{"id":"https://openalex.org/W2158299122","doi":"https://doi.org/10.1124/mol.114.097485","title":"Antiobesity Effect of a Small Molecule Repressor of ROR\u03b3","display_name":"Antiobesity Effect of a Small Molecule Repressor of ROR\u03b3","publication_year":2015,"publication_date":"2015-04-23","ids":{"openalex":"https://openalex.org/W2158299122","doi":"https://doi.org/10.1124/mol.114.097485","mag":"2158299122","pmid":"https://pubmed.ncbi.nlm.nih.gov/25904554","pmcid":"https://www.ncbi.nlm.nih.gov/pmc/articles/4468634"},"language":"en","primary_location":{"id":"doi:10.1124/mol.114.097485","doi":"https://doi.org/10.1124/mol.114.097485","is_oa":false,"landing_page_url":"https://doi.org/10.1124/mol.114.097485","pdf_url":null,"source":{"id":"https://openalex.org/S62949411","display_name":"Molecular Pharmacology","issn_l":"0026-895X","issn":["0026-895X","1521-0111"],"is_oa":false,"is_in_doaj":false,"is_core":true,"listed_in":["cwts-core","dongbi-c","doyens","jufo-2","ki-jl-2","medline","norway-2","poland-140","russia-white-list-1"],"host_organization":"https://openalex.org/P4310316283","host_organization_name":"American Society for Pharmacology and Experimental Therapeutics","host_organization_lineage":["https://openalex.org/P4310316283"],"host_organization_lineage_names":["American Society for Pharmacology and Experimental Therapeutics"],"type":"journal"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"Molecular Pharmacology","raw_type":"journal-article"},"volume":null,"type":"article","indexed_in":["crossref","pubmed"],"open_access":{"is_oa":true,"oa_status":"green","oa_url":"https://www.ncbi.nlm.nih.gov/pmc/articles/4468634","any_repository_has_fulltext":true},"authorships":[{"author_position":"first","author":{"id":"https://openalex.org/A5063830814","display_name":"Mi Ra Chang","orcid":"https://orcid.org/0000-0002-8594-825X","observed_orcids":["https://orcid.org/0000-0002-8594-825X"]},"institutions":[{"id":"https://openalex.org/I123431417","display_name":"Scripps Research Institute","ror":"https://ror.org/02dxx6824","country_code":"US","type":"nonprofit","lineage":["https://openalex.org/I123431417"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"Mi Ra Chang","raw_affiliation_strings":["Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.); and Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)","Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.)","Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.); and Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)","institution_ids":["https://openalex.org/I123431417"]},{"raw_affiliation_string":"Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.)","institution_ids":["https://openalex.org/I123431417"]},{"raw_affiliation_string":"Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)","institution_ids":[]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5038470522","display_name":"Yuanjun He","orcid":"https://orcid.org/0000-0002-3983-5529","observed_orcids":["https://orcid.org/0000-0002-3983-5529"]},"institutions":[{"id":"https://openalex.org/I123431417","display_name":"Scripps Research Institute","ror":"https://ror.org/02dxx6824","country_code":"US","type":"nonprofit","lineage":["https://openalex.org/I123431417"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"Yuanjun He","raw_affiliation_strings":["Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.); and Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)","Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.)","Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.); and Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)","institution_ids":["https://openalex.org/I123431417"]},{"raw_affiliation_string":"Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.)","institution_ids":["https://openalex.org/I123431417"]},{"raw_affiliation_string":"Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)","institution_ids":[]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5047202823","display_name":"Tanya M. Khan","orcid":"https://orcid.org/0000-0003-0323-8017","observed_orcids":["https://orcid.org/0000-0003-0323-8017"]},"institutions":[{"id":"https://openalex.org/I123431417","display_name":"Scripps Research Institute","ror":"https://ror.org/02dxx6824","country_code":"US","type":"nonprofit","lineage":["https://openalex.org/I123431417"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"Tanya