{"id":"https://openalex.org/W2078420177","doi":"https://doi.org/10.1016/0006-8993(78)90145-2","title":"Interaction of phencyclidines with the muscarinic and opiate receptors in the central nervous system","display_name":"Interaction of phencyclidines with the muscarinic and opiate receptors in the central nervous system","publication_year":1978,"publication_date":"1978-08-01","ids":{"openalex":"https://openalex.org/W2078420177","doi":"https://doi.org/10.1016/0006-8993(78)90145-2","mag":"2078420177","pmid":"https://pubmed.ncbi.nlm.nih.gov/79434"},"language":"en","primary_location":{"id":"doi:10.1016/0006-8993(78)90145-2","doi":"https://doi.org/10.1016/0006-8993(78)90145-2","is_oa":false,"landing_page_url":"https://doi.org/10.1016/0006-8993(78)90145-2","pdf_url":null,"source":{"id":"https://openalex.org/S96638545","display_name":"Brain Research","issn_l":"0006-8993","issn":["0006-8993","1872-6240"],"is_oa":false,"is_in_doaj":false,"is_core":true,"listed_in":["anvur-scientific","cwts-core","doyens","erih-plus","jufo-1","ki-jl-1","medline","norway-1","poland-100","russia-white-list-2","vabb-shw"],"host_organization":"https://openalex.org/P4310320990","host_organization_name":"Elsevier BV","host_organization_lineage":["https://openalex.org/P4310320990"],"host_organization_lineage_names":["Elsevier BV"],"type":"journal"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"Brain Research","raw_type":"journal-article"},"parent_works":[],"lineage":["https://openalex.org/W2078420177"],"child_works_count":0,"type":"article","is_traditional":true,"indexed_in":["crossref","pubmed"],"open_access":{"is_oa":false,"oa_status":"closed","oa_url":null,"any_repository_has_fulltext":false},"authorships":[{"author_position":"first","author":{"id":"https://openalex.org/A5108557967","display_name":"Jean\u2010Pierre Vincent","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I4210117840","display_name":"Institut de Biologie Valrose","ror":"https://ror.org/03bnma344","country_code":"FR","type":"facility","lineage":["https://openalex.org/I1294671590","https://openalex.org/I154526488","https://openalex.org/I201841394","https://openalex.org/I4210096427","https://openalex.org/I4210117840"]}],"countries":["FR"],"is_corresponding":false,"raw_author_name":"J.P. Vincent","raw_affiliation_strings":["Centre de Biochimie, Facult\u00e9des Sciences, Parc Valrose, 06034 Nice France"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Centre de Biochimie, Facult\u00e9des Sciences, Parc Valrose, 06034 Nice France","institution_ids":["https://openalex.org/I4210117840"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5025062255","display_name":"Daniel Cavey","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I4210117840","display_name":"Institut de Biologie Valrose","ror":"https://ror.org/03bnma344","country_code":"FR","type":"facility","lineage":["https://openalex.org/I1294671590","https://openalex.org/I154526488","https://openalex.org/I201841394","https://openalex.org/I4210096427","https://openalex.org/I4210117840"]}],"countries":["FR"],"is_corresponding":false,"raw_author_name":"D. Cavey","raw_affiliation_strings":["Centre de Biochimie, Facult\u00e9des Sciences, Parc Valrose, 06034 Nice France"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Centre de Biochimie, Facult\u00e9des Sciences, Parc Valrose, 06034 Nice France","institution_ids":["https://openalex.org/I4210117840"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5111739438","display_name":"Jean Marc Kamenka","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I11935315","display_name":"\u00c9cole Nationale Sup\u00e9rieure de Chimie de Montpellier","ror":"https://ror.org/03sgyqj04","country_code":"FR","type":"education","lineage":["https://openalex.org/I11935315","https://openalex.org/I19894307"]},{"id":"https://openalex.org/I4210117840","display_name":"Institut de Biologie Valrose","ror":"https://ror.org/03bnma344","country_code":"FR","type":"facility","lineage":["https://openalex.org/I1294671590","https://openalex.org/I154526488","https://openalex.org/I201841394","https://openalex.org/I4210096427","https://openalex.org/I4210117840"]}],"countries":["FR"],"is_corresponding":false,"raw_author_name":"J.M. Kamenka","raw_affiliation_strings":["Centre de Biochimie, Facult\u00e9des Sciences, Parc