{"id":"https://openalex.org/W2010508570","doi":"https://doi.org/10.1016/s0039-6060(97)90029-5","title":"Antiproliferative and antiinvasive effects of carboxyamido-triazole on breast cancer cell lines","display_name":"Antiproliferative and antiinvasive effects of carboxyamido-triazole on breast cancer cell lines","publication_year":1997,"publication_date":"1997-08-01","ids":{"openalex":"https://openalex.org/W2010508570","doi":"https://doi.org/10.1016/s0039-6060(97)90029-5","mag":"2010508570","pmid":"https://pubmed.ncbi.nlm.nih.gov/9288143"},"language":"en","primary_location":{"id":"doi:10.1016/s0039-6060(97)90029-5","doi":"https://doi.org/10.1016/s0039-6060(97)90029-5","is_oa":false,"landing_page_url":"https://doi.org/10.1016/s0039-6060(97)90029-5","pdf_url":null,"source":{"id":"https://openalex.org/S4210173306","display_name":"Surgery","issn_l":"0039-6060","issn":["0039-6060","1532-7361"],"is_oa":false,"is_in_doaj":false,"is_core":true,"listed_in":["anvur-scientific","cwts-core","dongbi-b","doyens","jufo-2","ki-jl-2","medline","norway-2","poland-100","russia-white-list-1"],"host_organization":"https://openalex.org/P4310320990","host_organization_name":"Elsevier BV","host_organization_lineage":["https://openalex.org/P4310320990"],"host_organization_lineage_names":["Elsevier BV"],"type":"journal"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"Surgery","raw_type":"journal-article"},"volume":null,"type":"article","indexed_in":["crossref","pubmed"],"open_access":{"is_oa":false,"oa_status":"closed","oa_url":null,"any_repository_has_fulltext":false},"authorships":[{"author_position":"first","author":{"id":"https://openalex.org/A5049020656","display_name":"Paul A. Lambert","orcid":"https://orcid.org/0000-0003-2287-3489","observed_orcids":["https://orcid.org/0000-0003-2287-3489"]},"institutions":[{"id":"https://openalex.org/I156802259","display_name":"Eastern Virginia Medical School","ror":"https://ror.org/056hr4255","country_code":"US","type":"education","lineage":["https://openalex.org/I156802259"]},{"id":"https://openalex.org/I4210140884","display_name":"National Cancer Institute","ror":"https://ror.org/040gcmg81","country_code":"US","type":"government","lineage":["https://openalex.org/I1299022934","https://openalex.org/I1299303238","https://openalex.org/I4210140884"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"Paul A Lambert","raw_affiliation_strings":["Department of Surgery, Eastern Virginia Medical School, Norfolk 23507, USA","From the Departments of Surgery, Microbiology, and Immunology, Eastern Virginia Medical School, Norfolk, Va., USA","From the Laboratory of Pathology, National Cancer Institute, Bethesda, Md., USA"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Department of Surgery, Eastern Virginia Medical School, Norfolk 23507, USA","institution_ids":["https://openalex.org/I156802259"]},{"raw_affiliation_string":"From the Departments of Surgery, Microbiology, and Immunology, Eastern Virginia Medical School, Norfolk, Va., USA","institution_ids":["https://openalex.org/I156802259"]},{"raw_affiliation_string":"From the Laboratory of Pathology, National Cancer Institute, Bethesda, Md., USA","institution_ids":["https://openalex.org/I4210140884"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5112151011","display_name":"Kenneth D. Somers","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I156802259","display_name":"Eastern Virginia Medical School","ror":"https://ror.org/056hr4255","country_code":"US","type":"education","lineage":["https://openalex.org/I156802259"]},{"id":"https://openalex.org/I4210140884","display_name":"National Cancer Institute","ror":"https://ror.org/040gcmg81","country_code":"US","type":"government","lineage":["https://openalex.org/I1299022934","https://openalex.org/I1299303238","https://openalex.org/I4210140884"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"Kenneth D Somers","raw_affiliation_strings":["From the Departments of Surgery, Microbiology, and Immunology, Eastern Virginia Medical