M. Khan","raw_affiliation_strings":["Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.); and Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)","Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.)","Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.); and Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)","institution_ids":["https://openalex.org/I123431417"]},{"raw_affiliation_string":"Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.)","institution_ids":["https://openalex.org/I123431417"]},{"raw_affiliation_string":"Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)","institution_ids":[]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5062971256","display_name":"Dana S. Kuruvilla","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I123431417","display_name":"Scripps Research Institute","ror":"https://ror.org/02dxx6824","country_code":"US","type":"nonprofit","lineage":["https://openalex.org/I123431417"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"Dana S. Kuruvilla","raw_affiliation_strings":["Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.); and Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)","Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.)","Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.); and Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)","institution_ids":["https://openalex.org/I123431417"]},{"raw_affiliation_string":"Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.)","institution_ids":["https://openalex.org/I123431417"]},{"raw_affiliation_string":"Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)","institution_ids":[]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5023186460","display_name":"Rub\u00e9n D. Garcia-Ordo\u00f1ez","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I123431417","display_name":"Scripps Research Institute","ror":"https://ror.org/02dxx6824","country_code":"US","type":"nonprofit","lineage":["https://openalex.org/I123431417"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"Ruben Garcia-Ordonez","raw_affiliation_strings":["Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.); and Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)","Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.)","Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.); and Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)","institution_ids":["https://openalex.org/I123431417"]},{"raw_affiliation_string":"Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.)","institution_ids":["https://openalex.org/I123431417"]},{"raw_affiliation_string":"Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)","institution_ids":[]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5016309219","display_name":"Cesar A. Corzo","orcid":"https://orcid.org/0000-0002-9592-450X","observed_orcids":["https://orcid.org/0000-0002-9592-450X"]},"institutions":[{"id":"https://openalex.org/I123431417","display_name":"Scripps Research Institute","ror":"https://ror.org/02dxx6824","country_code":"US","type":"nonprofit","lineage":["https://openalex.org/I123431417"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"Cesar A. Corzo","raw_affiliation_strings":["Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.); and Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)","Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.)","Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.); and Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)","institution_ids":["https://openalex.org/I123431417"]},{"raw_affiliation_string":"Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.)","institution_ids":["https://openalex.org/I123431417"]},{"raw_affiliation_string":"Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)","institution_ids":[]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5033009352","display_name":"Thaddeus J. Unger","orcid":"https://orcid.org/0000-0002-5780-4857","observed_orcids":["https://orcid.org/0000-0002-5780-4857"]},"institutions":[{"id":"https://openalex.org/I123431417","display_name":"Scripps Research Institute","ror":"https://ror.org/02dxx6824","country_code":"US","type":"nonprofit","lineage":["https://openalex.org/I123431417"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"Thaddeus J. Unger","raw_affiliation_strings":["Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.); and Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)","Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.)","Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.); and Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)","institution_ids":["https://openalex.org/I123431417"]},{"raw_affiliation_string":"Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.)","institution_ids":["https://openalex.org/I123431417"]},{"raw_affiliation_string":"Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)","institution_ids":[]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5103457199","display_name":"David