{"id":"https://openalex.org/W1995243183","doi":"https://doi.org/10.3109/10717544.2013.870260","title":"Formulation by design-based proniosome for accentuated transdermal delivery of risperidone: in vitro characterization and in vivo pharmacokinetic study","display_name":"Formulation by design-based proniosome for accentuated transdermal delivery of risperidone: in vitro characterization and in vivo pharmacokinetic study","publication_year":2014,"publication_date":"2014-01-29","ids":{"openalex":"https://openalex.org/W1995243183","doi":"https://doi.org/10.3109/10717544.2013.870260","mag":"1995243183","pmid":"https://pubmed.ncbi.nlm.nih.gov/24471715"},"language":"en","primary_location":{"id":"doi:10.3109/10717544.2013.870260","doi":"https://doi.org/10.3109/10717544.2013.870260","is_oa":true,"landing_page_url":"https://doi.org/10.3109/10717544.2013.870260","pdf_url":"https://www.tandfonline.com/doi/pdf/10.3109/10717544.2013.870260?needAccess=true&role=button","source":{"id":"https://openalex.org/S70174254","display_name":"Drug Delivery","issn_l":"1071-7544","issn":["1071-7544","1521-0464"],"is_oa":false,"is_in_doaj":true,"is_core":true,"listed_in":["anvur-scientific","cwts-core","doaj","dongbi-b","doyens","jufo-1","medline","oarl","poland-100","russia-white-list-1","vabb-shw"],"host_organization":"https://openalex.org/P4310320547","host_organization_name":"Taylor & Francis","host_organization_lineage":["https://openalex.org/P4310320547","https://openalex.org/P4310320449"],"host_organization_lineage_names":["Taylor & Francis","Informa"],"type":"journal"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"Drug Delivery","raw_type":"journal-article"},"volume":null,"type":"article","is_traditional":true,"indexed_in":["crossref","doaj","pubmed"],"open_access":{"is_oa":true,"oa_status":"bronze","oa_url":"https://www.tandfonline.com/doi/pdf/10.3109/10717544.2013.870260?needAccess=true&role=button","any_repository_has_fulltext":false},"authorships":[{"author_position":"first","author":{"id":"https://openalex.org/A5003677451","display_name":"Syed Sarim Imam","orcid":"https://orcid.org/0000-0002-8913-0826","observed_orcids":["https://orcid.org/0000-0002-8913-0826"]},"institutions":[],"countries":[],"is_corresponding":false,"raw_author_name":"Syed Sarim Imam","raw_affiliation_strings":["a Department of Pharmaceutics and"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"a Department of Pharmaceutics and","institution_ids":[]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5089261501","display_name":"Mohd. Aqil","orcid":"https://orcid.org/0000-0001-6797-3104","observed_orcids":["https://orcid.org/0000-0001-6797-3104"]},"institutions":[],"countries":[],"is_corresponding":true,"raw_author_name":"Mohammed Aqil","raw_affiliation_strings":["a Department of Pharmaceutics and","Department of Pharmaceutics and"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"a Department of Pharmaceutics and","institution_ids":[]},{"raw_affiliation_string":"Department of Pharmaceutics and","institution_ids":[]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5086044687","display_name":"Mohammed Akhtar","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I19716509","display_name":"Jamia Hamdard","ror":"https://ror.org/03dwxvb85","country_code":"IN","type":"education","lineage":["https://openalex.org/I19716509"]}],"countries":["IN"],"is_corresponding":false,"raw_author_name":"Mohammed Akhtar","raw_affiliation_strings":["b Department of Pharmacology , Faculty of Pharmacy, Jamia Hamdard , New Delhi , India"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"b Department of Pharmacology , Faculty of Pharmacy, Jamia Hamdard , New Delhi , India","institution_ids":["https://openalex.org/I19716509"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5064337706","display_name":"Yasmin Sultana","orcid":"https://orcid.org/0000-0002-3979-6574","observed_orcids":["https://orcid.org/0000-0002-3979-6574"]},"institutions":[],"countries":[],"is_corresponding":false,"raw_author_name":"Yasmin