School, Norfolk, Va., USA","From the Laboratory of Pathology, National Cancer Institute, Bethesda, Md., USA"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"From the Departments of Surgery, Microbiology, and Immunology, Eastern Virginia Medical School, Norfolk, Va., USA","institution_ids":["https://openalex.org/I156802259"]},{"raw_affiliation_string":"From the Laboratory of Pathology, National Cancer Institute, Bethesda, Md., USA","institution_ids":["https://openalex.org/I4210140884"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5005621340","display_name":"Elise C. Kohn","orcid":"https://orcid.org/0000-0002-8631-9762","observed_orcids":["https://orcid.org/0000-0002-8631-9762"]},"institutions":[{"id":"https://openalex.org/I156802259","display_name":"Eastern Virginia Medical School","ror":"https://ror.org/056hr4255","country_code":"US","type":"education","lineage":["https://openalex.org/I156802259"]},{"id":"https://openalex.org/I4210140884","display_name":"National Cancer Institute","ror":"https://ror.org/040gcmg81","country_code":"US","type":"government","lineage":["https://openalex.org/I1299022934","https://openalex.org/I1299303238","https://openalex.org/I4210140884"]}],"countries":["US"],"is_corresponding":false,"raw_author_name":"Elise C Kohn","raw_affiliation_strings":["From the Departments of Surgery, Microbiology, and Immunology, Eastern Virginia Medical School, Norfolk, Va., USA","From the Laboratory of Pathology, National Cancer Institute, Bethesda, Md., USA"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"From the Departments of Surgery, Microbiology, and Immunology, Eastern Virginia Medical School, Norfolk, Va., USA","institution_ids":["https://openalex.org/I156802259"]},{"raw_affiliation_string":"From the Laboratory of Pathology, National Cancer Institute, Bethesda, Md., USA","institution_ids":["https://openalex.org/I4210140884"]}]},{"author_position":"last","author":{"id":"https://openalex.org/A5000472567","display_name":"Roger R Perry","orcid":"https://orcid.org/0000-0001-9726-3402","observed_orcids":["https://orcid.org/0000-0001-9726-3402"]},"institutions":[{"id":"https://openalex.org/I156802259","display_name":"Eastern Virginia Medical School","ror":"https://ror.org/056hr4255","country_code":"US","type":"education","lineage":["https://openalex.org/I156802259"]},{"id":"https://openalex.org/I4210140884","display_name":"National Cancer Institute","ror":"https://ror.org/040gcmg81","country_code":"US","type":"government","lineage":["https://openalex.org/I1299022934","https://openalex.org/I1299303238","https://openalex.org/I4210140884"]}],"countries":["US"],"is_corresponding":true,"raw_author_name":"Roger R Perry","raw_affiliation_strings":["From the Departments of Surgery, Microbiology, and Immunology, Eastern Virginia Medical School, Norfolk, Va., USA","From the Laboratory of Pathology, National Cancer Institute, Bethesda, Md., USA"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"From the Departments of Surgery, Microbiology, and Immunology, Eastern Virginia Medical School, Norfolk, Va., USA","institution_ids":["https://openalex.org/I156802259"]},{"raw_affiliation_string":"From the Laboratory of Pathology, National Cancer Institute, Bethesda, Md., USA","institution_ids":["https://openalex.org/I4210140884"]}]}],"institutions":[],"countries_distinct_count":1,"institutions_distinct_count":2,"corresponding_author_ids":["https://openalex.org/A5000472567"],"corresponding_institution_ids":["https://openalex.org/I156802259","https://openalex.org/I4210140884"],"apc_list":{"value":4130,"currency":"USD","value_usd":4130},"apc_paid":null,"fwci":1.0667,"has_fulltext":false,"cited_by_count":48,"citation_normalized_percentile":{"value":0.75452532,"is_in_top_1_percent":false,"is_in_top_10_percent":false},"cited_by_percentile_year":{"min":89,"max":96},"biblio":{"volume":"122","issue":"2","first_page":"372","last_page":"379"},"is_retracted":false,"is_paratext":false,"is_xpac":false,"primary_topic":{"id":"https://openalex.org/T13437","display_name":"Mechanisms