{"id":"https://openalex.org/W128284052","doi":"https://doi.org/10.2174/1386207054867328","title":"The Novartis Compound Archive - From Concept to Reality","display_name":"The Novartis Compound Archive - From Concept to Reality","publication_year":2005,"publication_date":"2005-08-30","ids":{"openalex":"https://openalex.org/W128284052","doi":"https://doi.org/10.2174/1386207054867328","mag":"128284052","pmid":"https://pubmed.ncbi.nlm.nih.gov/16178810"},"language":"en","primary_location":{"id":"doi:10.2174/1386207054867328","doi":"https://doi.org/10.2174/1386207054867328","is_oa":false,"landing_page_url":"https://doi.org/10.2174/1386207054867328","pdf_url":null,"source":{"id":"https://openalex.org/S50933791","display_name":"Combinatorial Chemistry & High Throughput Screening","issn_l":"1386-2073","issn":["1386-2073","1875-5402"],"is_oa":false,"is_in_doaj":false,"is_core":true,"listed_in":["cwts-core","dongbi-d","jufo-1","ki-jl-1","medline","norway-1","poland-40","russia-white-list-3"],"host_organization":"https://openalex.org/P4310320079","host_organization_name":"Bentham Science Publishers","host_organization_lineage":["https://openalex.org/P4310320079"],"host_organization_lineage_names":["Bentham Science Publishers"],"type":"journal"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"Combinatorial Chemistry &amp; High Throughput Screening","raw_type":"journal-article"},"volume":null,"type":"article","is_traditional":true,"indexed_in":["crossref","pubmed"],"open_access":{"is_oa":false,"oa_status":"closed","oa_url":null,"any_repository_has_fulltext":false},"authorships":[{"author_position":"first","author":{"id":"https://openalex.org/A5022269771","display_name":"Ulrich Schopfer","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I1283582996","display_name":"Novartis (Switzerland)","ror":"https://ror.org/02f9zrr09","country_code":"CH","type":"company","lineage":["https://openalex.org/I1283582996"]},{"id":"https://openalex.org/I4400600974","display_name":"Novartis Institutes for BioMedical Research","ror":"https://ror.org/053gv2m95","country_code":"CH","type":"funder","lineage":["https://openalex.org/I1283582996","https://openalex.org/I4400600974"]}],"countries":["CH"],"is_corresponding":false,"raw_author_name":"U. Schopfer","raw_affiliation_strings":["Compound Logistics and Properties Unit/ Novartis Compound Archive, Novartis Institutes for BioMedical Research, CH-4002 Basel, Switzerland. ulrich.schopfer@novartis.com"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Compound Logistics and Properties Unit/ Novartis Compound Archive, Novartis Institutes for BioMedical Research, CH-4002 Basel, Switzerland. ulrich.schopfer@novartis.com","institution_ids":["https://openalex.org/I1283582996","https://openalex.org/I4400600974"]}]},{"author_position":"middle","author":{"id":"https://openalex.org/A5061979088","display_name":"Caroline Engeloch","orcid":null,"observed_orcids":[]},"institutions":[],"countries":[],"is_corresponding":false,"raw_author_name":"C. Engeloch","raw_affiliation_strings":[],"raw_orcid":null,"affiliations":[]},{"author_position":"middle","author":{"id":"https://openalex.org/A5085909775","display_name":"Jan J. Stanek","orcid":"https://orcid.org/0000-0001-5108-7175","observed_orcids":["https://orcid.org/0000-0001-5108-7175"]},"institutions":[],"countries":[],"is_corresponding":false,"raw_author_name":"J. Stanek","raw_affiliation_strings":[],"raw_orcid":null,"affiliations":[]},{"author_position":"middle","author":{"id":null,"display_name":"M. Girod","orcid":null,"observed_orcids":[]},"institutions":[],"countries":[],"is_corresponding":false,"raw_author_name":"M. Girod","raw_affiliation_strings":[],"raw_orcid":null,"affiliations":[]},{"author_position":"middle","author":{"id":"https://openalex.org/A5029464406","display_name":"Ansgar