Sultana","raw_affiliation_strings":["a Department of Pharmaceutics and","Department of Pharmaceutics and"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"a Department of Pharmaceutics and","institution_ids":[]},{"raw_affiliation_string":"Department of Pharmaceutics and","institution_ids":[]}]},{"author_position":"last","author":{"id":"https://openalex.org/A5102963709","display_name":"Asgar Ali","orcid":"https://orcid.org/0000-0002-9603-3995","observed_orcids":["https://orcid.org/0000-0002-9603-3995"]},"institutions":[],"countries":[],"is_corresponding":false,"raw_author_name":"Asgar Ali","raw_affiliation_strings":["a Department of Pharmaceutics and","Department of Pharmaceutics and"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"a Department of Pharmaceutics and","institution_ids":[]},{"raw_affiliation_string":"Department of Pharmaceutics and","institution_ids":[]}]}],"institutions":[],"countries_distinct_count":1,"institutions_distinct_count":1,"corresponding_author_ids":["https://openalex.org/A5089261501"],"corresponding_institution_ids":[],"apc_list":{"value":2335,"currency":"GBP","value_usd":2864},"apc_paid":null,"fwci":3.6127,"has_fulltext":true,"cited_by_count":100,"citation_normalized_percentile":{"value":0.92350841,"is_in_top_1_percent":false,"is_in_top_10_percent":true},"cited_by_percentile_year":{"min":93,"max":100},"biblio":{"volume":"22","issue":"8","first_page":"1059","last_page":"1070"},"is_retracted":false,"is_paratext":false,"is_xpac":false,"primary_topic":{"id":"https://openalex.org/T10704","display_name":"Advancements in Transdermal Drug Delivery","score":1.0,"subfield":{"id":"https://openalex.org/subfields/3003","display_name":"Pharmaceutical Science"},"field":{"id":"https://openalex.org/fields/30","display_name":"Pharmacology, Toxicology and Pharmaceutics"},"domain":{"id":"https://openalex.org/domains/1","display_name":"Life Sciences"}},"topics":[{"id":"https://openalex.org/T10704","display_name":"Advancements in Transdermal Drug Delivery","score":1.0,"subfield":{"id":"https://openalex.org/subfields/3003","display_name":"Pharmaceutical Science"},"field":{"id":"https://openalex.org/fields/30","display_name":"Pharmacology, Toxicology and Pharmaceutics"},"domain":{"id":"https://openalex.org/domains/1","display_name":"Life Sciences"}},{"id":"https://openalex.org/T10920","display_name":"Advanced Drug Delivery Systems","score":9.999999747378752e-05,"subfield":{"id":"https://openalex.org/subfields/3003","display_name":"Pharmaceutical Science"},"field":{"id":"https://openalex.org/fields/30","display_name":"Pharmacology, Toxicology and Pharmaceutics"},"domain":{"id":"https://openalex.org/domains/1","display_name":"Life Sciences"}},{"id":"https://openalex.org/T10256","display_name":"Drug Solubulity and Delivery Systems","score":0.0,"subfield":{"id":"https://openalex.org/subfields/3003","display_name":"Pharmaceutical Science"},"field":{"id":"https://openalex.org/fields/30","display_name":"Pharmacology, Toxicology and Pharmaceutics"},"domain":{"id":"https://openalex.org/domains/1","display_name":"Life Sciences"}}],"keywords":[{"id":"https://openalex.org/keywords/risperidone","display_name":"risperidone","score":0.8669999837875366},{"id":"https://openalex.org/keywords/proniosomes","display_name":"proniosomes","score":0.9490000009536743},{"id":"https://openalex.org/keywords/transdermal-drug-delivery","display_name":"transdermal drug delivery","score":0.9449999928474426},{"id":"https://openalex.org/keywords/transdermal-therapeutic-systems","display_name":"transdermal therapeutic systems","score":0.906000018119812},{"id":"https://openalex.org/keywords/factorial-design","display_name":"factorial design","score":0.6629999876022339},{"id":"https://openalex.org/keywords/vesicle-size","display_name":"vesicle size","score":0.9129999876022339},{"id":"https://openalex.org/keywords/encapsulation-efficiency","display_name":"encapsulation