Valrose, 06034 Nice France","Laboratoire de Chimie Organique Physique Appliq\u00e9e, Ecole Nationale Sup\u00e9rieure de Chimie, 8 Rue Ecole Normale, 34075 Montpellier France"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Centre de Biochimie, Facult\u00e9des Sciences, Parc Valrose, 06034 Nice France","institution_ids":["https://openalex.org/I4210117840"]},{"raw_affiliation_string":"Laboratoire de Chimie Organique Physique Appliq\u00e9e, Ecole Nationale Sup\u00e9rieure de Chimie, 8 Rue Ecole Normale, 34075 Montpellier France","institution_ids":["https://openalex.org/I11935315"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5071795511","display_name":"PATRICK GENESTE","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I11935315","display_name":"\u00c9cole Nationale Sup\u00e9rieure de Chimie de Montpellier","ror":"https://ror.org/03sgyqj04","country_code":"FR","type":"education","lineage":["https://openalex.org/I11935315","https://openalex.org/I19894307"]},{"id":"https://openalex.org/I4210117840","display_name":"Institut de Biologie Valrose","ror":"https://ror.org/03bnma344","country_code":"FR","type":"facility","lineage":["https://openalex.org/I1294671590","https://openalex.org/I154526488","https://openalex.org/I201841394","https://openalex.org/I4210096427","https://openalex.org/I4210117840"]}],"countries":["FR"],"is_corresponding":false,"raw_author_name":"P. Geneste","raw_affiliation_strings":["Centre de Biochimie, Facult\u00e9des Sciences, Parc Valrose, 06034 Nice France","Laboratoire de Chimie Organique Physique Appliq\u00e9e, Ecole Nationale Sup\u00e9rieure de Chimie, 8 Rue Ecole Normale, 34075 Montpellier France"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Centre de Biochimie, Facult\u00e9des Sciences, Parc Valrose, 06034 Nice France","institution_ids":["https://openalex.org/I4210117840"]},{"raw_affiliation_string":"Laboratoire de Chimie Organique Physique Appliq\u00e9e, Ecole Nationale Sup\u00e9rieure de Chimie, 8 Rue Ecole Normale, 34075 Montpellier France","institution_ids":["https://openalex.org/I11935315"]}]},{"author_position":"last","author":{"id":"https://openalex.org/A5068045779","display_name":"Michel Lazdunski","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I4210117840","display_name":"Institut de Biologie Valrose","ror":"https://ror.org/03bnma344","country_code":"FR","type":"facility","lineage":["https://openalex.org/I1294671590","https://openalex.org/I154526488","https://openalex.org/I201841394","https://openalex.org/I4210096427","https://openalex.org/I4210117840"]}],"countries":["FR"],"is_corresponding":true,"raw_author_name":"M. Lazdunski","raw_affiliation_strings":["Centre de Biochimie, Facult\u00e9des Sciences, Parc Valrose, 06034 Nice France"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Centre de Biochimie, Facult\u00e9des Sciences, Parc Valrose, 06034 Nice France","institution_ids":["https://openalex.org/I4210117840"]}]}],"institutions":[],"countries_distinct_count":1,"institutions_distinct_count":2,"corresponding_author_ids":["https://openalex.org/A5068045779"],"corresponding_institution_ids":["https://openalex.org/I4210117840"],"apc_list":{"value":3360,"currency":"USD","value_usd":3360},"apc_paid":null,"fwci":4.0086,"has_fulltext":false,"cited_by_count":178,"citation_normalized_percentile":{"value":0.94869359,"is_in_top_1_percent":false,"is_in_top_10_percent":true},"cited_by_percentile_year":{"min":87,"max":95},"biblio":{"volume":"152","issue":"1","first_page":"176","last_page":"182"},"is_retracted":false,"is_paratext":false,"is_xpac":false,"primary_topic":{"id":"https://openalex.org/T10077","display_name":"Neuroscience and Neuropharmacology Research","score":0.25679999589920044,"subfield":{"id":"https://openalex.org/subfields/2804","display_name":"Cellular and Molecular Neuroscience"},"field":{"id":"https://openalex.org/fields/28","display_name":"Neuroscience"},"domain":{"id":"https://openalex.org/domains/1","display_name":"Life Sciences"}},"topics":[{"id":"https://openalex.org/T10077","display_name":"Neuroscience and Neuropharmacology Research","score":0.25679999589920044,"subfield":{"id":"https://openalex.org/subfields/2804","display_name":"Cellular and Molecular Neuroscience"},"field":{"id":"https://openalex.org/fields/28","display_name":"Neuroscience"},"domain":{"id":"https://openalex.org/domains/1","display_name":"Life