of cancer metastasis","score":0.5663999915122986,"subfield":{"id":"https://openalex.org/subfields/1312","display_name":"Molecular Biology"},"field":{"id":"https://openalex.org/fields/13","display_name":"Biochemistry, Genetics and Molecular Biology"},"domain":{"id":"https://openalex.org/domains/1","display_name":"Life Sciences"}},"topics":[{"id":"https://openalex.org/T13437","display_name":"Mechanisms of cancer metastasis","score":0.5663999915122986,"subfield":{"id":"https://openalex.org/subfields/1312","display_name":"Molecular Biology"},"field":{"id":"https://openalex.org/fields/13","display_name":"Biochemistry, Genetics and Molecular Biology"},"domain":{"id":"https://openalex.org/domains/1","display_name":"Life Sciences"}},{"id":"https://openalex.org/T10620","display_name":"Protease and Inhibitor Mechanisms","score":0.20000000298023224,"subfield":{"id":"https://openalex.org/subfields/1306","display_name":"Cancer Research"},"field":{"id":"https://openalex.org/fields/13","display_name":"Biochemistry, Genetics and Molecular Biology"},"domain":{"id":"https://openalex.org/domains/1","display_name":"Life Sciences"}},{"id":"https://openalex.org/T10336","display_name":"Cancer Cells and Metastasis","score":0.13590000569820404,"subfield":{"id":"https://openalex.org/subfields/2730","display_name":"Oncology"},"field":{"id":"https://openalex.org/fields/27","display_name":"Medicine"},"domain":{"id":"https://openalex.org/domains/4","display_name":"Health Sciences"}}],"keywords":[{"id":"https://openalex.org/keywords/breast-cancer","display_name":"breast cancer","score":0.8019999861717224},{"id":"https://openalex.org/keywords/cell-invasion","display_name":"cell invasion","score":0.5839999914169312},{"id":"https://openalex.org/keywords/antiproliferative-activity","display_name":"antiproliferative activity","score":0.8920000195503235},{"id":"https://openalex.org/keywords/calcium-influx-inhibition","display_name":"calcium influx inhibition","score":0.8109999895095825},{"id":"https://openalex.org/keywords/matrix-metalloproteinases","display_name":"matrix metalloproteinases","score":0.8650000095367432},{"id":"https://openalex.org/keywords/estrogen-receptor","display_name":"estrogen receptor","score":0.5590000152587891},{"id":"https://openalex.org/keywords/p-glycoprotein","display_name":"P-glycoprotein","score":0.9710000157356262},{"id":"https://openalex.org/keywords/drug-resistance","display_name":"drug resistance","score":0.7139999866485596},{"id":"https://openalex.org/keywords/metastasis","display_name":"metastasis","score":0.7049999833106995},{"id":"https://openalex.org/keywords/mcf-7-cells","display_name":"MCF-7 cells","score":0.7699999809265137},{"id":"https://openalex.org/keywords/mda-mb-231-cells","display_name":"MDA-MB-231 cells","score":0.9570000171661377},{"id":"https://openalex.org/keywords/bt474-cells","display_name":"BT474 cells","score":0.996999979019165}],"concepts":[{"id":"https://openalex.org/C71924100","wikidata":"https://www.wikidata.org/wiki/Q11190","display_name":"Medicine","level":0,"score":0.6674309372901917},{"id":"https://openalex.org/C81885089","wikidata":"https://www.wikidata.org/wiki/Q189082","display_name":"Cell culture","level":2,"score":0.6545450091362},{"id":"https://openalex.org/C2778608917","wikidata":"https://www.wikidata.org/wiki/Q6787805","display_name":"Matrigel","level":3,"score":0.6462511420249939},{"id":"https://openalex.org/C84606932","wikidata":"https://www.wikidata.org/wiki/Q416496","display_name":"Estrogen receptor","level":4,"score":0.5964376926422119},{"id":"https://openalex.org/C2775958869","wikidata":"https://www.wikidata.org/wiki/Q16966320","display_name":"Matrix metalloproteinase inhibitor","level":3,"score":0.5331719517707825},{"id":"https://openalex.org/C109523444","wikidata":"https://www.wikidata.org/wiki/Q424216","display_name":"Matrix