{"id":"https://openalex.org/W2009220054","doi":"https://doi.org/10.1194/jlr.r024075","title":"Cholesteryl ester transfer protein inhibition as a strategy to reduce cardiovascular risk","display_name":"Cholesteryl ester transfer protein inhibition as a strategy to reduce cardiovascular risk","publication_year":2012,"publication_date":"2012-05-02","ids":{"openalex":"https://openalex.org/W2009220054","doi":"https://doi.org/10.1194/jlr.r024075","mag":"2009220054","pmid":"https://pubmed.ncbi.nlm.nih.gov/22550134","pmcid":"https://www.ncbi.nlm.nih.gov/pmc/articles/3413218"},"language":"en","primary_location":{"id":"doi:10.1194/jlr.r024075","doi":"https://doi.org/10.1194/jlr.r024075","is_oa":true,"landing_page_url":"https://doi.org/10.1194/jlr.r024075","pdf_url":"http://www.jlr.org/content/53/9/1755.full.pdf","source":{"id":"https://openalex.org/S11400418","display_name":"Journal of Lipid Research","issn_l":"0022-2275","issn":["0022-2275","1539-7262"],"is_oa":false,"is_in_doaj":true,"is_core":true,"listed_in":["cwts-core","doaj","dongbi-c","doyens","jufo-1","ki-jl-1","medline","norway-1","oarl","poland-140","vabb-shw"],"host_organization":"https://openalex.org/P4310320990","host_organization_name":"Elsevier BV","host_organization_lineage":["https://openalex.org/P4310320990"],"host_organization_lineage_names":["Elsevier BV"],"type":"journal"},"license":"cc-by","license_id":"https://openalex.org/licenses/cc-by","version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"Journal of Lipid Research","raw_type":"journal-article"},"volume":null,"type":"review","is_traditional":true,"indexed_in":["crossref","doaj","pubmed"],"open_access":{"is_oa":true,"oa_status":"hybrid","oa_url":"http://www.jlr.org/content/53/9/1755.full.pdf","any_repository_has_fulltext":true},"authorships":[{"author_position":"first","author":{"id":"https://openalex.org/A5013655811","display_name":"Philip J. Barter","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I129604602","display_name":"The University of Sydney","ror":"https://ror.org/0384j8v12","country_code":"AU","type":"education","lineage":["https://openalex.org/I129604602"]},{"id":"https://openalex.org/I2801241159","display_name":"The Heart Research Institute","ror":"https://ror.org/046fa4y88","country_code":"AU","type":"facility","lineage":["https://openalex.org/I2801241159"]}],"countries":["AU"],"is_corresponding":true,"raw_author_name":"Philip J. Barter","raw_affiliation_strings":["The Heart Research Institute, Sydney, New South Wales, 2042, Australia. barter@hri.org.au","*The Heart Research Institute, Sydney, New South Wales, 2042, Australia","Faculty of Medicine, University of Sydney, Sydney, New South Wales, 2006, Australia"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"The Heart Research Institute, Sydney, New South Wales, 2042, Australia. barter@hri.org.au","institution_ids":["https://openalex.org/I2801241159"]},{"raw_affiliation_string":"*The Heart Research Institute, Sydney, New South Wales, 2042, Australia","institution_ids":["https://openalex.org/I2801241159"]},{"raw_affiliation_string":"Faculty of Medicine, University of Sydney, Sydney, New South Wales, 2006, Australia","institution_ids":["https://openalex.org/I129604602"]}]},{"author_position":"last","author":{"id":"https://openalex.org/A5110733633","display_name":"K.-A. Rye","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I129604602","display_name":"The University of Sydney","ror":"https://ror.org/0384j8v12","country_code":"AU","type":"education","lineage":["https://openalex.org/I129604602"]},{"id":"https://openalex.org/I165779595","display_name":"The University of Melbourne","ror":"https://ror.org/01ej9dk98","country_code":"AU","type":"education","lineage":["https://openalex.org/I165779595"]},{"id":"https://openalex.org/I2801241159","display_name":"The Heart Research