{"id":"https://openalex.org/W2051560554","doi":"https://doi.org/10.1016/0006-2952(83)90081-3","title":"Inhibition of cytochrome oxidase activity by local anaesthetics","display_name":"Inhibition of cytochrome oxidase activity by local anaesthetics","publication_year":1983,"publication_date":"1983-09-01","ids":{"openalex":"https://openalex.org/W2051560554","doi":"https://doi.org/10.1016/0006-2952(83)90081-3","mag":"2051560554","pmid":"https://pubmed.ncbi.nlm.nih.gov/6313007"},"language":"en","primary_location":{"id":"doi:10.1016/0006-2952(83)90081-3","doi":"https://doi.org/10.1016/0006-2952(83)90081-3","is_oa":false,"landing_page_url":"https://doi.org/10.1016/0006-2952(83)90081-3","pdf_url":null,"source":{"id":"https://openalex.org/S185534594","display_name":"Biochemical Pharmacology","issn_l":"0006-2952","issn":["0006-2952","1873-2968"],"is_oa":false,"is_in_doaj":false,"is_core":true,"listed_in":["cwts-core","dongbi-c","doyens","jufo-2","ki-jl-1","medline","norway-1","poland-100","russia-white-list-1","vabb-shw"],"host_organization":"https://openalex.org/P4310320990","host_organization_name":"Elsevier BV","host_organization_lineage":["https://openalex.org/P4310320990"],"host_organization_lineage_names":["Elsevier BV"],"type":"journal"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"Biochemical Pharmacology","raw_type":"journal-article"},"volume":null,"type":"article","is_traditional":true,"indexed_in":["crossref","pubmed"],"open_access":{"is_oa":false,"oa_status":"closed","oa_url":null,"any_repository_has_fulltext":false},"authorships":[{"author_position":"first","author":{"id":null,"display_name":"A.M. Casanovas","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I4405258862","display_name":"Universit\u00e9 de Toulouse","ror":"https://ror.org/01ahyrz84","country_code":"FR","type":"education","lineage":["https://openalex.org/I4405258862"]}],"countries":["FR"],"is_corresponding":true,"raw_author_name":"A.M. Casanovas","raw_affiliation_strings":["Laboratoire de Biophysique et Biomath\u00e9matiques, Facult\u00e9 des Sciences Pharmaceutiques, 35 Chemin des Mara\u00eechers, 31062 Toulouse C\u00e9dex, France"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Laboratoire de Biophysique et Biomath\u00e9matiques, Facult\u00e9 des Sciences Pharmaceutiques, 35 Chemin des Mara\u00eechers, 31062 Toulouse C\u00e9dex, France","institution_ids":["https://openalex.org/I4405258862"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5035229772","display_name":"Marie-France Malmary","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I4405258862","display_name":"Universit\u00e9 de Toulouse","ror":"https://ror.org/01ahyrz84","country_code":"FR","type":"education","lineage":["https://openalex.org/I4405258862"]}],"countries":["FR"],"is_corresponding":false,"raw_author_name":"M.F. Malmary Nebot","raw_affiliation_strings":["Laboratoire de Biophysique et Biomath\u00e9matiques, Facult\u00e9 des Sciences Pharmaceutiques, 35 Chemin des Mara\u00eechers, 31062 Toulouse C\u00e9dex, France"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Laboratoire de Biophysique et Biomath\u00e9matiques, Facult\u00e9 des Sciences Pharmaceutiques, 35 Chemin des Mara\u00eechers, 31062 Toulouse C\u00e9dex, France","institution_ids":["https://openalex.org/I4405258862"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5108495255","display_name":"P. H. Courriere","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I4405258862","display_name":"Universit\u00e9 de Toulouse","ror":"https://ror.org/01ahyrz84","country_code":"FR","type":"education","lineage":["https://openalex.org/I4405258862"]}],"countries":["FR"],"is_corresponding":false,"raw_author_name":"Ph. Courri\u00e8re","raw_affiliation_strings":["Laboratoire