W. White","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I123431417","display_name":"Scripps Research Institute","ror":"https://ror.org/02dxx6824","country_code":"US","type":"nonprofit","lineage":["https://openalex.org/I123431417"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"David W. White","raw_affiliation_strings":["Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.); and Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)","Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.)","Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.); and Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)","institution_ids":["https://openalex.org/I123431417"]},{"raw_affiliation_string":"Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.)","institution_ids":["https://openalex.org/I123431417"]},{"raw_affiliation_string":"Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)","institution_ids":[]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5100862873","display_name":"Susan Khan","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I123431417","display_name":"Scripps Research Institute","ror":"https://ror.org/02dxx6824","country_code":"US","type":"nonprofit","lineage":["https://openalex.org/I123431417"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"Susan Khan","raw_affiliation_strings":["Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.); and Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)","Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.)","Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.); and Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)","institution_ids":["https://openalex.org/I123431417"]},{"raw_affiliation_string":"Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.)","institution_ids":["https://openalex.org/I123431417"]},{"raw_affiliation_string":"Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)","institution_ids":[]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5100609560","display_name":"Li Lin","orcid":"https://orcid.org/0000-0002-3707-0745","observed_orcids":["https://orcid.org/0000-0002-3707-0745"]},"institutions":[{"id":"https://openalex.org/I123431417","display_name":"Scripps Research Institute","ror":"https://ror.org/02dxx6824","country_code":"US","type":"nonprofit","lineage":["https://openalex.org/I123431417"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"Li Lin","raw_affiliation_strings":["Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.); and Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)","Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.)","Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.); and Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)","institution_ids":["https://openalex.org/I123431417"]},{"raw_affiliation_string":"Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.)","institution_ids":["https://openalex.org/I123431417"]},{"raw_affiliation_string":"Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)","institution_ids":[]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5041449809","display_name":"Michael D. Cameron","orcid":"https://orcid.org/0000-0003-3154-4775","observed_orcids":["https://orcid.org/0000-0003-3154-4775"]},"institutions":[{"id":"https://openalex.org/I123431417","display_name":"Scripps Research Institute","ror":"https://ror.org/02dxx6824","country_code":"US","type":"nonprofit","lineage":["https://openalex.org/I123431417"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"Michael D. Cameron","raw_affiliation_strings":["Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.); and Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)","Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.)","Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.); and Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)","institution_ids":["https://openalex.org/I123431417"]},{"raw_affiliation_string":"Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.)","institution_ids":["https://openalex.org/I123431417"]},{"raw_affiliation_string":"Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)","institution_ids":[]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5066500327","display_name":"Theodore M. Kamenecka","orcid":"https://orcid.org/0000-0002-3077-0167","observed_orcids":["https://orcid.org/0000-0002-3077-0167"]},"institutions":[{"id":"https://openalex.org/I123431417","display_name":"Scripps Research