Schuffenhauer","orcid":"https://orcid.org/0000-0001-6385-0414","observed_orcids":["https://orcid.org/0000-0001-6385-0414"]},"institutions":[],"countries":[],"is_corresponding":false,"raw_author_name":"A. Schuffenhauer","raw_affiliation_strings":[],"raw_orcid":null,"affiliations":[]},{"author_position":"middle","author":{"id":"https://openalex.org/A5036331925","display_name":"Edgar Jacoby","orcid":"https://orcid.org/0000-0003-4312-9448","observed_orcids":["https://orcid.org/0000-0003-4312-9448"]},"institutions":[],"countries":[],"is_corresponding":false,"raw_author_name":"E. Jacoby","raw_affiliation_strings":[],"raw_orcid":null,"affiliations":[]},{"author_position":"last","author":{"id":"https://openalex.org/A5034309251","display_name":"Pierre Acklin","orcid":null,"observed_orcids":[]},"institutions":[{"id":"https://openalex.org/I1283582996","display_name":"Novartis (Switzerland)","ror":"https://ror.org/02f9zrr09","country_code":"CH","type":"company","lineage":["https://openalex.org/I1283582996"]},{"id":"https://openalex.org/I4400600974","display_name":"Novartis Institutes for BioMedical Research","ror":"https://ror.org/053gv2m95","country_code":"CH","type":"funder","lineage":["https://openalex.org/I1283582996","https://openalex.org/I4400600974"]}],"countries":["CH"],"is_corresponding":true,"raw_author_name":"P. Acklin","raw_affiliation_strings":["Novartis Compound Archive, Novartis Institutes for BioMedical Research, CH-4002 Basel, Switzerland.,Switzerland"],"raw_orcid":null,"affiliations":[{"raw_affiliation_string":"Novartis Compound Archive, Novartis Institutes for BioMedical Research, CH-4002 Basel, Switzerland.,Switzerland","institution_ids":["https://openalex.org/I1283582996","https://openalex.org/I4400600974"]}]}],"institutions":[],"countries_distinct_count":1,"institutions_distinct_count":2,"corresponding_author_ids":["https://openalex.org/A5034309251"],"corresponding_institution_ids":["https://openalex.org/I1283582996","https://openalex.org/I4400600974"],"apc_list":null,"apc_paid":null,"fwci":1.3356,"has_fulltext":false,"cited_by_count":31,"citation_normalized_percentile":{"value":0.75753486,"is_in_top_1_percent":false,"is_in_top_10_percent":false},"cited_by_percentile_year":{"min":88,"max":98},"biblio":{"volume":"8","issue":"6","first_page":"513","last_page":"519"},"is_retracted":false,"is_paratext":false,"is_xpac":false,"primary_topic":{"id":"https://openalex.org/T10211","display_name":"Computational Drug Discovery Methods","score":0.6039999723434448,"subfield":{"id":"https://openalex.org/subfields/3002","display_name":"Drug Discovery"},"field":{"id":"https://openalex.org/fields/30","display_name":"Pharmacology, Toxicology and Pharmaceutics"},"domain":{"id":"https://openalex.org/domains/1","display_name":"Life Sciences"}},"topics":[{"id":"https://openalex.org/T10211","display_name":"Computational Drug Discovery Methods","score":0.6039999723434448,"subfield":{"id":"https://openalex.org/subfields/3002","display_name":"Drug Discovery"},"field":{"id":"https://openalex.org/fields/30","display_name":"Pharmacology, Toxicology and Pharmaceutics"},"domain":{"id":"https://openalex.org/domains/1","display_name":"Life Sciences"}},{"id":"https://openalex.org/T10911","display_name":"Chemical Synthesis and Analysis","score":0.14810000360012054,"subfield":{"id":"https://openalex.org/subfields/1605","display_name":"Organic Chemistry"},"field":{"id":"https://openalex.org/fields/16","display_name":"Chemistry"},"domain":{"id":"https://openalex.org/domains/3","display_name":"Physical Sciences"}},{"id":"https://openalex.org/T11460","display_name":"Analytical Methods in Pharmaceuticals","score":0.02459999918937683,"subfield":{"id":"https://openalex.org/subfields/1602","display_name":"Analytical Chemistry"},"field":{"id":"https://openalex.org/fields/16","display_name":"Chemistry"},"domain":{"id":"https://openalex.org/domains/3","display_name":"Physical Sciences"}}],"keywords":[{"id":"https://openalex.org/keywords/compound-stability","display_name":"compound stability","score":0.6100000143051147},{"id":"https://openalex.org/keywords/freeze-thaw-cycles","display_name":"freeze-thaw