efficiency","score":0.9990000128746033},{"id":"https://openalex.org/keywords/skin-permeation","display_name":"skin permeation","score":0.9509999752044678},{"id":"https://openalex.org/keywords/bioavailability","display_name":"bioavailability","score":0.6060000061988831},{"id":"https://openalex.org/keywords/cholesterol","display_name":"cholesterol","score":0.37599998712539673},{"id":"https://openalex.org/keywords/span-60","display_name":"Span 60","score":0.8989999890327454},{"id":"https://openalex.org/keywords/antipsychotic-drug-delivery","display_name":"antipsychotic drug delivery","score":0.7179999947547913},{"id":"https://openalex.org/keywords/schizophrenia","display_name":"schizophrenia","score":0.9449999928474426}],"concepts":[{"id":"https://openalex.org/C205679159","wikidata":"https://www.wikidata.org/wiki/Q3375179","display_name":"Transdermal","level":2,"score":0.8840773701667786},{"id":"https://openalex.org/C98274493","wikidata":"https://www.wikidata.org/wiki/Q128406","display_name":"Pharmacology","level":1,"score":0.6307373046875},{"id":"https://openalex.org/C181389837","wikidata":"https://www.wikidata.org/wiki/Q461809","display_name":"Bioavailability","level":2,"score":0.6244028806686401},{"id":"https://openalex.org/C2780057945","wikidata":"https://www.wikidata.org/wiki/Q412443","display_name":"Risperidone","level":3,"score":0.6078757047653198},{"id":"https://openalex.org/C185154212","wikidata":"https://www.wikidata.org/wiki/Q410454","display_name":"Liposome","level":2,"score":0.585869312286377},{"id":"https://openalex.org/C72918618","wikidata":"https://www.wikidata.org/wiki/Q1993211","display_name":"Niosome","level":4,"score":0.5847170352935791},{"id":"https://openalex.org/C22979827","wikidata":"https://www.wikidata.org/wiki/Q5137311","display_name":"Cmax","level":3,"score":0.5793404579162598},{"id":"https://openalex.org/C169222746","wikidata":"https://www.wikidata.org/wiki/Q4116558","display_name":"Factorial experiment","level":2,"score":0.5242947936058044},{"id":"https://openalex.org/C112705442","wikidata":"https://www.wikidata.org/wiki/Q323936","display_name":"Pharmacokinetics","level":2,"score":0.4684220552444458},{"id":"https://openalex.org/C207001950","wikidata":"https://www.wikidata.org/wiki/Q141124","display_name":"In vivo","level":2,"score":0.4501788020133972},{"id":"https://openalex.org/C192562407","wikidata":"https://www.wikidata.org/wiki/Q228736","display_name":"Materials science","level":0,"score":0.42195558547973633},{"id":"https://openalex.org/C43617362","wikidata":"https://www.wikidata.org/wiki/Q170050","display_name":"Chromatography","level":1,"score":0.3511437475681305},{"id":"https://openalex.org/C71924100","wikidata":"https://www.wikidata.org/wiki/Q11190","display_name":"Medicine","level":0,"score":0.34035906195640564},{"id":"https://openalex.org/C136229726","wikidata":"https://www.wikidata.org/wiki/Q327092","display_name":"Biomedical engineering","level":1,"score":0.32963889837265015},{"id":"https://openalex.org/C185592680","wikidata":"https://www.wikidata.org/wiki/Q2329","display_name":"Chemistry","level":0,"score":0.2856197953224182},{"id":"https://openalex.org/C130316041","wikidata":"https://www.wikidata.org/wiki/Q189206","display_name":"Vesicle","level":3,"score":0.2166980803012848},{"id":"https://openalex.org/C33923547","wikidata":"https://www.wikidata.org/wiki/Q395","display_name":"Mathematics","level":0,"score":0.2147742211818695},{"id":"https://openalex.org/C171250308","wikidata":"https://www.wikidata.org/wiki/Q11468","display_name":"Nanotechnology","level":1,"score":0.21410447359085083},{"id":"https://openalex.org/C41625074","wikidata":"https://www.wikidata.org/wiki/Q176088","display_name":"Membrane","level":2,"score":0.15185722708702087},{"id":"https://openalex.org/C150903083","wikidata":"https://www.wikidata.org/wiki/Q7108","display_name":"Biotechnology","level":1,"score":0.0677376389503479},{"id":"https://openalex.org/C55493867","wikidata":"https://www.wikidata.org/wiki/Q7094","display_name":"Biochemistry","level":1,"score":0.06723812222480774},{"id":"https://openalex.org/C2776412080","wikidata":"https://www.wikidata.org/wiki/Q7431605","display_name":"Schizophrenia (object-oriented programming)","level":2,"score":0.0},{"id":"https://openalex.org/C86803240","wikidata":"https://www.wikidata.org/wiki/Q420","display_name":"Biology","level":0,"score":0.0},{"id":"https://openalex.org/C105795698","wikidata":"https://www.wikidata.org/wiki/Q12483","display_name":"Statistics","level":1,"score":0.0},{"id":"https://openalex.org/C118552586","wikidata":"https://www.wikidata.org/wiki/Q7867","display_name":"Psychiatry","level":1,"score":0.0}],"mesh":[],"locations_count":2,"locations":[{"id":"doi:10.3109/10717544.2013.870260","doi":"https://doi.org/10.3109/10717544.2013.870260","is_oa":true,"landing_page_url":"https://doi.org/10.3109/10717544.2013.870260","pdf_url":"https://www.tandfonline.com/doi/pdf/10.3109/10717544.2013.870260?needAccess=true&role=button","source":{"id":"https://openalex.org/S70174254","display_name":"Drug Delivery","issn_l":"1071-7544","issn":["1071-7544","1521-0464"],"is_oa":false,"is_in_doaj":true,"is_core":true,"listed_in":["anvur-scientific","cwts-core","doaj","dongbi-b","doyens","jufo-1","medline","oarl","poland-100","russia-white-list-1","vabb-shw"],"host_organization":"https://openalex.org/P4310320547","host_organization_name":"Taylor & Francis","host_organization_lineage":["https://openalex.org/P4310320547","https://openalex.org/P4310320449"],"host_organization_lineage_names":["Taylor & Francis","Informa"],"type":"journal"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"Drug Delivery","raw_type":"journal-article"},{"id":"pmid:24471715","doi":null,"is_oa":false,"landing_page_url":"https://pubmed.ncbi.nlm.nih.gov/24471715","pdf_url":null,"source":{"id":"https://openalex.org/S4306525036","display_name":"PubMed","issn_l":null,"issn":null,"is_oa":false,"is_in_doaj":false,"is_core":false,"listed_in":[],"host_organization":"https://openalex.org/I1299303238","host_organization_name":"National Institutes of Health","host_organization_lineage":["https://openalex.org/I1299303238"],"host_organization_lineage_names":[],"type":"repository"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"Drug delivery","raw_type":"Journal Article"}],"best_oa_location":{"id":"doi:10.3109/10717544.2013.870260","doi":"https://doi.org/10.3109/10717544.2013.870260","is_oa":true,"landing_page_url":"https://doi.org/10.3109/10717544.2013.870260","pdf_url":"https://www.tandfonline.com/doi/pdf/10.3109/10717544.2013.870260?needAccess=true&role=button","source":{"id":"https://openalex.org/S70174254","display_name":"Drug Delivery","issn_l":"1071-7544","issn":["1071-7544","1521-0464"],"is_oa":false,"is_in_doaj":true,"is_core":true,"listed_in":["anvur-scientific","cwts-core","doaj","dongbi-b","doyens","jufo-1","medline","oarl","poland-100","russia-white-list-1","vabb-shw"],"host_organization":"https://openalex.org/P4310320547","host_organization_name":"Taylor & Francis","host_organization_lineage":["https://openalex.org/P4310320547","https://openalex.org/P4310320449"],"host_organization_lineage_names":["Taylor & Francis","Informa"],"type":"journal"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"Drug Delivery","raw_type":"journal-article"},"sustainable_development_goals":[{"display_name":"Good health and well-being","score":0.9391000270843506,"id":"https://metadata.un.org/sdg/3"}],"study_designs":[],"awards":[],"funders":[{"id":"https://openalex.org/F4320320720","display_name":"Indian Council of Medical Research","ror":"https://ror.org/0492wrx28"},{"id":"https://openalex.org/F4320324337","display_name":"All-India Institute of Medical