Institute","ror":"https://ror.org/02dxx6824","country_code":"US","type":"nonprofit","lineage":["https://openalex.org/I123431417"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"Theodore M. Kamenecka","raw_affiliation_strings":["Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.); and Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)","Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.)","Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.); and Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)","institution_ids":["https://openalex.org/I123431417"]},{"raw_affiliation_string":"Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.)","institution_ids":["https://openalex.org/I123431417"]},{"raw_affiliation_string":"Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)","institution_ids":[]}]},{"author_position":"last","author":{"id":"https://openalex.org/A5000139914","display_name":"Patrick R. Griffin","orcid":"https://orcid.org/0000-0002-3404-690X","observed_orcids":["https://orcid.org/0000-0002-3404-690X"]},"institutions":[{"id":"https://openalex.org/I123431417","display_name":"Scripps Research Institute","ror":"https://ror.org/02dxx6824","country_code":"US","type":"nonprofit","lineage":["https://openalex.org/I123431417"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"Patrick R. Griffin","raw_affiliation_strings":["Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.); and Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.) pgriffin@scripps.edu","Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.)","Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.); and Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.) pgriffin@scripps.edu","institution_ids":["https://openalex.org/I123431417"]},{"raw_affiliation_string":"Department of Molecular Therapeutics, The Scripps Research Institute, Jupiter, Florida (M.R.C., Y.H., T.M.K., D.S.K., R.G.-O., C.A.C., S.K., L.L., M.D.C., Th.M.K., P.R.G.)","institution_ids":["https://openalex.org/I123431417"]},{"raw_affiliation_string":"Ember Therapeutics, Watertown, Massachusetts (T.J.U., D.W.W.)","institution_ids":[]}]}],"institutions":[],"countries_distinct_count":1,"institutions_distinct_count":1,"corresponding_author_ids":[],"corresponding_institution_ids":["https://openalex.org/I123431417"],"apc_list":{"value":3600,"currency":"USD","value_usd":3600},"apc_paid":null,"fwci":2.8929,"has_fulltext":false,"cited_by_count":34,"citation_normalized_percentile":{"value":0.90423063,"is_in_top_1_percent":false,"is_in_top_10_percent":true},"cited_by_percentile_year":{"min":90,"max":99},"biblio":{"volume":"88","issue":"1","first_page":"48","last_page":"56"},"is_retracted":false,"is_paratext":false,"is_xpac":false,"primary_topic":{"id":"https://openalex.org/T11457","display_name":"Adipose Tissue and Metabolism","score":0.7782999873161316,"subfield":{"id":"https://openalex.org/subfields/2737","display_name":"Physiology (medical)"},"field":{"id":"https://openalex.org/fields/27","display_name":"Medicine"},"domain":{"id":"https://openalex.org/domains/4","display_name":"Health Sciences"}},"topics":[{"id":"https://openalex.org/T11457","display_name":"Adipose Tissue and Metabolism","score":0.7782999873161316,"subfield":{"id":"https://openalex.org/subfields/2737","display_name":"Physiology (medical)"},"field":{"id":"https://openalex.org/fields/27","display_name":"Medicine"},"domain":{"id":"https://openalex.org/domains/4","display_name":"Health Sciences"}},{"id":"https://openalex.org/T10528","display_name":"Adipokines, Inflammation, and Metabolic Diseases","score":0.1289999932050705,"subfield":{"id":"https://openalex.org/subfields/2713","display_name":"Epidemiology"},"field":{"id":"https://openalex.org/fields/27","display_name":"Medicine"},"domain":{"id":"https://openalex.org/domains/4","display_name":"Health Sciences"}},{"id":"https://openalex.org/T11072","display_name":"Peroxisome Proliferator-Activated Receptors","score":0.031300000846385956,"subfield":{"id":"https://openalex.org/subfields/1312","display_name":"Molecular Biology"},"field":{"id":"https://openalex.org/fields/13","display_name":"Biochemistry, Genetics and Molecular Biology"},"domain":{"id":"https://openalex.org/domains/1","display_name":"Life Sciences"}}],"keywords":[{"id":"https://openalex.org/keywords/rorgamma","display_name":"ROR\u03b3","score":0.9879999756813049},{"id":"https://openalex.org/keywords/anti-obesity-effect","display_name":"anti-obesity","score":0.7179999947547913},{"id":"https://openalex.org/keywords/th17-differentiation","display_name":"Th17 cell