cycles","score":0.7990000247955322},{"id":"https://openalex.org/keywords/water-uptake","display_name":"water absorption","score":0.9210000038146973},{"id":"https://openalex.org/keywords/automated-weighing","display_name":"automated weighing","score":0.7570000290870667},{"id":"https://openalex.org/keywords/novartis","display_name":"Novartis","score":0.8050000071525574}],"concepts":[{"id":"https://openalex.org/C155574463","wikidata":"https://www.wikidata.org/wiki/Q170731","display_name":"Solubility","level":2,"score":0.7021815180778503},{"id":"https://openalex.org/C158960510","wikidata":"https://www.wikidata.org/wiki/Q180600","display_name":"Relative humidity","level":2,"score":0.5096056461334229},{"id":"https://openalex.org/C12590798","wikidata":"https://www.wikidata.org/wiki/Q3933199","display_name":"Replication (statistics)","level":2,"score":0.4699559211730957},{"id":"https://openalex.org/C41008148","wikidata":"https://www.wikidata.org/wiki/Q21198","display_name":"Computer science","level":0,"score":0.42921650409698486},{"id":"https://openalex.org/C171250308","wikidata":"https://www.wikidata.org/wiki/Q11468","display_name":"Nanotechnology","level":1,"score":0.3722299635410309},{"id":"https://openalex.org/C185592680","wikidata":"https://www.wikidata.org/wiki/Q2329","display_name":"Chemistry","level":0,"score":0.36569491028785706},{"id":"https://openalex.org/C21880701","wikidata":"https://www.wikidata.org/wiki/Q2144042","display_name":"Process engineering","level":1,"score":0.3654922842979431},{"id":"https://openalex.org/C192562407","wikidata":"https://www.wikidata.org/wiki/Q228736","display_name":"Materials science","level":0,"score":0.3629872798919678},{"id":"https://openalex.org/C39432304","wikidata":"https://www.wikidata.org/wiki/Q188847","display_name":"Environmental science","level":0,"score":0.360181987285614},{"id":"https://openalex.org/C42360764","wikidata":"https://www.wikidata.org/wiki/Q83588","display_name":"Chemical engineering","level":1,"score":0.35934001207351685},{"id":"https://openalex.org/C21951064","wikidata":"https://www.wikidata.org/wiki/Q899212","display_name":"Combinatorial chemistry","level":1,"score":0.3333355784416199},{"id":"https://openalex.org/C178790620","wikidata":"https://www.wikidata.org/wiki/Q11351","display_name":"Organic chemistry","level":1,"score":0.2395525574684143},{"id":"https://openalex.org/C33923547","wikidata":"https://www.wikidata.org/wiki/Q395","display_name":"Mathematics","level":0,"score":0.1598992943763733},{"id":"https://openalex.org/C127413603","wikidata":"https://www.wikidata.org/wiki/Q11023","display_name":"Engineering","level":0,"score":0.11700239777565002},{"id":"https://openalex.org/C97355855","wikidata":"https://www.wikidata.org/wiki/Q11473","display_name":"Thermodynamics","level":1,"score":0.110003262758255},{"id":"https://openalex.org/C121332964","wikidata":"https://www.wikidata.org/wiki/Q413","display_name":"Physics","level":0,"score":0.10452196002006531},{"id":"https://openalex.org/C105795698","wikidata":"https://www.wikidata.org/wiki/Q12483","display_name":"Statistics","level":1,"score":0.0}],"mesh":[{"descriptor_ui":"D001331","descriptor_name":"Automation","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D004345","descriptor_name":"Drug Industry","qualifier_ui":"Q000458","qualifier_name":"organization & administration","is_major_topic":true},{"descriptor_ui":"D004355","descriptor_name":"Drug Stability","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D004356","descriptor_name":"Drug Storage","qualifier_ui":null,"qualifier_name":null,"is_major_topic":true},{"descriptor_ui":"D012371","descriptor_name":"Robotics","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D012995","descriptor_name":"Solubility","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false},{"descriptor_ui":"D012996","descriptor_name":"Solutions","qualifier_ui":null,"qualifier_name":null,"is_major_topic":false}],"locations_count":2,"locations":[{"id":"doi:10.2174/1386207054867328","doi":"https://doi.org/10.2174/1386207054867328","is_oa":false,"landing_page_url":"https://doi.org/10.2174/1386207054867328","pdf_url":null,"source":{"id":"https://openalex.org/S50933791","display_name":"Combinatorial