Institute","ror":"https://ror.org/046fa4y88","country_code":"AU","type":"facility","lineage":["https://openalex.org/I2801241159"]}],"countries":["AU"],"is_corresponding":false,"raw_author_name":"Kerry-Anne Rye","raw_affiliation_strings":["Department of Medicine, University of Melbourne, Melbourne, Victoria, 3010, Australia","Faculty of Medicine, University of Sydney, Sydney, New South Wales, 2006, Australia","The Heart Research Institute, Sydney, New South Wales, 2042, Australia"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Department of Medicine, University of Melbourne, Melbourne, Victoria, 3010, Australia","institution_ids":["https://openalex.org/I165779595"]},{"raw_affiliation_string":"Faculty of Medicine, University of Sydney, Sydney, New South Wales, 2006, Australia","institution_ids":["https://openalex.org/I129604602"]},{"raw_affiliation_string":"The Heart Research Institute, Sydney, New South Wales, 2042, Australia","institution_ids":["https://openalex.org/I2801241159"]}]}],"institutions":[],"countries_distinct_count":1,"institutions_distinct_count":3,"corresponding_author_ids":["https://openalex.org/A5013655811"],"corresponding_institution_ids":["https://openalex.org/I129604602","https://openalex.org/I2801241159"],"apc_list":{"value":3430,"currency":"USD","value_usd":3430},"apc_paid":{"value":3430,"currency":"USD","value_usd":3430},"fwci":3.7648,"has_fulltext":true,"cited_by_count":148,"citation_normalized_percentile":{"value":0.96372348,"is_in_top_1_percent":false,"is_in_top_10_percent":true},"cited_by_percentile_year":{"min":93,"max":100},"biblio":{"volume":"53","issue":"9","first_page":"1755","last_page":"1766"},"is_retracted":false,"is_paratext":false,"is_xpac":false,"primary_topic":{"id":"https://openalex.org/T10394","display_name":"Lipoproteins and Cardiovascular Health","score":0.6807000041007996,"subfield":{"id":"https://openalex.org/subfields/2705","display_name":"Cardiology and Cardiovascular Medicine"},"field":{"id":"https://openalex.org/fields/27","display_name":"Medicine"},"domain":{"id":"https://openalex.org/domains/4","display_name":"Health Sciences"}},"topics":[{"id":"https://openalex.org/T10394","display_name":"Lipoproteins and Cardiovascular Health","score":0.6807000041007996,"subfield":{"id":"https://openalex.org/subfields/2705","display_name":"Cardiology and Cardiovascular Medicine"},"field":{"id":"https://openalex.org/fields/27","display_name":"Medicine"},"domain":{"id":"https://openalex.org/domains/4","display_name":"Health Sciences"}},{"id":"https://openalex.org/T11618","display_name":"Cholesterol and Lipid Metabolism","score":0.2992999851703644,"subfield":{"id":"https://openalex.org/subfields/1303","display_name":"Biochemistry"},"field":{"id":"https://openalex.org/fields/13","display_name":"Biochemistry, Genetics and Molecular Biology"},"domain":{"id":"https://openalex.org/domains/1","display_name":"Life Sciences"}},{"id":"https://openalex.org/T12975","display_name":"Paraoxonase enzyme and polymorphisms","score":0.0071000000461936,"subfield":{"id":"https://openalex.org/subfields/1308","display_name":"Clinical Biochemistry"},"field":{"id":"https://openalex.org/fields/13","display_name":"Biochemistry, Genetics and Molecular Biology"},"domain":{"id":"https://openalex.org/domains/1","display_name":"Life Sciences"}}],"keywords":[{"id":"https://openalex.org/keywords/cholesteryl-ester-transfer-protein","display_name":"cholesteryl ester transfer protein","score":0.9679999947547913},{"id":"https://openalex.org/keywords/cetp-inhibition","display_name":"CETP inhibition","score":0.8489999771118164},{"id":"https://openalex.org/keywords/torcetrapib","display_name":"torcetrapib","score":0.871999979019165},{"id":"https://openalex.org/keywords/dalcetrapib","display_name":"dalcetrapib","score":0.9990000128746033},{"id":"https://openalex.org/keywords/anacetrapib","display_name":"anacetrapib","score":0.9800000190734863},{"id":"https://openalex.org/keywords/evacetrapib","display_name":"evacetrapib","score":1.0},{"id":"https://openalex.org/keywords/hdl-cholesterol","display_name":"HDL