{"id":"https://openalex.org/W2013754122","doi":"https://doi.org/10.1016/j.bcp.2011.07.020","title":"The (\u03b14)3(\u03b22)2 nAChR has a benzodiazepine-like modulatory binding site in the \u03b1\u03b1-subunit interface as revealed by studies with NS9283","display_name":"The (\u03b14)3(\u03b22)2 nAChR has a benzodiazepine-like modulatory binding site in the \u03b1\u03b1-subunit interface as revealed by studies with NS9283","publication_year":2011,"publication_date":"2011-08-22","ids":{"openalex":"https://openalex.org/W2013754122","doi":"https://doi.org/10.1016/j.bcp.2011.07.020","mag":"2013754122"},"language":"en","primary_location":{"id":"doi:10.1016/j.bcp.2011.07.020","doi":"https://doi.org/10.1016/j.bcp.2011.07.020","is_oa":false,"landing_page_url":"https://doi.org/10.1016/j.bcp.2011.07.020","pdf_url":null,"source":{"id":"https://openalex.org/S185534594","display_name":"Biochemical Pharmacology","issn_l":"0006-2952","issn":["0006-2952","1873-2968"],"is_oa":false,"is_in_doaj":false,"is_core":true,"listed_in":["cwts-core","dongbi-c","doyens","jufo-2","ki-jl-1","medline","norway-1","poland-100","russia-white-list-1","vabb-shw"],"host_organization":"https://openalex.org/P4310320990","host_organization_name":"Elsevier BV","host_organization_lineage":["https://openalex.org/P4310320990"],"host_organization_lineage_names":["Elsevier BV"],"type":"journal"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"Biochemical Pharmacology","raw_type":"journal-article"},"volume":null,"type":"article","is_traditional":true,"indexed_in":["crossref"],"open_access":{"is_oa":false,"oa_status":"closed","oa_url":null,"any_repository_has_fulltext":false},"authorships":[{"author_position":"first","author":{"id":"https://openalex.org/A5064333539","display_name":"Philip Ki\u00e6r Ahring","orcid":"https://orcid.org/0000-0003-1807-3331","observed_orcids":["https://orcid.org/0000-0003-1807-3331"]},"institutions":[{"id":"https://openalex.org/I4210118034","display_name":"NeuroSearch (Denmark)","ror":"https://ror.org/027x7jn80","country_code":"DK","type":"company","lineage":["https://openalex.org/I4210118034"]}],"countries":["DK"],"is_corresponding":true,"raw_author_name":"Philip K. Ahring","raw_affiliation_strings":["NeuroSearch A/S, Ballerup, Denmark"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"NeuroSearch A/S, Ballerup, Denmark","institution_ids":["https://openalex.org/I4210118034"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5084968972","display_name":"Dan Peters","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I4210118034","display_name":"NeuroSearch (Denmark)","ror":"https://ror.org/027x7jn80","country_code":"DK","type":"company","lineage":["https://openalex.org/I4210118034"]}],"countries":["DK"],"is_corresponding":false,"raw_author_name":"Dan Peters","raw_affiliation_strings":["NeuroSearch A/S, Ballerup, Denmark"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"NeuroSearch A/S, Ballerup, Denmark","institution_ids":["https://openalex.org/I4210118034"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5100517952","display_name":"Jeppe K. Christensen","orcid":"https://orcid.org/0009-0002-2330-881X","observed_orcids":["https://orcid.org/0009-0002-2330-881X"]},"institutions":[{"id":"https://openalex.org/I4210118034","display_name":"NeuroSearch (Denmark)","ror":"https://ror.org/027x7jn80","country_code":"DK","type":"company","lineage":["https://openalex.org/I4210118034"]}],"countries":["DK"],"is_corresponding":false,"raw_author_name":"Jeppe K. Christensen","raw_affiliation_strings":["NeuroSearch A/S, Ballerup, Denmark"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"NeuroSearch A/S, Ballerup, Denmark","institution_ids":["https://openalex.org/I4210118034"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5038439825","display_name":"Marianne Lerbech Jensen","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I4210118034","display_name":"NeuroSearch (Denmark)","ror":"https://ror.org/027x7jn80","country_code":"DK","type":"company","lineage":["https://openalex.org/I4210118034"]}],"countries":["DK"],"is_corresponding":false,"raw_author_name":"Marianne L. Jensen","raw_affiliation_strings":["NeuroSearch A/S, Ballerup, Denmark"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"NeuroSearch A/S, Ballerup, Denmark","institution_ids":["https://openalex.org/I4210118034"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5048035528","display_name":"Kasper