de Biophysique et Biomath\u00e9matiques, Facult\u00e9 des Sciences Pharmaceutiques, 35 Chemin des Mara\u00eechers, 31062 Toulouse C\u00e9dex, France"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Laboratoire de Biophysique et Biomath\u00e9matiques, Facult\u00e9 des Sciences Pharmaceutiques, 35 Chemin des Mara\u00eechers, 31062 Toulouse C\u00e9dex, France","institution_ids":["https://openalex.org/I4405258862"]}]},{"author_position":"last","author":{"id":"https://openalex.org/A5000499509","display_name":"Jean Oustrin","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I4405258862","display_name":"Universit\u00e9 de Toulouse","ror":"https://ror.org/01ahyrz84","country_code":"FR","type":"education","lineage":["https://openalex.org/I4405258862"]}],"countries":["FR"],"is_corresponding":false,"raw_author_name":"J. Oustrin","raw_affiliation_strings":["Laboratoire de Biophysique et Biomath\u00e9matiques, Facult\u00e9 des Sciences Pharmaceutiques, 35 Chemin des Mara\u00eechers, 31062 Toulouse C\u00e9dex, France"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Laboratoire de Biophysique et Biomath\u00e9matiques, Facult\u00e9 des Sciences Pharmaceutiques, 35 Chemin des Mara\u00eechers, 31062 Toulouse C\u00e9dex, France","institution_ids":["https://openalex.org/I4405258862"]}]}],"institutions":[],"countries_distinct_count":1,"institutions_distinct_count":1,"corresponding_author_ids":[],"corresponding_institution_ids":["https://openalex.org/I4405258862"],"apc_list":{"value":3590,"currency":"USD","value_usd":3590},"apc_paid":null,"fwci":0.5342,"has_fulltext":false,"cited_by_count":18,"citation_normalized_percentile":{"value":0.55585995,"is_in_top_1_percent":false,"is_in_top_10_percent":false},"cited_by_percentile_year":{"min":88,"max":93},"biblio":{"volume":"32","issue":"18","first_page":"2715","last_page":"2719"},"is_retracted":false,"is_paratext":false,"is_xpac":false,"primary_topic":{"id":"https://openalex.org/T10301","display_name":"Mitochondrial Function and Pathology","score":0.5327000021934509,"subfield":{"id":"https://openalex.org/subfields/1312","display_name":"Molecular Biology"},"field":{"id":"https://openalex.org/fields/13","display_name":"Biochemistry, Genetics and Molecular Biology"},"domain":{"id":"https://openalex.org/domains/1","display_name":"Life Sciences"}},"topics":[{"id":"https://openalex.org/T10301","display_name":"Mitochondrial Function and Pathology","score":0.5327000021934509,"subfield":{"id":"https://openalex.org/subfields/1312","display_name":"Molecular Biology"},"field":{"id":"https://openalex.org/fields/13","display_name":"Biochemistry, Genetics and Molecular Biology"},"domain":{"id":"https://openalex.org/domains/1","display_name":"Life Sciences"}},{"id":"https://openalex.org/T10189","display_name":"Anesthesia and Pain Management","score":0.08950000256299973,"subfield":{"id":"https://openalex.org/subfields/2703","display_name":"Anesthesiology and Pain Medicine"},"field":{"id":"https://openalex.org/fields/27","display_name":"Medicine"},"domain":{"id":"https://openalex.org/domains/4","display_name":"Health Sciences"}},{"id":"https://openalex.org/T11908","display_name":"Protein Interaction Studies and Fluorescence Analysis","score":0.05209999904036522,"subfield":{"id":"https://openalex.org/subfields/1312","display_name":"Molecular Biology"},"field":{"id":"https://openalex.org/fields/13","display_name":"Biochemistry, Genetics and Molecular Biology"},"domain":{"id":"https://openalex.org/domains/1","display_name":"Life Sciences"}}],"keywords":[{"id":"https://openalex.org/keywords/local-anesthetics","display_name":"local anesthetics","score":0.9369999766349792},{"id":"https://openalex.org/keywords/cytochrome-c-oxidase","display_name":"cytochrome