cholesterol","score":0.9290000200271606},{"id":"https://openalex.org/keywords/atherosclerosis","display_name":"atherosclerosis","score":0.8560000061988831},{"id":"https://openalex.org/keywords/cardiovascular-risk-reduction","display_name":"cardiovascular risk reduction","score":0.8830000162124634},{"id":"https://openalex.org/keywords/lipoprotein-metabolism","display_name":"lipoprotein metabolism","score":0.47699999809265137}],"concepts":[{"id":"https://openalex.org/C45505151","wikidata":"https://www.wikidata.org/wiki/Q424706","display_name":"Cholesterylester transfer protein","level":4,"score":0.9933586716651917},{"id":"https://openalex.org/C185592680","wikidata":"https://www.wikidata.org/wiki/Q2329","display_name":"Chemistry","level":0,"score":0.5660817623138428},{"id":"https://openalex.org/C2780072125","wikidata":"https://www.wikidata.org/wiki/Q28350","display_name":"Lipoprotein","level":3,"score":0.5181209444999695},{"id":"https://openalex.org/C2776448209","wikidata":"https://www.wikidata.org/wiki/Q415555","display_name":"Cholesteryl ester","level":4,"score":0.5158704519271851},{"id":"https://openalex.org/C98274493","wikidata":"https://www.wikidata.org/wiki/Q128406","display_name":"Pharmacology","level":1,"score":0.4566967785358429},{"id":"https://openalex.org/C2778163477","wikidata":"https://www.wikidata.org/wiki/Q43656","display_name":"Cholesterol","level":2,"score":0.45549070835113525},{"id":"https://openalex.org/C110459506","wikidata":"https://www.wikidata.org/wiki/Q7318217","display_name":"Reverse cholesterol transport","level":4,"score":0.44312289357185364},{"id":"https://openalex.org/C134018914","wikidata":"https://www.wikidata.org/wiki/Q162606","display_name":"Endocrinology","level":1,"score":0.41640007495880127},{"id":"https://openalex.org/C126322002","wikidata":"https://www.wikidata.org/wiki/Q11180","display_name":"Internal medicine","level":1,"score":0.4129423201084137},{"id":"https://openalex.org/C71924100","wikidata":"https://www.wikidata.org/wiki/Q11190","display_name":"Medicine","level":0,"score":0.2987062931060791},{"id":"https://openalex.org/C55493867","wikidata":"https://www.wikidata.org/wiki/Q7094","display_name":"Biochemistry","level":1,"score":0.2764604091644287}],"mesh":[{"descriptor_ui":"D000818","descriptor_name":"Animals","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D002318","descriptor_name":"Cardiovascular Diseases","qualifier_ui":"Q000097","qualifier_name":"blood","is_major_topic":false},{"descriptor_ui":"D002318","descriptor_name":"Cardiovascular Diseases","qualifier_ui":"Q000188","qualifier_name":"drug therapy","is_major_topic":false},{"descriptor_ui":"D002318","descriptor_name":"Cardiovascular Diseases","qualifier_ui":"Q000378","qualifier_name":"metabolism","is_major_topic":false},{"descriptor_ui":"D002318","descriptor_name":"Cardiovascular Diseases","qualifier_ui":"Q000517","qualifier_name":"prevention & control","is_major_topic":true},{"descriptor_ui":"D006801","descriptor_name":"Humans","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D012306","descriptor_name":"Risk","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D053480","descriptor_name":"Cholesterol Ester Transfer Proteins","qualifier_ui":"Q000037","qualifier_name":"antagonists & inhibitors","is_major_topic":true},{"descriptor_ui":"D054852","descriptor_name":"Small Molecule Libraries","qualifier_ui":"Q000494","qualifier_name":"pharmacology","is_major_topic":false},{"descriptor_ui":"D054852","descriptor_name":"Small Molecule Libraries","qualifier_ui":"Q000627","qualifier_name":"therapeutic use","is_major_topic":false},{"descriptor_ui":"D058990","descriptor_name":"Molecular Targeted