Harps\u00f8e","orcid":"https://orcid.org/0000-0002-9326-9644","observed_orcids":["https://orcid.org/0000-0002-9326-9644"]},"institutions":[{"id":"https://openalex.org/I124055696","display_name":"University of Copenhagen","ror":"https://ror.org/035b05819","country_code":"DK","type":"education","lineage":["https://openalex.org/I124055696"]}],"countries":["DK"],"is_corresponding":false,"raw_author_name":"Kasper Harps\u00f8e","raw_affiliation_strings":["Department of Medicinal Chemistry, University of Copenhagen, Copenhagen, Denmark"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Department of Medicinal Chemistry, University of Copenhagen, Copenhagen, Denmark","institution_ids":["https://openalex.org/I124055696"]}]},{"author_position":"last","author":{"id":"https://openalex.org/A5069077291","display_name":"Thomas Balle","orcid":"https://orcid.org/0000-0002-0233-8350","observed_orcids":["https://orcid.org/0000-0002-0233-8350"]},"institutions":[{"id":"https://openalex.org/I124055696","display_name":"University of Copenhagen","ror":"https://ror.org/035b05819","country_code":"DK","type":"education","lineage":["https://openalex.org/I124055696"]}],"countries":["DK"],"is_corresponding":false,"raw_author_name":"Thomas Balle","raw_affiliation_strings":["Department of Medicinal Chemistry, University of Copenhagen, Copenhagen, Denmark"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Department of Medicinal Chemistry, University of Copenhagen, Copenhagen, Denmark","institution_ids":["https://openalex.org/I124055696"]}]}],"institutions":[],"countries_distinct_count":1,"institutions_distinct_count":2,"corresponding_author_ids":["https://openalex.org/A5064333539"],"corresponding_institution_ids":["https://openalex.org/I4210118034"],"apc_list":{"value":3590,"currency":"USD","value_usd":3590},"apc_paid":null,"fwci":0.0,"has_fulltext":false,"cited_by_count":1,"citation_normalized_percentile":{"value":0.09169215,"is_in_top_1_percent":false,"is_in_top_10_percent":false},"cited_by_percentile_year":{"min":88,"max":93},"biblio":{"volume":"82","issue":"8","first_page":"1029","last_page":"1030"},"is_retracted":false,"is_paratext":false,"is_xpac":false,"primary_topic":{"id":"https://openalex.org/T11818","display_name":"Nicotinic Acetylcholine Receptors Study","score":0.9990000128746033,"subfield":{"id":"https://openalex.org/subfields/1312","display_name":"Molecular Biology"},"field":{"id":"https://openalex.org/fields/13","display_name":"Biochemistry, Genetics and Molecular Biology"},"domain":{"id":"https://openalex.org/domains/1","display_name":"Life Sciences"}},"topics":[{"id":"https://openalex.org/T11818","display_name":"Nicotinic Acetylcholine Receptors Study","score":0.9990000128746033,"subfield":{"id":"https://openalex.org/subfields/1312","display_name":"Molecular Biology"},"field":{"id":"https://openalex.org/fields/13","display_name":"Biochemistry, Genetics and Molecular Biology"},"domain":{"id":"https://openalex.org/domains/1","display_name":"Life Sciences"}},{"id":"https://openalex.org/T10086","display_name":"Alzheimer's disease research and treatments","score":0.0005000000237487257,"subfield":{"id":"https://openalex.org/subfields/2804","display_name":"Cellular and Molecular Neuroscience"},"field":{"id":"https://openalex.org/fields/28","display_name":"Neuroscience"},"domain":{"id":"https://openalex.org/domains/1","display_name":"Life Sciences"}},{"id":"https://openalex.org/T10077","display_name":"Neuroscience and Neuropharmacology Research","score":0.00019999999494757503,"subfield":{"id":"https://openalex.org/subfields/2804","display_name":"Cellular and Molecular Neuroscience"},"field":{"id":"https://openalex.org/fields/28","display_name":"Neuroscience"},"domain":{"id":"https://openalex.org/domains/1","display_name":"Life Sciences"}}],"keywords":[{"id":"https://openalex.org/keywords/alpha7-nicotinic-acetylcholine-receptor","display_name":"alpha7 nicotinic acetylcholine receptor","score":0.9279999732971191},{"id":"https://openalex.org/keywords/alpha4beta2-nachr","display_name":"alpha4beta2 nAChR","score":0.7870000004768372},{"id":"https://openalex.org/keywords/galantamine","display_name":"galantamine","score":0.9700000286102295},{"id":"https://openalex.org/keywords/methyllycaconitine","display_name":"methyllycaconitine","score":0.8420000076293945},{"id":"https://openalex.org/keywords/amyloid-beta-25-35","display_name":"amyloid