Chemistry & High Throughput Screening","issn_l":"1386-2073","issn":["1386-2073","1875-5402"],"is_oa":false,"is_in_doaj":false,"is_core":true,"listed_in":["cwts-core","dongbi-d","jufo-1","ki-jl-1","medline","norway-1","poland-40","russia-white-list-3"],"host_organization":"https://openalex.org/P4310320079","host_organization_name":"Bentham Science Publishers","host_organization_lineage":["https://openalex.org/P4310320079"],"host_organization_lineage_names":["Bentham Science Publishers"],"type":"journal"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"Combinatorial Chemistry &amp; High Throughput Screening","raw_type":"journal-article"},{"id":"pmid:16178810","doi":null,"is_oa":false,"landing_page_url":"https://pubmed.ncbi.nlm.nih.gov/16178810","pdf_url":null,"source":{"id":"https://openalex.org/S4306525036","display_name":"PubMed","issn_l":null,"issn":null,"is_oa":false,"is_in_doaj":false,"is_core":false,"listed_in":[],"host_organization":"https://openalex.org/I1299303238","host_organization_name":"National Institutes of Health","host_organization_lineage":["https://openalex.org/I1299303238"],"host_organization_lineage_names":[],"type":"repository"},"license":null,"license_id":null,"version":"publishedVersion","is_accepted":true,"is_published":true,"raw_source_name":"Combinatorial chemistry & high throughput screening","raw_type":"Journal Article"}],"best_oa_location":null,"sustainable_development_goals":[],"study_designs":[],"awards":[],"funders":[{"id":"https://openalex.org/F4320333796","display_name":"Novartis Institutes for BioMedical Research","ror":"https://ror.org/053gv2m95"}],"has_content":{"pdf":false,"grobid_xml":false},"content_urls":null,"referenced_works_count":0,"referenced_works":[],"related_works":["https://openalex.org/W2115315740","https://openalex.org/W2111530399","https://openalex.org/W2137118400","https://openalex.org/W2152854510","https://openalex.org/W2104715506","https://openalex.org/W2158613743","https://openalex.org/W7220611047","https://openalex.org/W7132480616","https://openalex.org/W3176147046","https://openalex.org/W2062462877"],"abstract_inverted_index":{"As":[0],"HTS":[1],"technologies":[2],"come":[3],"of":[4,14,84],"age,":[5],"pharmaceutical":[6],"companies":[7],"are":[8,28,51,58],"focusing":[9],"increasingly":[10],"on":[11,23],"the":[12],"quality":[13],"their":[15,21],"screening":[16],"collections.":[17],"Storage":[18],"conditions":[19],"and":[20,26,73,76],"influence":[22],"compound":[24],"stability":[25],"solubility":[27],"debated":[29],"intensely.":[30],"At":[31],"Novartis,":[32],"a":[33,66],"strategy":[34],"was":[35],"developed":[36],"that":[37],"is":[38],"different":[39],"to":[40,69,77],"most":[41],"other":[42],"companies:":[43],"(1)":[44],"compounds":[45,57,85],"unsuitable":[46],"for":[47],"storage":[48,92],"in":[49,65],"solution":[50,97,101],"excluded":[52],"by":[53],"computational":[54],"methods;":[55],"(2)":[56],"stored":[59],"at":[60,86],"4":[61],"C/20%":[62],"relative":[63],"humidity":[64],"DMSO/water":[67],"mixture":[68],"avoid":[70],"freeze-thaw":[71],"cycles":[72],"water":[74],"uptake":[75],"allow":[78],"rapid":[79],"plate":[80],"replication;":[81],"(3)":[82],"resolubilisation":[83],"regular":[87],"intervals.":[88],"Keywords:":[89],"Compound":[90],"management,":[91,100],"conditions,":[93],"automated":[94,96],"weighing,":[95],"production,":[98],"lifecycle":[99],"archive":[102]},"counts_by_year":[{"year":2026,"cited_by_count":1},{"year":2024,"cited_by_count":1},{"year":2020,"cited_by_count":2},{"year":2018,"cited_by_count":1},{"year":2016,"cited_by_count":3},{"year":2012,"cited_by_count":6}],"updated_date":"2026-11-04T10:54:05.112534","created_date":"2016-06-24T00:00:00"}