Therapy","qualifier_ui":"Q000379","qualifier_name":"methods","is_major_topic":true}],"locations_count":6,"locations":[{"id":"doi:10.1194/jlr.r024075","doi":"https://doi.org/10.1194/jlr.r024075","is_oa":true,"landing_page_url":"https://doi.org/10.1194/jlr.r024075","pdf_url":"http://www.jlr.org/content/53/9/1755.full.pdf","source":{"id":"https://openalex.org/S11400418","display_name":"Journal of Lipid Research","issn_l":"0022-2275","issn":["0022-2275","1539-7262"],"is_oa":false,"is_in_doaj":true,"is_core":true,"listed_in":["cwts-core","doaj","dongbi-c","doyens","jufo-1","ki-jl-1","medline","norway-1","oarl","poland-140","vabb-shw"],"host_organization":"https://openalex.org/P4310320990","host_organization_name":"Elsevier BV","host_organization_lineage":["https://openalex.org/P4310320990"],"host_organization_lineage_names":["Elsevier BV"],"type":"journal"},"license":"cc-by","license_id":"https://openalex.org/licenses/cc-by","version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"Journal of Lipid Research","raw_type":"journal-article"},{"id":"pmh:oai:europepmc.org:2749774","doi":null,"is_oa":true,"landing_page_url":"https://www.ncbi.nlm.nih.gov/pmc/articles/3413218","pdf_url":null,"source":{"id":"https://openalex.org/S4306400806","display_name":"Europe PMC (PubMed Central)","issn_l":null,"issn":null,"is_oa":false,"is_in_doaj":false,"is_core":false,"listed_in":[],"host_organization":"https://openalex.org/I1303153112","host_organization_name":"European Bioinformatics Institute","host_organization_lineage":["https://openalex.org/I1303153112"],"host_organization_lineage_names":[],"type":"repository"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":null,"raw_type":"Text"},{"id":"pmid:22550134","doi":null,"is_oa":false,"landing_page_url":"https://pubmed.ncbi.nlm.nih.gov/22550134","pdf_url":null,"source":{"id":"https://openalex.org/S4306525036","display_name":"PubMed","issn_l":null,"issn":null,"is_oa":false,"is_in_doaj":false,"is_core":false,"listed_in":[],"host_organization":"https://openalex.org/I1299303238","host_organization_name":"National Institutes of Health","host_organization_lineage":["https://openalex.org/I1299303238"],"host_organization_lineage_names":[],"type":"repository"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"Journal of lipid research","raw_type":"Journal Article"},{"id":"pmh:oai:pubmedcentral.nih.gov:3413218","doi":null,"is_oa":true,"landing_page_url":"https://pmc.ncbi.nlm.nih.gov/articles/PMC3413218/","pdf_url":null,"source":{"id":"https://openalex.org/S2764455111","display_name":"PubMed Central","issn_l":null,"issn":null,"is_oa":true,"is_in_doaj":false,"is_core":false,"listed_in":[],"host_organization":"https://openalex.org/I1299303238","host_organization_name":"National Institutes of Health","host_organization_lineage":["https://openalex.org/I1299303238"],"host_organization_lineage_names":[],"type":"repository"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"J Lipid Res","raw_type":"Text"},{"id":"pmh:oai:doaj.org/article:6c1af9c4fbd9418ca556bf0f982d1fd1","doi":null,"is_oa":true,"landing_page_url":"https://doaj.org/article/6c1af9c4fbd9418ca556bf0f982d1fd1","pdf_url":null,"source":{"id":"https://openalex.org/S4306401280","display_name":"DOAJ (DOAJ: Directory of Open Access Journals)","issn_l":null,"issn":null,"is_oa":false,"is_in_doaj":false,"is_core":false,"listed_in":[],"host_organization":null,"host_organization_name":null,"host_organization_lineage":[],"host_organization_lineage_names":[],"type":"repository"},"license":"cc-by-sa","license_id":"https://openalex.org/licenses/cc-by-sa","version":"submittedVersion","is_accepted":false,"is_published":false,"raw_source_name":"Journal of Lipid Research, Vol 53, Iss 9, Pp 1755-1766 (2012)","raw_type":"article"},{"id":"mag:2187412430","doi":null,"is_oa":false,"landing_page_url":"http://www.jlr.org/content/53/9/1755.full.pdf","pdf_url":null,"source":null,"license":null,"license_id":null,"version":null,"is_accepted":false,"is_published":false,"raw_source_name":null,"raw_type":null}],"best_oa_location":{"id":"doi:10.1194/jlr.r024075","doi":"https://doi.org/10.1194/jlr.r024075","is_oa":true,"landing_page_url":"https://doi.org/10.1194/jlr.r024075","pdf_url":"http://www.jlr.org/content/53/9/1755.full.pdf","source":{"id":"https://openalex.org/S11400418","display_name":"Journal