differentiation","score":0.7670000195503235},{"id":"https://openalex.org/keywords/fgf21","display_name":"FGF21","score":0.8679999709129333},{"id":"https://openalex.org/keywords/adiponectin","display_name":"adiponectin","score":0.9509999752044678},{"id":"https://openalex.org/keywords/thermogenesis","display_name":"thermogenesis","score":0.847000002861023},{"id":"https://openalex.org/keywords/fatty-acid-oxidation","display_name":"fatty acid oxidation","score":0.8190000057220459},{"id":"https://openalex.org/keywords/hormone-sensitive-lipase","display_name":"hormone-sensitive lipase","score":0.9810000061988831},{"id":"https://openalex.org/keywords/insulin-sensitivity","display_name":"insulin sensitivity","score":0.9779999852180481},{"id":"https://openalex.org/keywords/obesity","display_name":"obesity","score":0.6549999713897705},{"id":"https://openalex.org/keywords/adipocytes","display_name":"adipocytes","score":0.5429999828338623},{"id":"https://openalex.org/keywords/free-fatty-acids","display_name":"free fatty acids","score":0.6790000200271606},{"id":"https://openalex.org/keywords/circadian-rhythm-genes","display_name":"circadian rhythm genes","score":0.43799999356269836}],"concepts":[{"id":"https://openalex.org/C134018914","wikidata":"https://www.wikidata.org/wiki/Q162606","display_name":"Endocrinology","level":1,"score":0.6715285778045654},{"id":"https://openalex.org/C126322002","wikidata":"https://www.wikidata.org/wiki/Q11180","display_name":"Internal medicine","level":1,"score":0.6641011238098145},{"id":"https://openalex.org/C185592680","wikidata":"https://www.wikidata.org/wiki/Q2329","display_name":"Chemistry","level":0,"score":0.5558640360832214},{"id":"https://openalex.org/C71315377","wikidata":"https://www.wikidata.org/wiki/Q11364","display_name":"Hormone","level":2,"score":0.5349563360214233},{"id":"https://openalex.org/C74737994","wikidata":"https://www.wikidata.org/wiki/Q18031207","display_name":"RAR-related orphan receptor gamma","level":4,"score":0.495508074760437},{"id":"https://openalex.org/C2778938600","wikidata":"https://www.wikidata.org/wiki/Q389934","display_name":"Agonist","level":3,"score":0.463817298412323},{"id":"https://openalex.org/C170493617","wikidata":"https://www.wikidata.org/wiki/Q208467","display_name":"Receptor","level":2,"score":0.44838595390319824},{"id":"https://openalex.org/C171089720","wikidata":"https://www.wikidata.org/wiki/Q193583","display_name":"Adipose tissue","level":2,"score":0.43168947100639343},{"id":"https://openalex.org/C151279926","wikidata":"https://www.wikidata.org/wiki/Q965695","display_name":"Thermogenesis","level":3,"score":0.4293971359729767},{"id":"https://openalex.org/C26291073","wikidata":"https://www.wikidata.org/wiki/Q310484","display_name":"Ex vivo","level":3,"score":0.42273688316345215},{"id":"https://openalex.org/C89951826","wikidata":"https://www.wikidata.org/wiki/Q1671731","display_name":"Inverse agonist","level":4,"score":0.4180854260921478},{"id":"https://openalex.org/C63932345","wikidata":"https://www.wikidata.org/wiki/Q422500","display_name":"Nuclear receptor","level":4,"score":0.41300058364868164},{"id":"https://openalex.org/C202751555","wikidata":"https://www.wikidata.org/wiki/Q221681","display_name":"In vitro","level":2,"score":0.3182666003704071},{"id":"https://openalex.org/C86803240","wikidata":"https://www.wikidata.org/wiki/Q420","display_name":"Biology","level":0,"score":0.2693115472793579},{"id":"https://openalex.org/C55493867","wikidata":"https://www.wikidata.org/wiki/Q7094","display_name":"Biochemistry","level":1,"score":0.24815696477890015},{"id":"https://openalex.org/C104317684","wikidata":"https://www.wikidata.org/wiki/Q7187","display_name":"Gene","level":2,"score":0.20201730728149414},{"id":"https://openalex.org/C71924100","wikidata":"https://www.wikidata.org/wiki/Q11190","display_name":"Medicine","level":0,"score":0.12654179334640503},{"id":"https://openalex.org/C86339819","wikidata":"https://www.wikidata.org/wiki/Q407384","display_name":"Transcription factor","level":3,"score":0.0}],"mesh":[{"descriptor_ui":"D000818","descriptor_name":"Animals","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D001713","descriptor_name":"Biphenyl Compounds","qualifier_ui":"Q000008","qualifier_name":"administration & dosage","is_major_topic":true},{"descriptor_ui":"D001713","descriptor_name":"Biphenyl Compounds","qualifier_ui":"Q000138","qualifier_name":"chemical synthesis","is_major_topic":false},{"descriptor_ui":"D001713","descriptor_name":"Biphenyl Compounds","qualifier_ui":"Q000494","qualifier_name":"pharmacology","is_major_topic":false},{"descriptor_ui":"D001835","descriptor_name":"Body Weight","qualifier_ui":"Q000187","qualifier_name":"drug