qualifier_ui":"Q000378","qualifier_name":"metabolism","is_major_topic":false},{"descriptor_ui":"D023041","descriptor_name":"Xenograft Model Antitumor Assays","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D045744","descriptor_name":"Cell Line, Tumor","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D051379","descriptor_name":"Mice","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false}],"locations_count":4,"locations":[{"id":"doi:10.1002/cmdc.201000191","doi":"https://doi.org/10.1002/cmdc.201000191","is_oa":false,"landing_page_url":"https://doi.org/10.1002/cmdc.201000191","pdf_url":null,"source":{"id":"https://openalex.org/S136164820","display_name":"ChemMedChem","issn_l":"1860-7179","issn":["1860-7179","1860-7187"],"is_oa":false,"is_in_doaj":false,"is_core":true,"listed_in":["cwts-core","dongbi-c","jufo-1","ki-jl-1","medline","norway-1","poland-100","russia-white-list-2","vabb-shw"],"host_organization":"https://openalex.org/P4310320595","host_organization_name":"Wiley","host_organization_lineage":["https://openalex.org/P4310320595"],"host_organization_lineage_names":["Wiley"],"type":"journal"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"ChemMedChem","raw_type":"journal-article"},{"id":"pmid:20806312","doi":null,"is_oa":false,"landing_page_url":"https://pubmed.ncbi.nlm.nih.gov/20806312","pdf_url":null,"source":{"id":"https://openalex.org/S4306525036","display_name":"PubMed","issn_l":null,"issn":null,"is_oa":false,"is_in_doaj":false,"is_core":false,"listed_in":[],"host_organization":"https://openalex.org/I1299303238","host_organization_name":"National Institutes of Health","host_organization_lineage":["https://openalex.org/I1299303238"],"host_organization_lineage_names":[],"type":"repository"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"ChemMedChem","raw_type":"Journal Article"},{"id":"pmh:oai:dora:psi_50401","doi":null,"is_oa":false,"landing_page_url":"https://www.dora.lib4ri.ch/psi/item/psi:50401","pdf_url":null,"source":{"id":"https://openalex.org/S4306402574","display_name":"DORA PSI (Paul Scherrer Institute)","issn_l":null,"issn":null,"is_oa":false,"is_in_doaj":false,"is_core":false,"listed_in":[],"host_organization":"https://openalex.org/I2802229908","host_organization_name":"Paul Scherrer Institute","host_organization_lineage":["https://openalex.org/I2802229908"],"host_organization_lineage_names":[],"type":"repository"},"license":null,"license_id":null,"version":"submittedVersion","is_accepted":false,"is_published":false,"raw_source_name":"ChemMedChem","raw_type":"info:eu-repo/semantics/article"},{"id":"pmh:oai:vubissmart:VUBISSMART:2000:68793","doi":null,"is_oa":false,"landing_page_url":"https://biblio.vub.ac.be/vubir/synthesis-and-evaluation-of-bombesin-analogues-conjugated-to-two-different-triazolylderived-chelators-for-tc99m-labeling(896e4ebf-c183-4528-a430-989f3f7c36bd).html","pdf_url":null,"source":{"id":"https://openalex.org/S4306402573","display_name":"VUBIR (Vrije Universiteit Brussel)","issn_l":null,"issn":null,"is_oa":false,"is_in_doaj":false,"is_core":false,"listed_in":[],"host_organization":"https://openalex.org/I13469542","host_organization_name":"Vrije Universiteit Brussel","host_organization_lineage":["https://openalex.org/I13469542"],"host_organization_lineage_names":[],"type":"repository"},"license":null,"license_id":null,"version":"submittedVersion","is_accepted":false,"is_published":false,"raw_source_name":null,"raw_type":"article"}],"best_oa_location":null,"sustainable_development_goals":[{"score":0.6240000128746033,"id":"https://metadata.un.org/sdg/3","display_name":"Good health and