beta 25-35","score":0.8970000147819519},{"id":"https://openalex.org/keywords/alzheimer-s-disease","display_name":"Alzheimer's disease","score":0.9440000057220459},{"id":"https://openalex.org/keywords/cognitive-impairment","display_name":"cognitive impairment","score":0.8379999995231628},{"id":"https://openalex.org/keywords/working-memory","display_name":"working memory","score":0.7120000123977661},{"id":"https://openalex.org/keywords/reference-memory","display_name":"reference memory","score":0.972000002861023},{"id":"https://openalex.org/keywords/neuroprotection","display_name":"neuroprotection","score":0.8199999928474426}],"concepts":[{"id":"https://openalex.org/C2780374058","wikidata":"https://www.wikidata.org/wiki/Q3333710","display_name":"Methyllycaconitine","level":5,"score":0.8489025831222534},{"id":"https://openalex.org/C44752575","wikidata":"https://www.wikidata.org/wiki/Q1417562","display_name":"Morris water navigation task","level":3,"score":0.6268659234046936},{"id":"https://openalex.org/C98274493","wikidata":"https://www.wikidata.org/wiki/Q128406","display_name":"Pharmacology","level":1,"score":0.5686076283454895},{"id":"https://openalex.org/C185592680","wikidata":"https://www.wikidata.org/wiki/Q2329","display_name":"Chemistry","level":0,"score":0.5488161444664001},{"id":"https://openalex.org/C2778938600","wikidata":"https://www.wikidata.org/wiki/Q389934","display_name":"Agonist","level":3,"score":0.5461261868476868},{"id":"https://openalex.org/C2779570518","wikidata":"https://www.wikidata.org/wiki/Q412256","display_name":"Nicotinic acetylcholine receptor","level":4,"score":0.5151092410087585},{"id":"https://openalex.org/C188987157","wikidata":"https://www.wikidata.org/wiki/Q7030581","display_name":"Nicotinic agonist","level":3,"score":0.4665610194206238},{"id":"https://openalex.org/C170493617","wikidata":"https://www.wikidata.org/wiki/Q208467","display_name":"Receptor","level":2,"score":0.4214462637901306},{"id":"https://openalex.org/C134018914","wikidata":"https://www.wikidata.org/wiki/Q162606","display_name":"Endocrinology","level":1,"score":0.30657488107681274},{"id":"https://openalex.org/C71924100","wikidata":"https://www.wikidata.org/wiki/Q11190","display_name":"Medicine","level":0,"score":0.20143342018127441},{"id":"https://openalex.org/C2781161787","wikidata":"https://www.wikidata.org/wiki/Q48360","display_name":"Hippocampus","level":2,"score":0.19933781027793884},{"id":"https://openalex.org/C55493867","wikidata":"https://www.wikidata.org/wiki/Q7094","display_name":"Biochemistry","level":1,"score":0.1865123212337494}],"mesh":[],"locations_count":1,"locations":[{"id":"doi:10.1016/j.bcp.2011.07.020","doi":"https://doi.org/10.1016/j.bcp.2011.07.020","is_oa":false,"landing_page_url":"https://doi.org/10.1016/j.bcp.2011.07.020","pdf_url":null,"source":{"id":"https://openalex.org/S185534594","display_name":"Biochemical Pharmacology","issn_l":"0006-2952","issn":["0006-2952","1873-2968"],"is_oa":false,"is_in_doaj":false,"is_core":true,"listed_in":["cwts-core","dongbi-c","doyens","jufo-2","ki-jl-1","medline","norway-1","poland-100","russia-white-list-1","vabb-shw"],"host_organization":"https://openalex.org/P4310320990","host_organization_name":"Elsevier BV","host_organization_lineage":["https://openalex.org/P4310320990"],"host_organization_lineage_names":["Elsevier BV"],"type":"journal"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"Biochemical Pharmacology","raw_type":"journal-article"}],"best_oa_location":null,"sustainable_development_goals":[{"score":0.9391000270843506,"id":"https://metadata.un.org/sdg/3","display_name":"Good health and well-being"}],"study_designs":[],"awards":[],"funders":[],"has_content":{"pdf":false,"grobid_xml":false},"content_urls":null,"referenced_works_count":0,"referenced_works":[],"related_works":["https://openalex.org/W2014688027","https://openalex.org/W2328293891","https://openalex.org/W2120063222","https://openalex.org/W141939965","https://openalex.org/W4309631411","https://openalex.org/W2526009790","https://openalex.org/W2261295753","https://openalex.org/W2767064823","https://openalex.org/W2027131229","https://openalex.org/W2770200004"],"abstract_inverted_index":null,"counts_by_year":[{"year":2022,"cited_by_count":1}],"updated_date":"2026-11-04T10:54:05.112534","created_date":"2016-06-24T00:00:00"}