c oxidase","score":0.9819999933242798},{"id":"https://openalex.org/keywords/enzyme-inhibition","display_name":"enzyme inhibition","score":0.8209999799728394},{"id":"https://openalex.org/keywords/mitochondrial-electron-transport-chain","display_name":"mitochondrial electron transport chain","score":0.9700000286102295},{"id":"https://openalex.org/keywords/electrostatic-interactions","display_name":"electrostatic interactions","score":0.7799999713897705},{"id":"https://openalex.org/keywords/lipophilic-interactions","display_name":"lipophilic interactions","score":0.6620000004768372},{"id":"https://openalex.org/keywords/octanol-water-partition-coefficient","display_name":"octanol-water partition coefficient","score":0.9940000176429749}],"concepts":[{"id":"https://openalex.org/C123249941","wikidata":"https://www.wikidata.org/wiki/Q306116","display_name":"Cytochrome c oxidase","level":3,"score":0.7067131400108337},{"id":"https://openalex.org/C185592680","wikidata":"https://www.wikidata.org/wiki/Q2329","display_name":"Chemistry","level":0,"score":0.6910923719406128},{"id":"https://openalex.org/C3017770426","wikidata":"https://www.wikidata.org/wiki/Q1868462","display_name":"Local anaesthetic","level":2,"score":0.6607361435890198},{"id":"https://openalex.org/C2780768313","wikidata":"https://www.wikidata.org/wiki/Q408068","display_name":"Cytochrome","level":3,"score":0.4556252956390381},{"id":"https://openalex.org/C12554922","wikidata":"https://www.wikidata.org/wiki/Q7100","display_name":"Biophysics","level":1,"score":0.44904083013534546},{"id":"https://openalex.org/C29311851","wikidata":"https://www.wikidata.org/wiki/Q408223","display_name":"Cytochrome c","level":3,"score":0.4233795702457428},{"id":"https://openalex.org/C55493867","wikidata":"https://www.wikidata.org/wiki/Q7094","display_name":"Biochemistry","level":1,"score":0.4224146008491516},{"id":"https://openalex.org/C38485361","wikidata":"https://www.wikidata.org/wiki/Q576379","display_name":"Oxidase test","level":3,"score":0.4223192036151886},{"id":"https://openalex.org/C192552737","wikidata":"https://www.wikidata.org/wiki/Q898797","display_name":"Partition coefficient","level":2,"score":0.42142346501350403},{"id":"https://openalex.org/C181199279","wikidata":"https://www.wikidata.org/wiki/Q8047","display_name":"Enzyme","level":2,"score":0.4189299941062927},{"id":"https://openalex.org/C41625074","wikidata":"https://www.wikidata.org/wiki/Q176088","display_name":"Membrane","level":2,"score":0.4156964123249054},{"id":"https://openalex.org/C188518856","wikidata":"https://www.wikidata.org/wiki/Q899397","display_name":"Polarography","level":2,"score":0.41562575101852417},{"id":"https://openalex.org/C24840226","wikidata":"https://www.wikidata.org/wiki/Q211016","display_name":"Electron transport chain","level":2,"score":0.411306232213974},{"id":"https://openalex.org/C28859421","wikidata":"https://www.wikidata.org/wiki/Q39572","display_name":"Mitochondrion","level":2,"score":0.37751805782318115},{"id":"https://openalex.org/C86803240","wikidata":"https://www.wikidata.org/wiki/Q420","display_name":"Biology","level":0,"score":0.12132680416107178},{"id":"https://openalex.org/C42219234","wikidata":"https://www.wikidata.org/wiki/Q131130","display_name":"Anesthesia","level":1,"score":0.12037971615791321},{"id":"https://openalex.org/C43617362","wikidata":"https://www.wikidata.org/wiki/Q170050","display_name":"Chromatography","level":1,"score":0.10306274890899658},{"id":"https://openalex.org/C71924100","wikidata":"https://www.wikidata.org/wiki/Q11190","display_name":"Medicine","level":0,"score":0.0},{"id":"https://openalex.org/C179104552","wikidata":"https://www.wikidata.org/wiki/Q11165","display_name":"Inorganic