of Lipid Research","issn_l":"0022-2275","issn":["0022-2275","1539-7262"],"is_oa":false,"is_in_doaj":true,"is_core":true,"listed_in":["cwts-core","doaj","dongbi-c","doyens","jufo-1","ki-jl-1","medline","norway-1","oarl","poland-140","vabb-shw"],"host_organization":"https://openalex.org/P4310320990","host_organization_name":"Elsevier BV","host_organization_lineage":["https://openalex.org/P4310320990"],"host_organization_lineage_names":["Elsevier BV"],"type":"journal"},"license":"cc-by","license_id":"https://openalex.org/licenses/cc-by","version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"Journal of Lipid Research","raw_type":"journal-article"},"sustainable_development_goals":[{"score":1.0,"display_name":"Good health and well-being","id":"https://metadata.un.org/sdg/3"}],"study_designs":[],"awards":[],"funders":[],"has_content":{"pdf":true,"grobid_xml":true},"content_urls":{"pdf":"https://content.openalex.org/works/W2009220054.pdf","grobid_xml":"https://content.openalex.org/works/W2009220054.grobid-xml"},"referenced_works_count":90,"referenced_works":["https://openalex.org/W48117387","https://openalex.org/W1240353884","https://openalex.org/W1487086438","https://openalex.org/W1501497997","https://openalex.org/W1559740306","https://openalex.org/W1606186836","https://openalex.org/W1877509451","https://openalex.org/W1966124841","https://openalex.org/W1967600226","https://openalex.org/W1967702791","https://openalex.org/W1967999737","https://openalex.org/W1972597429","https://openalex.org/W1973355122","https://openalex.org/W1973740761","https://openalex.org/W1977321522","https://openalex.org/W1983012279","https://openalex.org/W1984236807","https://openalex.org/W1984820374","https://openalex.org/W1988448764","https://openalex.org/W1990231896","https://openalex.org/W1991272474","https://openalex.org/W1996069880","https://openalex.org/W1998091483","https://openalex.org/W1998187767","https://openalex.org/W1999352468","https://openalex.org/W1999461242","https://openalex.org/W2003671495","https://openalex.org/W2003803208","https://openalex.org/W2004359169","https://openalex.org/W2005795571","https://openalex.org/W2014137262","https://openalex.org/W2014558113","https://openalex.org/W2017062359","https://openalex.org/W2020028771","https://openalex.org/W2033590944","https://openalex.org/W2035973872","https://openalex.org/W2044105509","https://openalex.org/W2048481833","https://openalex.org/W2048760408","https://openalex.org/W2059048963","https://openalex.org/W2063992255","https://openalex.org/W2064861744","https://openalex.org/W2079633354","https://openalex.org/W2083791620","https://openalex.org/W2090464684","https://openalex.org/W2092176760","https://openalex.org/W2095507444","https://openalex.org/W2100791808","https://openalex.org/W2101092993","https://openalex.org/W2101396854","https://openalex.org/W2101975847","https://openalex.org/W2104650041","https://openalex.org/W2106624199","https://openalex.org/W2106839593","https://openalex.org/W2110549854","https://openalex.org/W2117416880","https://openalex.org/W2118624524","https://openalex.org/W2120751168","https://openalex.org/W2120808705","https://openalex.org/W2124484649","https://openalex.org/W2126666720","https://openalex.org/W2127427274","https://openalex.org/W2131646844","https://openalex.org/W2132328792","https://openalex.org/W2134651226","https://openalex.org/W2134811220","https://openalex.org/W2135459459","https://openalex.org/W2139567444","https://openalex.org/W2140402044","https://openalex.org/W2141210634","https://openalex.org/W2141782781","https://openalex.org/W2142131197","https://openalex.org/W2145813488","https://openalex.org/W2147426030","https