effects","is_major_topic":false},{"descriptor_ui":"D002478","descriptor_name":"Cells, Cultured","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D005346","descriptor_name":"Fibroblast Growth Factors","qualifier_ui":"Q000378","qualifier_name":"metabolism","is_major_topic":false},{"descriptor_ui":"D007328","descriptor_name":"Insulin","qualifier_ui":"Q000378","qualifier_name":"metabolism","is_major_topic":true},{"descriptor_ui":"D008297","descriptor_name":"Male","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D009765","descriptor_name":"Obesity","qualifier_ui":"Q000139","qualifier_name":"chemically induced","is_major_topic":false},{"descriptor_ui":"D009765","descriptor_name":"Obesity","qualifier_ui":"Q000188","qualifier_name":"drug therapy","is_major_topic":true},{"descriptor_ui":"D009765","descriptor_name":"Obesity","qualifier_ui":"Q000235","qualifier_name":"genetics","is_major_topic":false},{"descriptor_ui":"D009765","descriptor_name":"Obesity","qualifier_ui":"Q000378","qualifier_name":"metabolism","is_major_topic":false},{"descriptor_ui":"D010879","descriptor_name":"Piperazines","qualifier_ui":"Q000008","qualifier_name":"administration & dosage","is_major_topic":true},{"descriptor_ui":"D010879","descriptor_name":"Piperazines","qualifier_ui":"Q000138","qualifier_name":"chemical synthesis","is_major_topic":false},{"descriptor_ui":"D010879","descriptor_name":"Piperazines","qualifier_ui":"Q000494","qualifier_name":"pharmacology","is_major_topic":false},{"descriptor_ui":"D019440","descriptor_name":"Anti-Obesity Agents","qualifier_ui":"Q000008","qualifier_name":"administration & dosage","is_major_topic":true},{"descriptor_ui":"D019440","descriptor_name":"Anti-Obesity Agents","qualifier_ui":"Q000138","qualifier_name":"chemical synthesis","is_major_topic":false},{"descriptor_ui":"D019440","descriptor_name":"Anti-Obesity Agents","qualifier_ui":"Q000494","qualifier_name":"pharmacology","is_major_topic":false},{"descriptor_ui":"D041721","descriptor_name":"3T3-L1 Cells","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D050156","descriptor_name":"Adipogenesis","qualifier_ui":"Q000187","qualifier_name":"drug effects","is_major_topic":false},{"descriptor_ui":"D051379","descriptor_name":"Mice","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D052242","descriptor_name":"Adiponectin","qualifier_ui":"Q000378","qualifier_name":"metabolism","is_major_topic":false},{"descriptor_ui":"D057132","descriptor_name":"Nuclear Receptor Subfamily 1, Group F, Member 3","qualifier_ui":"Q000037","qualifier_name":"antagonists & inhibitors","is_major_topic":true},{"descriptor_ui":"D057132","descriptor_name":"Nuclear Receptor Subfamily 1, Group F, Member 3","qualifier_ui":"Q000378","qualifier_name":"metabolism","is_major_topic":false},{"descriptor_ui":"D059305","descriptor_name":"Diet, High-Fat","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false}],"locations_count":3,"locations":[{"id":"doi:10.1124/mol.114.097485","doi":"https://doi.org/10.1124/mol.114.097485","is_oa":false,"landing_page_url":"https://doi.org/10.1124/mol.114.097485","pdf_url":null,"source":{"id":"https://openalex.org/S62949411","display_name":"Molecular Pharmacology","issn_l":"0026-895X","issn":["0026-895X","1521-0111"],"is_oa":false,"is_in_doaj":false,"is_core":true,"listed_in":["cwts-core","dongbi-c","doyens","jufo-2","ki-jl-2","medline","norway-2","poland-140","russia-white-list-1"],"host_organization":"https://openalex.org/P4310316283","host_organization_name":"American Society for Pharmacology and Experimental Therapeutics","host_organization_lineage":["https://openalex.org/P4310316283"],"host_organization_lineage_names":["American Society for Pharmacology and Experimental Therapeutics"],"type":"journal"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"Molecular Pharmacology","raw_type":"journal-article"},{"id":"pmh:oai:pubmedcentral.nih.gov:4468634","doi":null,"is_oa":true,"landing_page_url":"https://www.ncbi.nlm.nih.gov/pmc/articles/4468634","pdf_url":null,"source":{"id":"https://openalex.org/S2764455111","display_name":"PubMed Central","issn_l":null,"issn":null,"is_oa":true,"is_in_doaj":false,"is_core":false,"listed_in":[],"host_organization":"https://openalex.org/I1299303238","host_organization_name":"National Institutes of Health","host_organization_lineage":["https://openalex.org/I1299303238"],"host_organization_lineage_names":[],"type":"repository"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"Mol