chemistry","level":1,"score":0.0}],"mesh":[{"descriptor_ui":"D000779","descriptor_name":"Anesthetics, Local","qualifier_ui":"Q000494","qualifier_name":"pharmacology","is_major_topic":true},{"descriptor_ui":"D001667","descriptor_name":"Binding, Competitive","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D003576","descriptor_name":"Electron Transport Complex IV","qualifier_ui":"Q000037","qualifier_name":"antagonists & inhibitors","is_major_topic":true},{"descriptor_ui":"D007700","descriptor_name":"Kinetics","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D011048","descriptor_name":"Polarography","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D013329","descriptor_name":"Structure-Activity Relationship","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false}],"locations_count":2,"locations":[{"id":"doi:10.1016/0006-2952(83)90081-3","doi":"https://doi.org/10.1016/0006-2952(83)90081-3","is_oa":false,"landing_page_url":"https://doi.org/10.1016/0006-2952(83)90081-3","pdf_url":null,"source":{"id":"https://openalex.org/S185534594","display_name":"Biochemical Pharmacology","issn_l":"0006-2952","issn":["0006-2952","1873-2968"],"is_oa":false,"is_in_doaj":false,"is_core":true,"listed_in":["cwts-core","dongbi-c","doyens","jufo-2","ki-jl-1","medline","norway-1","poland-100","russia-white-list-1","vabb-shw"],"host_organization":"https://openalex.org/P4310320990","host_organization_name":"Elsevier BV","host_organization_lineage":["https://openalex.org/P4310320990"],"host_organization_lineage_names":["Elsevier BV"],"type":"journal"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"Biochemical Pharmacology","raw_type":"journal-article"},{"id":"pmid:6313007","doi":null,"is_oa":false,"landing_page_url":"https://pubmed.ncbi.nlm.nih.gov/6313007","pdf_url":null,"source":{"id":"https://openalex.org/S4306525036","display_name":"PubMed","issn_l":null,"issn":null,"is_oa":false,"is_in_doaj":false,"is_core":false,"listed_in":[],"host_organization":"https://openalex.org/I1299303238","host_organization_name":"National Institutes of Health","host_organization_lineage":["https://openalex.org/I1299303238"],"host_organization_lineage_names":[],"type":"repository"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"Biochemical pharmacology","raw_type":"Comparative Study"}],"best_oa_location":null,"sustainable_development_goals":[{"score":0.8048999905586243,"id":"https://metadata.un.org/sdg/3","display_name":"Good health and well-being"}],"study_designs":[],"awards":[],"funders":[],"has_content":{"pdf":false,"grobid_xml":false},"content_urls":null,"referenced_works_count":16,"referenced_works":["https://openalex.org/W1510944580","https://openalex.org/W1580198842","https://openalex.org/W1885778179","https://openalex.org/W1894569347","https://openalex.org/W1939618853","https://openalex.org/W1992287708","https://openalex.org/W1992656437","https://openalex.org/W2022864394","https://openalex.org/W2023042762","https://openalex.org/W2049322724","https://openalex.org/W2063869338","https://openalex.org/W2068312639","https://openalex.org/W2077406427","https://openalex.org/W2128265835","https://openalex.org/W2902079645","https://openalex.org/W3119784789"],"related_works":["https://openalex.org/W1510944580","https://openalex.org/W2122978519","https://openalex.org/W1811113994","https://openalex.org/W2438281171","https://openalex.org/W1992656437","https://openalex.org/W1988244124","https://openalex.org/W7208397189","https://openalex.org/W2402244000","https://openalex.org/W1968538813","https://openalex.org/W2419676508"],"abstract_inverted_index":null,"counts_by_year":[{"year":2014,"cited_by_count":1},{"year":2012,"cited_by_count":1}],"updated_date":"2026-10-31T12:09:11.096373","created_date":"2016-06-24T00:00:00"}