well-being"}],"study_designs":[],"awards":[],"funders":[],"has_content":{"pdf":false,"grobid_xml":false},"content_urls":null,"referenced_works_count":47,"referenced_works":["https://openalex.org/W1173924217","https://openalex.org/W1500549738","https://openalex.org/W1848804918","https://openalex.org/W1861064994","https://openalex.org/W1933901479","https://openalex.org/W1964916916","https://openalex.org/W1965895443","https://openalex.org/W1967250787","https://openalex.org/W1968652549","https://openalex.org/W1969531388","https://openalex.org/W1975737622","https://openalex.org/W1977066986","https://openalex.org/W1989505230","https://openalex.org/W1990332976","https://openalex.org/W1991297789","https://openalex.org/W2003515334","https://openalex.org/W2013794755","https://openalex.org/W2029389567","https://openalex.org/W2031956553","https://openalex.org/W2044059225","https://openalex.org/W2045681528","https://openalex.org/W2045687112","https://openalex.org/W2056584927","https://openalex.org/W2062098928","https://openalex.org/W2062301515","https://openalex.org/W2064888038","https://openalex.org/W2065571239","https://openalex.org/W2077108003","https://openalex.org/W2100676734","https://openalex.org/W2105248439","https://openalex.org/W2105255209","https://openalex.org/W2117243098","https://openalex.org/W2122452293","https://openalex.org/W2131897082","https://openalex.org/W2136155687","https://openalex.org/W2145661651","https://openalex.org/W2146122430","https://openalex.org/W2146183051","https://openalex.org/W2162586071","https://openalex.org/W2273366209","https://openalex.org/W2282139172","https://openalex.org/W2330091639","https://openalex.org/W2355013303","https://openalex.org/W2413660070","https://openalex.org/W2798513649","https://openalex.org/W2949921135","https://openalex.org/W4256503849"],"related_works":["https://openalex.org/W2003515334","https://openalex.org/W2131897082","https://openalex.org/W2026213405","https://openalex.org/W2026272847","https://openalex.org/W2044434912","https://openalex.org/W1980603852","https://openalex.org/W2085354753","https://openalex.org/W2413660070","https://openalex.org/W1933901479","https://openalex.org/W2294498814"],"abstract_inverted_index":{"Overexpression":[0],"of":[1,10,17,43,72,76,123,133],"the":[2,33,40,70,83,89,124,138],"gastrin-releasing":[3],"peptide":[4,48],"receptor":[5],"(GRPR)":[6],"in":[7,69,108,111],"a":[8,15,24,73],"variety":[9],"human":[11],"carcinomas":[12],"has":[13],"provided":[14],"means":[16],"diagnosis":[18],"and":[19,107,110,114],"treatment.":[20],"Previously":[21],"we":[22,63],"reported":[23],"metabolically":[25],"stable":[26],"(N(\u03b1)His)Ac-\u03b2Ala-\u03b2Ala-[Cha(13),Nle(14)]BBS(7-14)":[27],"analogue":[28],"with":[29,88,102,117],"high":[30],"affinity":[31],"for":[32,86],"GRPR.":[34],"We":[35],"have":[36],"also":[37],"shown":[38],"that":[39,132],"biodistribution":[41,127],"pattern":[42],"this":[44,66],"fairly":[45],"lipophilic,":[46],"radiolabeled":[47],"can":[49],"be":[50],"enhanced":[51],"by":[52,59],"glycation,":[53,134],"which":[54,135],"is":[55],"easily":[56],"carried":[57],"out":[58],"Cu(I)-catalyzed":[60],"cycloaddition.":[61],"Herein,":[62],"further":[64],"elaborate":[65],"\"click":[67],"approach\"":[68],"synthesis":[71,106],"new":[74,97],"series":[75],"triazole-based":[77],"chelating":[78,98],"systems":[79],"as":[80],"alternatives":[81],"to":[82,104],"(N(\u03b1)His)Ac":[84,119],"chelator":[85,125],"labeling":[87],"(99m)Tc(CO)(3)":[90],"core.":[91],"The":[92,121],"bombesin":[93],"analogues,":[94],"containing":[95],"these":[96],"systems,":[99],"were":[100,115],"evaluated":[101],"regard":[103],"their":[105,118],"vitro":[109],"vivo":[112],"properties,":[113],"compared":[116],"counterparts.":[120],"influence":[122],"on":[126],"properties":[128],"was":[129],"less":[130],"than":[131],"clearly":[136],"improved":[137],"tumor-to-background":[139],"ratios.":[140]},"counts_by_year":[{"year":2026,"cited_by_count":1},{"year":2025,"cited_by_count":1},{"year":2022,"cited_by_count":1},{"year":2020,"cited_by_count":3},{"year":2019,"cited_by_count":1},{"year":2017,"cited_by_count":3},{"year":2016,"cited_by_count":1},{"year":2014,"cited_by_count":4},{"year":2013,"cited_by_count":3},{"year":2012,"cited_by_count":2}],"updated_date":"2026-11-06T12:05:46.655746","created_date":"2016-06-24T00:00:00"}