Pharmacol","raw_type":"Text"},{"id":"pmid:25904554","doi":null,"is_oa":false,"landing_page_url":"https://pubmed.ncbi.nlm.nih.gov/25904554","pdf_url":null,"source":{"id":"https://openalex.org/S4306525036","display_name":"PubMed","issn_l":null,"issn":null,"is_oa":false,"is_in_doaj":false,"is_core":false,"listed_in":[],"host_organization":"https://openalex.org/I1299303238","host_organization_name":"National Institutes of Health","host_organization_lineage":["https://openalex.org/I1299303238"],"host_organization_lineage_names":[],"type":"repository"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"Molecular pharmacology","raw_type":"Journal Article"}],"best_oa_location":{"id":"pmh:oai:pubmedcentral.nih.gov:4468634","doi":null,"is_oa":true,"landing_page_url":"https://www.ncbi.nlm.nih.gov/pmc/articles/4468634","pdf_url":null,"source":{"id":"https://openalex.org/S2764455111","display_name":"PubMed Central","issn_l":null,"issn":null,"is_oa":true,"is_in_doaj":false,"is_core":false,"listed_in":[],"host_organization":"https://openalex.org/I1299303238","host_organization_name":"National Institutes of Health","host_organization_lineage":["https://openalex.org/I1299303238"],"host_organization_lineage_names":[],"type":"repository"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"Mol Pharmacol","raw_type":"Text"},"sustainable_development_goals":[{"id":"https://metadata.un.org/sdg/3","display_name":"Good health and well-being","score":0.9537000060081482}],"study_designs":[],"awards":[{"id":"https://openalex.org/G1142036056","display_name":"Mass spectrometry for small molecule profiling in the Scripps Florida DMPK core","funder_award_id":"1s10od010603-01a1","funder_id":"https://openalex.org/F4320332161","funder_display_name":"National Institutes of Health"},{"id":"https://openalex.org/G762420777","display_name":null,"funder_award_id":"U54-MH074404","funder_id":"https://openalex.org/F4320337346","funder_display_name":"National Institute of Mental Health"},{"id":"https://openalex.org/G8146888447","display_name":"Molecular Libraries Screening Centers Network (MLSCN)(RMI)","funder_award_id":"5u54mh074404-03","funder_id":"https://openalex.org/F4320332161","funder_display_name":"National Institutes of Health"}],"funders":[{"id":"https://openalex.org/F4320332161","display_name":"National Institutes of Health","ror":"https://ror.org/01cwqze88"},{"id":"https://openalex.org/F4320337346","display_name":"National Institute of Mental Health","ror":"https://ror.org/04xeg9z08"}],"has_content":{"grobid_xml":false,"pdf":false},"content_urls":null,"referenced_works_count":38,"referenced_works":["https://openalex.org/W1972815843","https://openalex.org/W1981675213","https://openalex.org/W1984789703","https://openalex.org/W1994210536","https://openalex.org/W1996840778","https://openalex.org/W2000366854","https://openalex.org/W2006640335","https://openalex.org/W2014682602","https://openalex.org/W2019796661","https://openalex.org/W2022860174","https://openalex.org/W2027753197","https://openalex.org/W2028423973","https://openalex.org/W2028940140","https://openalex.org/W2034016494","https://openalex.org/W2037468923","https://openalex.org/W2047756822","https://openalex.org/W2054173875","https://openalex.org/W2056048638","https://openalex.org/W2076452736","https://openalex.org/W2079071895","https://openalex.org/W2085933778","https://openalex.org/W2103714496","https://openalex.org/W2107572610","https://openalex.org/W2109041281","https://openalex.org/W2114496646","https://openalex.org/W2115908495","https://openalex.org/W2116623091","https://openalex.org/W2118055379","https://openalex.org/W2123289485","https://openalex.org/W2131517624","https://openalex.org/W2137323830","https://openalex.org/W2144821774","https://openalex.org/W2148017428","https://openalex.org/W2157305411","https://openalex.org/W2157739158","https://openalex.org/W2167370342","https://openalex.org/W2170874580","https://openalex.org/W2469307620"],"related_works":["https://openalex.org/W2148017428","https://openalex.org/W2171888909","https://openalex.org/W2355855388","https://openalex.org/W2169041076","https://openalex.org/W3109132879","https://openalex.org/W2094566719","https://openalex.org/W3156524618","https://openalex.org/W2802856290","https://openalex.org/W2059742529","https://openalex.org/W2079464913"],"abstract_inverted_index":null,"counts_by_year":[{"year":2025,"cited_by_count":1},{"year":2023,"cited_by_count":2},{"year":2022,"cited_by_count":2},{"year":2021,"cited_by_count":9},{"year":2020,"cited_by_count":3},{"year":2019,"cited_by_count":4},{"year":2018,"cited_by_count":4},{"year":2017,"cited_by_count":5},{"year":2016,"cited_by_count":4}],"updated_date":"2026-11-04T10:54:05.112534","created_date":"2016-06-24T00:00:00"}