Sciences"}},{"id":"https://openalex.org/T10800","display_name":"Forensic Toxicology and Drug Analysis","score":0.22579999268054962,"subfield":{"id":"https://openalex.org/subfields/3005","display_name":"Toxicology"},"field":{"id":"https://openalex.org/fields/30","display_name":"Pharmacology, Toxicology and Pharmaceutics"},"domain":{"id":"https://openalex.org/domains/1","display_name":"Life Sciences"}},{"id":"https://openalex.org/T10436","display_name":"Anesthesia and Sedative Agents","score":0.17409999668598175,"subfield":{"id":"https://openalex.org/subfields/2703","display_name":"Anesthesiology and Pain Medicine"},"field":{"id":"https://openalex.org/fields/27","display_name":"Medicine"},"domain":{"id":"https://openalex.org/domains/4","display_name":"Health Sciences"}}],"keywords":[{"id":"https://openalex.org/keywords/phencyclidine","display_name":"phencyclidine","score":0.9990000128746033},{"id":"https://openalex.org/keywords/ketamine","display_name":"ketamine","score":0.8640000224113464},{"id":"https://openalex.org/keywords/methoxetamine","display_name":"methoxetamine","score":0.9909999966621399},{"id":"https://openalex.org/keywords/nmda-receptor-antagonism","display_name":"NMDA receptor antagonism","score":0.8830000162124634},{"id":"https://openalex.org/keywords/muscarinic-receptors","display_name":"muscarinic receptors","score":0.968999981880188},{"id":"https://openalex.org/keywords/opioid-receptors","display_name":"opioid receptors","score":0.8769999742507935},{"id":"https://openalex.org/keywords/drug-toxicity","display_name":"drug toxicity","score":0.7039999961853027}],"concepts":[{"id":"https://openalex.org/C2778851735","wikidata":"https://www.wikidata.org/wiki/Q407324","display_name":"Phencyclidine","level":4,"score":0.8958656191825867},{"id":"https://openalex.org/C67018056","wikidata":"https://www.wikidata.org/wiki/Q414896","display_name":"NMDA receptor","level":3,"score":0.5915018320083618},{"id":"https://openalex.org/C98274493","wikidata":"https://www.wikidata.org/wiki/Q128406","display_name":"Pharmacology","level":1,"score":0.5679941773414612},{"id":"https://openalex.org/C2778140631","wikidata":"https://www.wikidata.org/wiki/Q2026938","display_name":"Opiate","level":3,"score":0.546738862991333},{"id":"https://openalex.org/C71924100","wikidata":"https://www.wikidata.org/wiki/Q11190","display_name":"Medicine","level":0,"score":0.509164035320282},{"id":"https://openalex.org/C124315065","wikidata":"https://www.wikidata.org/wiki/Q194270","display_name":"Hallucinogen","level":2,"score":0.5078476071357727},{"id":"https://openalex.org/C169760540","wikidata":"https://www.wikidata.org/wiki/Q207011","display_name":"Neuroscience","level":1,"score":0.4229472875595093},{"id":"https://openalex.org/C529278444","wikidata":"https://www.wikidata.org/wiki/Q47273","display_name":"Central nervous system","level":2,"score":0.4155467748641968},{"id":"https://openalex.org/C170493617","wikidata":"https://www.wikidata.org/wiki/Q208467","display_name":"Receptor","level":2,"score":0.2995472550392151},{"id":"https://openalex.org/C15744967","wikidata":"https://www.wikidata.org/wiki/Q9418","display_name":"Psychology","level":0,"score":0.29619598388671875},{"id":"https://openalex.org/C126322002","wikidata":"https://www.wikidata.org/wiki/Q11180","display_name":"Internal medicine","level":1,"score":0.14379560947418213}],"mesh":[{"descriptor_ui":"D000818","descriptor_name":"Animals","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D001667","descriptor_name":"Binding, Competitive","qualifier_ui":"Q000187","qualifier_name":"drug effects","is_major_topic":false},{"descriptor_ui":"D001921","descriptor_name":"Brain","qualifier_ui":"Q000378","qualifier_name":"metabolism","is_major_topic":false},{"descriptor_ui":"D004091","descriptor_name":"Hydromorphone","qualifier_ui":"Q000378","qualifier_name":"metabolism","is_major_topic":false},{"descriptor_ui":"D004347","descriptor_name":"Drug