Sciences","ror":"https://ror.org/02dwcqs71"}],"has_content":{"grobid_xml":true,"pdf":true},"content_urls":{"pdf":"https://content.openalex.org/works/W1995243183.pdf","grobid_xml":"https://content.openalex.org/works/W1995243183.grobid-xml"},"referenced_works_count":35,"referenced_works":["https://openalex.org/W8008152","https://openalex.org/W1968601352","https://openalex.org/W1971897151","https://openalex.org/W1972723441","https://openalex.org/W1974637913","https://openalex.org/W1976561097","https://openalex.org/W1979209041","https://openalex.org/W1988144726","https://openalex.org/W1990098432","https://openalex.org/W1992288425","https://openalex.org/W1993061546","https://openalex.org/W1993115176","https://openalex.org/W1994381824","https://openalex.org/W1997325051","https://openalex.org/W2003587134","https://openalex.org/W2033381869","https://openalex.org/W2033547005","https://openalex.org/W2038727769","https://openalex.org/W2039551585","https://openalex.org/W2043512639","https://openalex.org/W2053825412","https://openalex.org/W2058009653","https://openalex.org/W2064144933","https://openalex.org/W2066432116","https://openalex.org/W2075706054","https://openalex.org/W2079966725","https://openalex.org/W2084774646","https://openalex.org/W2085205359","https://openalex.org/W2085692671","https://openalex.org/W2090692853","https://openalex.org/W2093918270","https://openalex.org/W2104205848","https://openalex.org/W2154067623","https://openalex.org/W2161530911","https://openalex.org/W2311902495"],"related_works":["https://openalex.org/W2759503433","https://openalex.org/W2788122361","https://openalex.org/W2157430128","https://openalex.org/W4383619328","https://openalex.org/W2186568034","https://openalex.org/W2064144933","https://openalex.org/W2133566692","https://openalex.org/W2593626546","https://openalex.org/W2368632791","https://openalex.org/W4401346054"],"abstract_inverted_index":{"Aim:":[0],"The":[1,69,92,134],"aim":[2],"of":[3,11,17,40,65,86,101,111,123,150],"this":[4],"work":[5],"was":[6,32,105,125],"to":[7,34,81],"investigate":[8],"the":[9,15],"effects":[10,39],"formulation":[12,41,73],"variables":[13,42],"on":[14,55],"development":[16],"risperidone":[18,52,141],"proniosomal":[19,72],"formulations":[20],"as":[21],"potential":[22],"transdermal":[23,137],"delivery":[24],"systems.Materials":[25],"and":[26,37,51,62,67],"methods:":[27],"A":[28],"43":[29],"factorial":[30],"design":[31],"employed":[33],"evaluate":[35],"individual":[36],"combined":[38],"cholesterol":[43],"(X1),":[44],"span":[45],"60":[46],"(X2),":[47],"phospholipid":[48],"G90":[49],"(X3),":[50],"(X4)":[53],"added":[54],"vesicle":[56],"size":[57],"(Y1),":[58],"encapsulation":[59],"efficiency":[60],"(Y2),":[61],"flux":[63],"(Y3)":[64],"proniosomes.Results":[66],"discussion:":[68],"investigated":[70],"risperidone-loaded":[71],"shows":[74],"significantly":[75,126],"higher":[76,108],"skin":[77],"permeation":[78],"in":[79,95],"comparison":[80],"conventional":[82],"liposomes":[83],"with":[84],"ER":[85],"4.4":[87],"times":[88,107],"through":[89],"rat":[90],"skin.":[91],"bioavailability":[93],"studies":[94],"rats":[96],"indicated":[97],"that":[98,110,120],"mean":[99],"value":[100,122],"AUC0\u201348":[102],"by":[103],"ROPF-TTS":[104,124],"1.31":[106],"than":[109],"oral":[112],"dosage":[113],"form.":[114],"So":[115],"it":[116],"could":[117],"be":[118],"concluded":[119],"Cmax":[121],"reduced":[127],"while":[128],"AUC":[129],"values":[130],"were":[131],"apparently":[132],"increased.Conclusion:":[133],"developed":[135],"proniosomal-based":[136],"therapeutic":[138],"systems":[139],"incorporating":[140],"would":[142],"provide":[143],"a":[144],"useful":[145],"strategy":[146],"for":[147],"better":[148],"management":[149],"schizophrenia.":[151]},"counts_by_year":[{"year":2026,"cited_by_count":6},{"year":2025,"cited_by_count":4},{"year":2024,"cited_by_count":7},{"year":2023,"cited_by_count":5},{"year":2022,"cited_by_count":16},{"year":2021,"cited_by_count":12},{"year":2020,"cited_by_count":18},{"year":2019,"cited_by_count":8},{"year":2018,"cited_by_count":6},{"year":2017,"cited_by_count":8},{"year":2016,"cited_by_count":3},{"year":2015,"cited_by_count":2},{"year":2014,"cited_by_count":4}],"updated_date":"2026-11-07T11:25:07.637180","created_date":"2016-06-24T00:00:00"}