metalloproteinase","level":2,"score":0.5329568982124329},{"id":"https://openalex.org/C177430391","wikidata":"https://www.wikidata.org/wiki/Q1173648","display_name":"Zymography","level":3,"score":0.46112698316574097},{"id":"https://openalex.org/C109541995","wikidata":"https://www.wikidata.org/wiki/Q1881253","display_name":"MCF-7","level":5,"score":0.4580163061618805},{"id":"https://openalex.org/C2776193487","wikidata":"https://www.wikidata.org/wiki/Q32846","display_name":"Basement membrane","level":2,"score":0.42494791746139526},{"id":"https://openalex.org/C502942594","wikidata":"https://www.wikidata.org/wiki/Q3421914","display_name":"Cancer research","level":1,"score":0.385846883058548},{"id":"https://openalex.org/C153911025","wikidata":"https://www.wikidata.org/wiki/Q7202","display_name":"Molecular biology","level":1,"score":0.37372806668281555},{"id":"https://openalex.org/C96232424","wikidata":"https://www.wikidata.org/wiki/Q4118072","display_name":"Cancer cell","level":3,"score":0.3699432909488678},{"id":"https://openalex.org/C530470458","wikidata":"https://www.wikidata.org/wiki/Q128581","display_name":"Breast cancer","level":3,"score":0.3447492718696594},{"id":"https://openalex.org/C142724271","wikidata":"https://www.wikidata.org/wiki/Q7208","display_name":"Pathology","level":1,"score":0.33536064624786377},{"id":"https://openalex.org/C121608353","wikidata":"https://www.wikidata.org/wiki/Q12078","display_name":"Cancer","level":2,"score":0.3004504442214966},{"id":"https://openalex.org/C126322002","wikidata":"https://www.wikidata.org/wiki/Q11180","display_name":"Internal medicine","level":1,"score":0.2984025180339813},{"id":"https://openalex.org/C2780394083","wikidata":"https://www.wikidata.org/wiki/Q539568","display_name":"Angiogenesis","level":2,"score":0.22583332657814026},{"id":"https://openalex.org/C86803240","wikidata":"https://www.wikidata.org/wiki/Q420","display_name":"Biology","level":0,"score":0.21333715319633484},{"id":"https://openalex.org/C2994423619","wikidata":"https://www.wikidata.org/wiki/Q9103","display_name":"Human breast","level":4,"score":0.14795410633087158},{"id":"https://openalex.org/C54355233","wikidata":"https://www.wikidata.org/wiki/Q7162","display_name":"Genetics","level":1,"score":0.0}],"mesh":[{"descriptor_ui":"D000970","descriptor_name":"Antineoplastic Agents","qualifier_ui":"Q000633","qualifier_name":"toxicity","is_major_topic":true},{"descriptor_ui":"D001943","descriptor_name":"Breast Neoplasms","qualifier_ui":"Q000473","qualifier_name":"pathology","is_major_topic":true},{"descriptor_ui":"D002121","descriptor_name":"Calcium Channel Blockers","qualifier_ui":"Q000633","qualifier_name":"toxicity","is_major_topic":false},{"descriptor_ui":"D002470","descriptor_name":"Cell Survival","qualifier_ui":"Q000187","qualifier_name":"drug effects","is_major_topic":false},{"descriptor_ui":"D004354","descriptor_name":"Drug Screening Assays, Antitumor","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D005260","descriptor_name":"Female","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D006801","descriptor_name":"Humans","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D008666","descriptor_name":"Metalloendopeptidases","qualifier_ui":"Q000378","qualifier_name":"metabolism","is_major_topic":false},{"descriptor_ui":"D009361","descriptor_name":"Neoplasm Invasiveness","qualifier_ui":"Q000517","qualifier_name":"prevention & control","is_major_topic":false},{"descriptor_ui":"D011960","descriptor_name":"Receptors, Estrogen","qualifier_ui":"Q000032","qualifier_name":"analysis","is_major_topic":false},{"descriptor_ui":"D014230","descriptor_name":"Triazoles","qualifier_ui":"Q000633","qualifier_name":"toxicity","is_major_topic":true},{"descriptor_ui":"D014407","descriptor_name":"Tumor Cells, Cultured","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D017364","descriptor_name":"Collagenases","qualifier_ui":"Q000378","qualifier_name":"metabolism","is_major_topic":false},{"descriptor_ui":"D018093","descriptor_name":"Gelatinases","qualifier_ui":"Q000378","qualifier_name":"metabolism","is_major_topic":false},{"descriptor_ui":"D020168","descriptor_name":"ATP Binding Cassette