Interactions","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D010622","descriptor_name":"Phencyclidine","qualifier_ui":"Q000378","qualifier_name":"metabolism","is_major_topic":true},{"descriptor_ui":"D010622","descriptor_name":"Phencyclidine","qualifier_ui":"Q000494","qualifier_name":"pharmacology","is_major_topic":false},{"descriptor_ui":"D011812","descriptor_name":"Quinuclidines","qualifier_ui":"Q000378","qualifier_name":"metabolism","is_major_topic":false},{"descriptor_ui":"D011950","descriptor_name":"Receptors, Cholinergic","qualifier_ui":"Q000378","qualifier_name":"metabolism","is_major_topic":true},{"descriptor_ui":"D011957","descriptor_name":"Receptors, Opioid","qualifier_ui":"Q000378","qualifier_name":"metabolism","is_major_topic":true},{"descriptor_ui":"D011976","descriptor_name":"Receptors, Muscarinic","qualifier_ui":"Q000378","qualifier_name":"metabolism","is_major_topic":true},{"descriptor_ui":"D013237","descriptor_name":"Stereoisomerism","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D051381","descriptor_name":"Rats","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false}],"locations_count":2,"locations":[{"id":"doi:10.1016/0006-8993(78)90145-2","doi":"https://doi.org/10.1016/0006-8993(78)90145-2","is_oa":false,"landing_page_url":"https://doi.org/10.1016/0006-8993(78)90145-2","pdf_url":null,"source":{"id":"https://openalex.org/S96638545","display_name":"Brain Research","issn_l":"0006-8993","issn":["0006-8993","1872-6240"],"is_oa":false,"is_in_doaj":false,"is_core":true,"listed_in":["anvur-scientific","cwts-core","doyens","erih-plus","jufo-1","ki-jl-1","medline","norway-1","poland-100","russia-white-list-2","vabb-shw"],"host_organization":"https://openalex.org/P4310320990","host_organization_name":"Elsevier BV","host_organization_lineage":["https://openalex.org/P4310320990"],"host_organization_lineage_names":["Elsevier BV"],"type":"journal"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"Brain Research","raw_type":"journal-article"},{"id":"pmid:79434","doi":null,"is_oa":false,"landing_page_url":"https://pubmed.ncbi.nlm.nih.gov/79434","pdf_url":null,"source":{"id":"https://openalex.org/S4306525036","display_name":"PubMed","issn_l":null,"issn":null,"is_oa":false,"is_in_doaj":false,"is_core":false,"listed_in":[],"host_organization":"https://openalex.org/I1299303238","host_organization_name":"National Institutes of Health","host_organization_lineage":["https://openalex.org/I1299303238"],"host_organization_lineage_names":[],"type":"repository"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"Brain research","raw_type":"Journal Article"}],"best_oa_location":null,"sustainable_development_goals":[{"score":0.8048999905586243,"display_name":"Good health and well-being","id":"https://metadata.un.org/sdg/3"}],"study_designs":[],"awards":[],"funders":[],"has_content":{"grobid_xml":false,"pdf":false},"content_urls":null,"referenced_works_count":25,"referenced_works":["https://openalex.org/W196942043","https://openalex.org/W1534748687","https://openalex.org/W1840994181","https://openalex.org/W1969293801","https://openalex.org/W1977519142","https://openalex.org/W1980901689","https://openalex.org/W1993630443","https://openalex.org/W2000125000","https://openalex.org/W2014281089","https://openalex.org/W2019450096","https://openalex.org/W2023892570","https://openalex.org/W2027861706","https://openalex.org/W2030978007","https://openalex.org/W2050336058","https://openalex.org/W2069685558","https://openalex.org/W2080520820","https://openalex.org/W2093131407","https://openalex.org/W2115250531","https://openalex.org/W2138368199","https://openalex.org/W2307484198","https://openalex.org/W2335809166","https://openalex.org/W2417158750","https://openalex.org/W2530222122","https://openalex.org/W3027027291","https://openalex.org/W6607867490"],"related_works":["https://openalex.org/W4200590119","https://openalex.org/W2040237240","https://openalex.org/W4237246339","https://openalex.org/W4405542401","https://openalex.org/W1966529398","https://openalex.org/W4391215611","https://openalex.org/W2030152904","https://openalex.org/W4311957313","https://openalex.org/W2980732979","https://openalex.org/W2047375345"],"abstract_inverted_index":null,"counts_by_year":[{"year":2026,"cited_by_count":1},{"year":2024,"cited_by_count":1},{"year":2022,"cited_by_count":1},{"year":2021,"cited_by_count":1},{"year":2018,"cited_by_count":1},{"year":2017,"cited_by_count":1},{"year":2016,"cited_by_count":1},{"year":2015,"cited_by_count":1},{"year":2014,"cited_by_count":2}],"updated_date":"2026-11-13T13:42:25.865203","created_date":"2016-06-24T00:00:00"}