://openalex.org/W2151833491","https://openalex.org/W2152683287","https://openalex.org/W2155937325","https://openalex.org/W2157149097","https://openalex.org/W2158057499","https://openalex.org/W2159243445","https://openalex.org/W2160060571","https://openalex.org/W2164089346","https://openalex.org/W2164934684","https://openalex.org/W2166606079","https://openalex.org/W2166941513","https://openalex.org/W2185518424","https://openalex.org/W2186697990","https://openalex.org/W2187198350","https://openalex.org/W2312767599","https://openalex.org/W2334373370"],"related_works":["https://openalex.org/W2187412430","https://openalex.org/W1985322784","https://openalex.org/W2003803208","https://openalex.org/W2002932070","https://openalex.org/W2402655812","https://openalex.org/W1973014196","https://openalex.org/W2072786975","https://openalex.org/W2127608622","https://openalex.org/W1981220884","https://openalex.org/W2002194333"],"abstract_inverted_index":{"Human":[0],"and":[1,37,87,93,144,190,202],"rabbit":[2],"plasma":[3,26],"contain":[4],"a":[5,97,128],"cholesteryl":[6,17],"ester":[7],"transfer":[8],"protein":[9],"(CETP)":[10],"that":[11,162,167,174,195,203],"promotes":[12],"net":[13],"mass":[14],"transfers":[15],"of":[16,32,42,59,67,72,91,124,156,211],"esters":[18],"from":[19],"high":[20],"density":[21],"lipoproteins":[22],"(HDL)":[23],"to":[24,116,122],"other":[25],"lipoprotein":[27,149],"fractions.":[28,57],"As":[29],"predicted,":[30],"inhibition":[31,123],"CETP":[33,60,74,133,175,193],"in":[34,44,53,61,77,83,96,166,180,186],"both":[35],"humans":[36,78,181],"rabbits":[38,62],"increases":[39],"the":[40,45,65,73,106,131,172,207],"concentration":[41],"cholesterol":[43],"potentially":[46,54,118],"protective":[47],"HDL":[48,138],"fraction,":[49],"while":[50],"decreasing":[51],"it":[52],"proatherogenic":[55],"non-HDL":[56,148],"Inhibition":[58],"also":[63],"inhibits":[64],"development":[66],"diet-induced":[68],"atherosclerosis.":[69],"However,":[70],"use":[71],"inhibitor":[75,134],"torcetrapib":[76,110,143],"did":[79],"not":[80,146,205],"reduce":[81],"atheroma":[82],"three":[84],"imaging":[85],"trials":[86],"caused":[88,108,164],"an":[89],"excess":[90],"deaths":[92],"cardiovascular":[94],"events":[95],"large":[98],"clinical":[99],"outcome":[100],"trial.":[101,168],"The":[102],"precise":[103],"explanation":[104],"for":[105,154],"harm":[107,165],"by":[109],"is":[111,182],"unknown":[112],"but":[113],"may":[114],"relate":[115],"documented,":[117],"harmful":[119],"effects":[120,210],"unrelated":[121],"CETP.":[125],"More":[126],"recently,":[127],"trial":[129],"using":[130],"weak":[132],"dalcetrapib,":[135],"which":[136],"raises":[137],"levels":[139],"less":[140],"effectively":[141],"than":[142,200],"does":[145],"lower":[147],"levels,":[150],"was":[151,159],"terminated":[152],"early":[153],"reasons":[155],"futility.":[157],"There":[158],"no":[160],"evidence":[161],"dalcetrapib":[163,201],"Despite":[169],"these":[170],"setbacks,":[171],"hypothesis":[173],"inhibitors":[176,194],"will":[177],"be":[178],"antiatherogenic":[179],"still":[183],"being":[184],"tested":[185],"studies":[187],"with":[188],"anacetrapib":[189],"evacetrapib,":[191],"two":[192],"are":[196],"much":[197],"more":[198],"potent":[199],"do":[204],"share":[206],"off-target":[208],"adverse":[209],"torcetrapib.":[212]},"counts_by_year":[{"year":2026,"cited_by_count":3},{"year":2025,"cited_by_count":4},{"year":2024,"cited_by_count":5},{"year":2023,"cited_by_count":2},{"year":2022,"cited_by_count":4},{"year":2021,"cited_by_count":4},{"year":2020,"cited_by_count":3},{"year":2019,"cited_by_count":10},{"year":2018,"cited_by_count":10},{"year":2017,"cited_by_count":12},{"year":2016,"cited_by_count":15},{"year":2015,"cited_by_count":18},{"year":2014,"cited_by_count":23},{"year":2013,"cited_by_count":29},{"year":2012,"cited_by_count":6}],"updated_date":"2026-11-10T11:39:43.021295","created_date":"2016-06-24T00:00:00"}