Transporter, Subfamily B, Member 1","qualifier_ui":"Q000032","qualifier_name":"analysis","is_major_topic":false},{"descriptor_ui":"D020778","descriptor_name":"Matrix Metalloproteinase 2","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D020780","descriptor_name":"Matrix Metalloproteinase 9","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false}],"locations_count":2,"locations":[{"id":"doi:10.1016/s0039-6060(97)90029-5","doi":"https://doi.org/10.1016/s0039-6060(97)90029-5","is_oa":false,"landing_page_url":"https://doi.org/10.1016/s0039-6060(97)90029-5","pdf_url":null,"source":{"id":"https://openalex.org/S4210173306","display_name":"Surgery","issn_l":"0039-6060","issn":["0039-6060","1532-7361"],"is_oa":false,"is_in_doaj":false,"is_core":true,"listed_in":["anvur-scientific","cwts-core","dongbi-b","doyens","jufo-2","ki-jl-2","medline","norway-2","poland-100","russia-white-list-1"],"host_organization":"https://openalex.org/P4310320990","host_organization_name":"Elsevier BV","host_organization_lineage":["https://openalex.org/P4310320990"],"host_organization_lineage_names":["Elsevier BV"],"type":"journal"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"Surgery","raw_type":"journal-article"},{"id":"pmid:9288143","doi":null,"is_oa":false,"landing_page_url":"https://pubmed.ncbi.nlm.nih.gov/9288143","pdf_url":null,"source":{"id":"https://openalex.org/S4306525036","display_name":"PubMed","issn_l":null,"issn":null,"is_oa":false,"is_in_doaj":false,"is_core":false,"listed_in":[],"host_organization":"https://openalex.org/I1299303238","host_organization_name":"National Institutes of Health","host_organization_lineage":["https://openalex.org/I1299303238"],"host_organization_lineage_names":[],"type":"repository"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"Surgery","raw_type":"Journal Article"}],"best_oa_location":null,"sustainable_development_goals":[{"score":0.9763000011444092,"display_name":"Good health and well-being","id":"https://metadata.un.org/sdg/3"}],"sustainable_development_goals_aurora":[{"score":0.7900000214576721,"display_name":"Good health and well-being","id":"https://metadata.un.org/sdg/3"}],"study_designs":[],"awards":[],"funders":[],"has_content":{"grobid_xml":false,"pdf":false},"content_urls":null,"referenced_works_count":29,"referenced_works":["https://openalex.org/W1513691409","https://openalex.org/W1522871208","https://openalex.org/W1561226826","https://openalex.org/W1785041189","https://openalex.org/W1835282334","https://openalex.org/W1882182790","https://openalex.org/W1912071596","https://openalex.org/W1938617858","https://openalex.org/W1947125836","https://openalex.org/W2022732160","https://openalex.org/W2026151657","https://openalex.org/W2028063907","https://openalex.org/W2030686317","https://openalex.org/W2086640970","https://openalex.org/W2097616269","https://openalex.org/W2115653616","https://openalex.org/W2123238323","https://openalex.org/W2128018446","https://openalex.org/W2140927361","https://openalex.org/W2148553679","https://openalex.org/W2148890841","https://openalex.org/W2164629825","https://openalex.org/W2166105996","https://openalex.org/W2166452296","https://openalex.org/W2213636196","https://openalex.org/W2418070516","https://openalex.org/W6635512558","https://openalex.org/W6639266806","https://openalex.org/W6640100049"],"related_works":["https://openalex.org/W2022732160","https://openalex.org/W2113928000","https://openalex.org/W34501388","https://openalex.org/W2016592183","https://openalex.org/W1552180547","https://openalex.org/W1973415395","https://openalex.org/W31174271","https://openalex.org/W3017658449","https://openalex.org/W2071381923","https://openalex.org/W2296911346"],"abstract_inverted_index":null,"counts_by_year":[{"year":2023,"cited_by_count":2},{"year":2021,"cited_by_count":2},{"year":2020,"cited_by_count":2},{"year":2018,"cited_by_count":2},{"year":2015,"cited_by_count":1},{"year":2014,"cited_by_count":1}],"updated_date":"2026-10-31T12:09:11.096373","created_date":"2016-06-24T00:00:00"}
